Sfoglia per Autore
SYNTHESIS OF AMODIAQUINE ANALOGUES WITH POTENTIAL ANTIPROTOZOAL ACTIVITY
2007-01-01 guglielmo s.
Furoxan-, alkylnitrate-derivatives and related compoundsas anti-trypanosomatid agents: Mechanism of action studies
2008-01-01 Lucia Boiani; Gabriela Aguirre; Mercedes González; Hugo Cerecetto; Agustina Chidichimo; Juan J. Cazzulo; Massimo Bertinaria; Stefano Guglielmo
Unsymmetrically Substituted Furoxans. Part 19. Methyl and Phenylfuroxansulfonic Acids and Related Sulfonamides
2009-01-01 Konstantin Chegaev; Barbara Rolando; Stefano Guglielmo; Roberta Fruttero; Alberto Gasco
A new series of amodiaquine analogues modified in the basic side chain with in vitro antileishmanial and antiplasmodial activity
2009-01-01 Stefano Guglielmo; Massimo Bertinaria; Barbara Rolando; Marco Crosetti; Roberta Fruttero; Vanessa Yardley; Simon L. Croft; Alberto Gasco
Phenylsulfonylfuroxans as Modulators of Multidrug-Resistance-Associated Protein-1 and P-Glycoprotein
2010-01-01 Roberta Fruttero; Marco Crosetti; Konstantin Chegaev; Stefano Guglielmo; Alberto Gasco; Francesco Berardi; Mauro Niso; Roberto Perrone; Maria Antonietta Panaro; Nicola Antonio Colabufo
PHENYLSULFONYL FUROXANS AS MODULATORS OF MULTIDRUGRESISTANCE-ASSOCIATED PROTEIN-1 AND P-GLYCOPROTEIN
2010-01-01 Fruttero R.; Crosetti M.; Chegaev K.; Guglielmo S.; Gasco A.; Berardi F.; Niso M.; Perrone R.; Panaro M. A.; Colabufo N. A.
Praziquantel analogues containing NO-donor furoxans and related furazans as agents active against Schistosoma mansoni.
2011-01-01 Francesca Vottero; Stefano Guglielmo; Roberta Fruttero; Alberto Gasco; Daniela Cortese; Latasha Day; Valerie Kommer; David L. Williams
Hybrid praziquantel-oxadiazole oxides with activity against Schistosoma mansoni.
2011-01-01 Daniela Cortese; Francesca Vottero; Stefano Guglielmo; Roberta Fruttero; Alberto Gasco; Latasha Day and David L. Williams.
Nitric Oxide Donor Doxorubicins Accumulate into Doxorubicin-Resistant Human Colon Cancer Cells Inducing Cytotoxicity
2011-01-01 Konstantin Chegaev; Chiara Riganti; Loretta Lazzarato; Barbara Rolando; Stefano Guglielmo; Ivana Campia; Roberta Fruttero; Amalia Bosia; Alberto Gasco
New nitric oxide or hydrogen sulfide releasing aspirins
2011-01-01 Loretta Lazzarato; Konstantin Chegaev; Elisabetta Marini; Barbara Rolando; Emily Borretto; Stefano Guglielmo; Sony Joseph; Antonella Di Stilo; Roberta Fruttero; Alberto Gasco
Searching for new NO-donor aspirin-like molecules: furoxanylacyl derivatives of salicylic acid and related furazans
2011-01-01 Lazzarato Loretta; Cena Clara; Barbara Rolando; Elisabetta Marini; Marco Lucio Lolli; Guglielmo Stefano; Elena Guaita; Giuseppina Morini; Gabriella Coruzzi; Roberta Fruttero; Alberto Gasco
Synthesis and in vitro antimicrobial activities of new (cyano-NNO-azoxy)pyrazole derivatives
2011-01-01 Boschi, D.; Guglielmo, S.; Aiello, S.; Morace, G.; Borghi, E.; Fruttero, R.
