Sfoglia per Autore
Unsymmetrically substituted furoxans. Part 16 [1]. Reaction of benzenesulfonyl substituted furoxans with ethanol and ethanethiol in basic medium
1996-01-01 G. Sorba; G. Ermondi; R. Fruttero; U. Galli; A. Gasco
WATER SOLUBLE FUROXAN DERIVATIVES AS NO PRODRUGS
1997-01-01 G. SORBA; C. MEDANA; R. FRUTTERO; C. CENA; A. DI STILO; U. GALLI; A. GASCO
Identification of 2,3-diaminophenazine and of o-benzoquinone dioxime as the major in vitro metabolites of benzofuroxan
2004-01-01 G. GROSA; U. GALLI; B. ROLANDO; R. FRUTTERO; G. GERVASIO; A. GASCO
Synthesis and antimalarial activities of some furoxan sulfones and related furazans
2005-01-01 U. GALLI; L. LAZZARATO; M. BERTINARIA; G. SORBA; A. GASCO; S. PARAPINI; D. TARAMELLI
Design, Synthesis, and Biological Evaluation of New (2E,6E)-10-(Dimethylamino)-3,7-dimethyl-2,6-decadien-1-ol Ethers as Inhibitors of Human and Trypanosoma cruzi Oxidosqualene Cyclase.
2007-01-01 U. GALLI; S. OLIARO-BOSSO; S. TARAMINO; S. VENEGONI; E. PASTORE; GC. TRON; G. BALLIANO; F. VIOLA; G. SORBA
Replacement of the lactone moiety on podophyllotoxin and steganacin analogues with a 1,5-disubstituted 1,2,3-triazole via ruthenium-catalyzed click chemistry
2007-01-01 IMPERIO, DANIELA; PIRALI, Tracey; GALLI, Ubaldina; PAGLIAI, Francesca; Cafici L; CANONICO, Pier Luigi; SORBA, Giovanni; GENAZZANI, Armando; TRON, Gian Cesare
Synthesis and biological evaluation of isosteric analogues of FK866, an inhibitor of NAD salvage
2008-01-01 GALLI, Ubaldina; ERCOLANO, EMANUELA; CARRARO, Lorenzo Roberto; Blasi Roman CR; SORBA, Giovanni; CANONICO, Pier Luigi; GENAZZANI, Armando; TRON, Gian Cesare; BILLINGTON, Richard Andrew
Characterization of NAD uptake in mammalian cells
2008-01-01 BILLINGTON, Richard Andrew; TRAVELLI, Cristina; ERCOLANO, EMANUELA; GALLI, Ubaldina; Roman CB; GROLLA, AMBRA; CANONICO, Pier Luigi; CONDORELLI, Fabrizio; GENAZZANI, Armando
A novel potent nicotinamide phosphoribosyltransferase inhibitor synthesized via click chemistry
2010-01-01 COLOMBANO, GIAMPIERO; TRAVELLI, Cristina; GALLI, Ubaldina; CALDARELLI, ANTONIO; Chini MG; CANONICO, Pier Luigi; SORBA, Giovanni; Bifulco G; TRON, Gian Cesare; GENAZZANI, Armando
Reciprocal potentiation of the antitumoral activities of FK866, an inhibitor of nicotinamide phosphoribosyltransferase, and etoposide or cisplatin in neuroblastoma cells
2011-01-01 TRAVELLI, Cristina; DRAGO, VALENTINA; Maldi E; Kaludercic N; GALLI, Ubaldina; BOLDORINI, Renzo Luciano; Di Lisa F; TRON, Gian Cesare; CANONICO, Pier Luigi; GENAZZANI, Armando
QUINOLIN-4 (1H) -ONE DERIVATIVES AS INHIBITORS OF PHOSPHATIDYLINOSITOL 3-KINASES
2012-01-01 Giovanni Sorba; Gian Cesare Tron; Tracey Pirali; Ubaldina Galli; Alberto Massarotti; Emilio Hirsch; Elisa Ciraolo
Identification of a sirtuin 3 inhibitor that displays selectivity over sirtuin 1 and 2
2012-01-01 GALLI, Ubaldina; MESENZANI, Ornella; Coppo C; SORBA, Giovanni; CANONICO, Pier Luigi; TRON, Gian Cesare; GENAZZANI, Armando
