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Targeting the human Dihydroorotate Dehydrogenase (hDHODH) by combination of in-silico ligand/structural pharmacophore models and scaffold hopping bioisosteric approaches 2015 Mensa, Stefano; Carnovale, Irene M.; Pippione, Agnese Chiara; Sainas, Stefano; Giorgis, Marta; Piccinini, Marco; Lupino, Elisa; Al-Karadaghi, Salam; Boschi, Donatella; L. Lolli., Marco
Targeting the human Dihydroorotate Dehydrogenase (hDHODH) by a Scaffold Hopping Bioisosteric approach using Hydroxylated Pentaatomic Heterocycles 2016 Sainas, Stefano; Pippione, Agnese Chiara; Carnovale, IRENE MARIA; Giraudo, Alessandro; Giorgis, Marta; Braga Rodolpho Campos, ; Andrade Carolina Horta, ; Piccinini, Marco; Lupino, Elisa; Guedes, Rita; AL KARADAGHI, Salam; Boschi, Donatella; Lolli, Marco Lucio
NEW HYDROXYAZOLES INHIBITORS OF ALDO-KETO REDUCTASE 1C3 (AKR1C3) OBTAINED BY SCAFFOLD HOPPING FROM FLUFENAMIC ACID AND INDOMETHACIN FOR CASTRATE RESISTANT PROSTATE CANCER 2016 Boschi, Donatella; Pippione, Agnese Chiara; Giraudo, Alessandro; Carnovale, Irene Maria; Zorniotti, Sonia; Oliaro-Bosso, Simonetta; Ferrante, Terenzio; Marini, Elisabetta; Pors, Klaus; Festuccia, Claudio; Monache, Simona Delle; Zaffaroni, Nadia; Braga, Rodolpho Campos; Lucio, Marco; Lolli,
Targeting the human Dihydroorotate Dehydrogenase (hDHODH) by a Scaffold Hopping Bioisosteric approach using Hydroxylated Pentatomic Heterocycles 2016 Stefano Sainas, Agnese Chiara Pippione, Irene Maria Carnovale, Alessandro Giraudo, Marta Giorgis, Rodolpho B. Braga, Carolina H. Andrade, Noemi Villella, Marco Piccinini, Elisa Lupino, Rosmarie Friemann, Salam Al-Kadaraghi, Donatella Boschi, Marco L. Lolli
Targeting Castration Resistant Prostate Cancer (CRPC) by innovative AKR1C3 inhibitors based on the 3-hydroxybenzoisoxazole structure 2016 Carnovale, Irene Maria; Pippione, Agnese Chiara; Giraudo, Alessandro; Federico, Antonella; Zorniotti, Sonia; Simonetta Oliaro Bosso, ; Ferrante, Terenzio; Marini, Elisabetta; Pors, Klaus; Braga, Rodolpho Campos; Boschi, Donatella; Lucio Lolli, Marco
NEW HYDROXYAZOLES INHIBITORS OF AKR1C3 OBTAINED FROM NSAIDS BY SCAFFOLD HOPPING APPROACH AGAINST CASTRATE RESISTANT PROSTATE CANCER 2016 Boschi, Donatella; Pippione, Agnese Chiara; Giraudo, Alessandro; Carnovale, Irene Maria; Zorniotti, Sonia; Oliaro-Bosso, Simonetta; Ferrante, Terenzio; Marini, Elisabetta; Pors, Klaus; Festuccia, Claudio; Monache, Simona Delle; Zaffaroni, Nadia; Braga, Rodolpho Campos; Lucio Lolli, Marco
Targeting the human Dihydroorotate Dehydrogenase (hDHODH) by a Scaffold Hopping Bioisosteric approach using Hydroxylated Pentatomic Heterocycles 2016 Sainas Stefano; Pippione Agnese Chiara; Carnovale Irene Maria; Giraudo Alessandro; Giorgis Marta; de Campos Braga Rodolpho; Andrade Carolina H; Villella Noemi; Friemann Rosmarie; Piccinini Marco; Lupino Elisa; Al-karadaghi Salam; Boschi Donatella;Lolli Marco Lucio
Synthesis of new gadolinium complexes for magnetic resonance imaging with improved relaxivity 2017 Irene Maria Carnovale, ; Sonia Colombo Serra, ; Alberto Fringuello Mingo, ; Luciano, Lattuada; Marco Lucio Lolli,
Synthesis of new gadolinium complexes for magnetic resonance imaging with improved relaxivity 2017 Carnovale, I. M.; Colombo Serra, S.; Fringuello Mingo, A.; Lattuada, L.; Lolli, M. L.