Amodiaquine analogues containing NO-donor substructures: Synthesis and their preliminary evaluation as potential tools in the treatment of cerebral malaria
2011-01-01 Massimo Bertinaria; Stefano Guglielmo; Barbara Rolando; Marta Giorgis; Cristina Aragno; Roberta Fruttero; Alberto Gasco; Silvia Parapini; Donatella Taramelli; Yuri C. Martins; Leonardo J.M. Carvalho
Synthesis, physico-chemical characterization, andbiological activities of new carnosine derivatives stablein human serum as potential neuroprotective agents
2011-01-01 Massimo Bertinaria; Barbara Rolando; Marta Giorgis; Gabriele Montanaro; Stefano Guglielmo; M. Federica Buonsanti; Valentina Carabelli; Daniela Gavello; Pier Giuseppe Daniele; Roberta Fruttero; Alberto Gasco
Synthesis and preliminary biological profile of new NO-donor tolbutamide analogues.
2012-01-01 Yasinalli Tamboli; Loretta Lazzarato; Elisabetta Marini; Stefano Guglielmo; Michela Novelli; Pascale Beffy; Pellegrino Masiello; Roberta Fruttero; Alberto Gasco
Thymopentin down-regulates both activity and expression of iNOS in blood cells of Sézary syndrome patients
2012-01-01 Patruno A.; Tosco P.; Borretto E.; Franceschelli S.; Amerio P.; Pesce M.; Guglielmo S.; Campiglia P.; Bernengo M. G.; Fruttero R.
Praziquantel analogues containing NO-donor furoxans and related furazans as agents active against Schistosoma mansoni.
2013-01-01 Daniela Cortese; Stefano Guglielmo; Francesca Vottero; Valerie. P. Kommer; David L. Williams; Roberta Fruttero; Alberto Gasco.
Tandem Mass Spectrometry of Nitric Oxide and Hydrogen Sulfide Releasing Aspirins: A Hint into Activity Behavior
2013-01-01 Maria Elisa Crestoni; Barbara Chiavarino; Stefano Guglielmo; Valentina Lilla; Simonetta Fornarini
New potent and selective P-gp inhibitors
2013-01-01 Guglielmo S.; Bonomo S.; Colabufo N. A.; Contino M.; Perrone M. G.; Fruttero R.; Gasco A.
Doxorubicin-antioxidant multitarget drugs
2013-01-01 K Chegaev; C Riganti; B Rolando; L Lazzarato; E Gazzano; S Guglielmo; D Ghigo; R Fruttero; A Gasco
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
SYNTHESIS OF AMODIAQUINE ANALOGUES WITH POTENTIAL ANTIPROTOZOAL ACTIVITY | 2007 | guglielmo s. | |
Furoxan-, alkylnitrate-derivatives and related compoundsas anti-trypanosomatid agents: Mechanism of action studies | 2008 | Lucia Boiani; Gabriela Aguirre; Mercedes González; Hugo Cerecetto; Agustina Chidichimo; Juan J. Cazzulo; Massimo Bertinaria; Stefano Guglielmo | |
Unsymmetrically Substituted Furoxans. Part 19. Methyl and Phenylfuroxansulfonic Acids and Related Sulfonamides | 2009 | Konstantin Chegaev; Barbara Rolando; Stefano Guglielmo; Roberta Fruttero; Alberto Gasco | |
A new series of amodiaquine analogues modified in the basic side chain with in vitro antileishmanial and antiplasmodial activity | 2009 | Stefano Guglielmo; Massimo Bertinaria; Barbara Rolando; Marco Crosetti; Roberta Fruttero; Vanessa Yardley; Simon L. Croft; Alberto Gasco | |
Phenylsulfonylfuroxans as Modulators of Multidrug-Resistance-Associated Protein-1 and P-Glycoprotein | 2010 | Roberta Fruttero; Marco Crosetti; Konstantin Chegaev; Stefano Guglielmo; Alberto Gasco; Francesco Berardi; Mauro Niso; Roberto Perrone; Maria Antonietta Panaro; Nicola Antonio Colabufo | |
PHENYLSULFONYL FUROXANS AS MODULATORS OF MULTIDRUGRESISTANCE-ASSOCIATED PROTEIN-1 AND P-GLYCOPROTEIN | 2010 | Fruttero R.; Crosetti M.; Chegaev K.; Guglielmo S.; Gasco A.; Berardi F.; Niso M.; Perrone R.; Panaro M. A.; Colabufo N. A. | |