Nicotinamide phosphoribosyltransferase (NAMPT) is over-expressed in melanoma lesions
2013-01-01 Maldi E; TRAVELLI, Cristina; CALDARELLI, ANTONIO; Agazzone N; Cintura S; GALLI, Ubaldina; Scatolini M; Ostano P; Miglino B; Chiorino G; BOLDORINI, Renzo Luciano; GENAZZANI, Armando
Medicinal chemistry of nicotinamide phosphoribosyltransferase (NAMPT) inhibitors
2013-01-01 GALLI, Ubaldina; TRAVELLI, Cristina; MASSAROTTI, Alberto; Fakhfouri, G; Rahimian, R; TRON, Gian Cesare; GENAZZANI, Armando
Design, synthesis, and biological evaluation of combretabenzodiazepines: a novel class of anti-tubulin agents
2015-01-01 GALLI, Ubaldina; TRAVELLI, Cristina; APRILE, SILVIO; Arrigoni, Elena; TORRETTA, SIMONE; GROSA, Giorgio; MASSAROTTI, Alberto; SORBA, Giovanni; CANONICO, Pier Luigi; GENAZZANI, Armando; TRON, Gian Cesare
Identification of a novel NAMPT inhibitor by combinatorial click chemistry and chemical refinement
2015-01-01 Theeramunkong, S.; GALLI, Ubaldina; GROLLA, AMBRA; CALDARELLI, ANTONIO; TRAVELLI, Cristina; MASSAROTTI, Alberto; Troiani, M. P.; Alisi, M. A.; Orsomando, G.; GENAZZANI, Armando; TRON, Gian Cesare
Identification of Novel Triazole-Based Nicotinamide Phosphoribosyltransferase (NAMPT) Inhibitors Endowed with Antiproliferative and Antiinflammatory Activity
2017-01-01 TRAVELLI, Cristina; APRILE, SILVIO; Rahimian, Reza; Grolla, Ambra A.; ROGATI, FEDERICA; Bertolotti, Mattia; Malagnino, Floriana; Di Paola, Rosanna; Impellizzeri, Daniela; FUSCO, Roberta; MERCALLI, VALENTINA; MASSAROTTI, Alberto; Stortini, Giorgio; TERRAZZINO, SALVATORE; DEL GROSSO, Erika; Fakhfouri, Gohar; Troiani, Maria Pia; Alisi, Maria Alessandra; GROSA, Giorgio; SORBA, Giovanni; CANONICO, Pier Luigi; Orsomando, Giuseppe; Cuzzocrea, Salvatore; GENAZZANI, Armando; GALLI, Ubaldina; TRON, Gian Cesare
Pyrtriazoles, a Novel Class of Store-Operated Calcium Entry Modulators: Discovery, Biological Profiling, and in Vivo Proof-of-Concept Efficacy in Acute Pancreatitis
2018-01-01 Riva, Beatrice; Griglio, Alessia; Serafini, Marta; CORDERO SANCHEZ, CELIA; Aprile, Silvio; Di Paola, Rosanna; Gugliandolo, Enrico; Alansary, Dalia; BIOCOTINO, Isabella; Lim, Dmitry; Grosa, Giorgio; Galli, Ubaldina; Niemeyer, Barbara; Sorba, Giovanni; Canonico, Pier Luigi; Cuzzocrea, Salvatore; Genazzani, Armando; Pirali, Tracey
Drug Discovery for Soft Drugs on TRPV1 and TRPM8 Channels Using the Passerini Reaction
2019-01-01 Pirali, Tracey; Galli, Ubaldina; Serafini, Marta; Griglio, Alessia; Genazzani, Armando; Tron, Gian Cesare
Identification of potent triazolylpyridine nicotinamide phosphoribosyltransferase (NAMPT) inhibitors bearing a 1,2,3-triazole tail group
2019-01-01 Travelli, Cristina; Aprile, Silvio; Mattoteia, Daiana; Colombo, Giorgia; Clemente, Nausicaa; Scanziani, Eugenio; Terrazzino, Salvatore; Alisi, Maria Alessandra; Polenzani, Lorenzo; Grosa, Giorgio; Genazzani, Armando; Tron, Gian Cesare; Galli, Ubaldina
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