Synthesis of new Gadolinium complexes for magnetic resonance imaging with improved relaxivity 2017 Carnovale, Irene Maria; Serra, Sonia Colombo; Fringuello Mingo, Alberto; Lattuada, Luciano; Lolli, Marco Lucio
Macrocyclic paramagnetic agents for MRI: Determinants of relaxivity and strategies for their improvement 2017 Fringuello Mingo, Alberto; Colombo Serra, Sonia; Baroni, Simona; Cabella, Claudia; Napolitano, Roberta; Hawala, Ivan; Carnovale, Irene Maria; Lattuada, Luciano; Tedoldi, Fabio; Aime, Silvio
Hydroxytriazole derivatives as potent and selective aldo-keto reductase 1C3 (AKR1C3) inhibitors discovered by bioisosteric scaffold hopping approach 2017 Pippione, Agnese C.; Giraudo, Alessandro; Bonanni, Davide; Carnovale, Irene M.; Marini, Elisabetta; Cena, Clara; Costale, Annalisa; Zonari, Daniele; Pors, Klaus; Sadiq, Maria; Boschi, Donatella; Oliaro-Bosso, Simonetta; Lolli, Marco L
Exploring the intramolecular catalysis of the proton exchange process to modulate the relaxivity of Gd(iii)-complexes of HP-DO3A-like ligands 2018 Carnovale, Irene Maria; Lolli, Marco Lucio; Serra, Sonia Colombo; Mingo, Alberto Fringuello; Napolitano, Roberta; Boi, Valeria; Guidolin, Nicol; Lattuada, Luciano; Tedoldi, Fabio; Baranyai, Zsolt; Aime, Silvio
Potent and selective aldo-keto reductase 1C3 (AKR1C3) inhibitors based on the benzoisoxazole moiety: Application of a bioisosteric scaffold hopping approach to flufenamic acid 2018 Pippione, Agnese Chiara; Carnovale, Irene Maria; Bonanni, Davide; Sini, Marcella; Goyal, Parveen; Marini, Elisabetta; Pors, Klaus; Adinolfi, Salvatore; Zonari, Daniele; Festuccia, Claudio; Wahlgren, Weixiao Yuan; Friemann, Rosmarie; Bagnati, Renzo; Boschi, Donatella; Oliaro-Bosso, Simonetta; Lolli, Marco Lucio
Bioisosteres of Indomethacin as Inhibitors of Aldo-Keto Reductase 1C3 2019 Lolli, Marco L; Carnovale, Irene M; Pippione, Agnese C; Wahlgren, Weixiao Y; Bonanni, Davide; Marini, Elisabetta; Zonari, Daniele; Gallicchio, Margherita; Boscaro, Valentina; Goyal, Parveen; Friemann, Rosmarie; Rolando, Barbara; Bagnati, Renzo; Adinolfi, Salvatore; Oliaro-Bosso, Simonetta; Boschi, Donatella
H-Bonding and intramolecular catalysis of proton exchange affect the CEST properties of EuIIIcomplexes with HP-DO3A-like ligands 2021 Baroni S.; Carnovale I.M.; Carrera C.; Boccalon M.; Guidolin N.; Demitri N.; Lattuada L.; Tedoldi F.; Baranyai Z.; Aime S.
Mostrati risultati da 1 a 16 di 16
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