Praziquantel analogues containing NO-donor furoxans and related furazans as agents active against Schistosoma mansoni. | 2011 | Francesca Vottero; Stefano Guglielmo; Roberta Fruttero; Alberto Gasco; Daniela Cortese; Latasha Day; Valerie Kommer; David L. Williams | |
Hybrid praziquantel-oxadiazole oxides with activity against Schistosoma mansoni. | 2011 | Daniela Cortese; Francesca Vottero; Stefano Guglielmo; Roberta Fruttero; Alberto Gasco; Latasha Day and David L. Williams. | |
Nitric Oxide Donor Doxorubicins Accumulate into Doxorubicin-Resistant Human Colon Cancer Cells Inducing Cytotoxicity | 2011 | Konstantin Chegaev; Chiara Riganti; Loretta Lazzarato; Barbara Rolando; Stefano Guglielmo; Ivana Campia; Roberta Fruttero; Amalia Bosia; Alberto Gasco | |
New nitric oxide or hydrogen sulfide releasing aspirins | 2011 | Loretta Lazzarato; Konstantin Chegaev; Elisabetta Marini; Barbara Rolando; Emily Borretto; Stefano Guglielmo; Sony Joseph; Antonella Di Stilo; Roberta Fruttero; Alberto Gasco | |
Searching for new NO-donor aspirin-like molecules: furoxanylacyl derivatives of salicylic acid and related furazans | 2011 | Lazzarato Loretta; Cena Clara; Barbara Rolando; Elisabetta Marini; Marco Lucio Lolli; Guglielmo Stefano; Elena Guaita; Giuseppina Morini; Gabriella Coruzzi; Roberta Fruttero; Alberto Gasco | |
Synthesis and in vitro antimicrobial activities of new (cyano-NNO-azoxy)pyrazole derivatives | 2011 | Boschi, D.; Guglielmo, S.; Aiello, S.; Morace, G.; Borghi, E.; Fruttero, R. | |
Amodiaquine analogues containing NO-donor substructures: Synthesis and their preliminary evaluation as potential tools in the treatment of cerebral malaria | 2011 | Massimo Bertinaria; Stefano Guglielmo; Barbara Rolando; Marta Giorgis; Cristina Aragno; Roberta Fruttero; Alberto Gasco; Silvia Parapini; Donatella Taramelli; Yuri C. Martins; Leonardo J.M. Carvalho | |
Synthesis, physico-chemical characterization, andbiological activities of new carnosine derivatives stablein human serum as potential neuroprotective agents | 2011 | Massimo Bertinaria; Barbara Rolando; Marta Giorgis; Gabriele Montanaro; Stefano Guglielmo; M. Federica Buonsanti; Valentina Carabelli; Daniela Gavello; Pier Giuseppe Daniele; Roberta Fruttero; Alberto Gasco | |
Synthesis and preliminary biological profile of new NO-donor tolbutamide analogues. | 2012 | Yasinalli Tamboli; Loretta Lazzarato; Elisabetta Marini; Stefano Guglielmo; Michela Novelli; Pascale Beffy; Pellegrino Masiello; Roberta Fruttero; Alberto Gasco | |
Thymopentin down-regulates both activity and expression of iNOS in blood cells of Sézary syndrome patients | 2012 | Patruno A.; Tosco P.; Borretto E.; Franceschelli S.; Amerio P.; Pesce M.; Guglielmo S.; Campiglia P.; Bernengo M. G.; Fruttero R. | |
Praziquantel analogues containing NO-donor furoxans and related furazans as agents active against Schistosoma mansoni. | 2013 | Daniela Cortese; Stefano Guglielmo; Francesca Vottero; Valerie. P. Kommer; David L. Williams; Roberta Fruttero; Alberto Gasco. | |
Tandem Mass Spectrometry of Nitric Oxide and Hydrogen Sulfide Releasing Aspirins: A Hint into Activity Behavior | 2013 | Maria Elisa Crestoni; Barbara Chiavarino; Stefano Guglielmo; Valentina Lilla; Simonetta Fornarini | |
New potent and selective P-gp inhibitors | 2013 | Guglielmo S.; Bonomo S.; Colabufo N. A.; Contino M.; Perrone M. G.; Fruttero R.; Gasco A. | |
Doxorubicin-antioxidant multitarget drugs | 2013 | K Chegaev; C Riganti; B Rolando; L Lazzarato; E Gazzano; S Guglielmo; D Ghigo; R Fruttero; A Gasco |
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