Unsymmetrically substituted furoxans. Part 16 [1]. Reaction of benzenesulfonyl substituted furoxans with ethanol and ethanethiol in basic medium | 1996 | G. Sorba; G. Ermondi; R. Fruttero; U. Galli; A. Gasco | |
WATER SOLUBLE FUROXAN DERIVATIVES AS NO PRODRUGS | 1997 | G. SORBA; C. MEDANA; R. FRUTTERO; C. CENA; A. DI STILO; U. GALLI; A. GASCO | |
Identification of 2,3-diaminophenazine and of o-benzoquinone dioxime as the major in vitro metabolites of benzofuroxan | 2004 | G. GROSA; U. GALLI; B. ROLANDO; R. FRUTTERO; G. GERVASIO; A. GASCO | |
Synthesis and antimalarial activities of some furoxan sulfones and related furazans | 2005 | U. GALLI; L. LAZZARATO; M. BERTINARIA; G. SORBA; A. GASCO; S. PARAPINI; D. TARAMELLI | |
Design, Synthesis, and Biological Evaluation of New (2E,6E)-10-(Dimethylamino)-3,7-dimethyl-2,6-decadien-1-ol Ethers as Inhibitors of Human and Trypanosoma cruzi Oxidosqualene Cyclase. | 2007 | U. GALLI; S. OLIARO-BOSSO; S. TARAMINO; S. VENEGONI; E. PASTORE; GC. TRON; G. BALLIANO; F. VIOLA; G. SORBA | |
Replacement of the lactone moiety on podophyllotoxin and steganacin analogues with a 1,5-disubstituted 1,2,3-triazole via ruthenium-catalyzed click chemistry | 2007 | IMPERIO, DANIELA; PIRALI, Tracey; GALLI, Ubaldina; PAGLIAI, Francesca; Cafici L; CANONICO, Pier Luigi; SORBA, Giovanni; GENAZZANI, Armando; TRON, Gian Cesare | |
Synthesis and biological evaluation of isosteric analogues of FK866, an inhibitor of NAD salvage | 2008 | GALLI, Ubaldina; ERCOLANO, EMANUELA; CARRARO, Lorenzo Roberto; Blasi Roman CR; SORBA, Giovanni; CANONICO, Pier Luigi; GENAZZANI, Armando; TRON, Gian Cesare; BILLINGTON, Richard Andrew | |
Characterization of NAD uptake in mammalian cells | 2008 | BILLINGTON, Richard Andrew; TRAVELLI, Cristina; ERCOLANO, EMANUELA; GALLI, Ubaldina; Roman CB; GROLLA, AMBRA; CANONICO, Pier Luigi; CONDORELLI, Fabrizio; GENAZZANI, Armando | |
A novel potent nicotinamide phosphoribosyltransferase inhibitor synthesized via click chemistry | 2010 | COLOMBANO, GIAMPIERO; TRAVELLI, Cristina; GALLI, Ubaldina; CALDARELLI, ANTONIO; Chini MG; CANONICO, Pier Luigi; SORBA, Giovanni; Bifulco G; TRON, Gian Cesare; GENAZZANI, Armando | |
Reciprocal potentiation of the antitumoral activities of FK866, an inhibitor of nicotinamide phosphoribosyltransferase, and etoposide or cisplatin in neuroblastoma cells | 2011 | TRAVELLI, Cristina; DRAGO, VALENTINA; Maldi E; Kaludercic N; GALLI, Ubaldina; BOLDORINI, Renzo Luciano; Di Lisa F; TRON, Gian Cesare; CANONICO, Pier Luigi; GENAZZANI, Armando | |
QUINOLIN-4 (1H) -ONE DERIVATIVES AS INHIBITORS OF PHOSPHATIDYLINOSITOL 3-KINASES | 2012 | Giovanni Sorba; Gian Cesare Tron; Tracey Pirali; Ubaldina Galli; Alberto Massarotti; Emilio Hirsch; Elisa Ciraolo | |
Identification of a sirtuin 3 inhibitor that displays selectivity over sirtuin 1 and 2 | 2012 | GALLI, Ubaldina; MESENZANI, Ornella; Coppo C; SORBA, Giovanni; CANONICO, Pier Luigi; TRON, Gian Cesare; GENAZZANI, Armando | |
Nicotinamide phosphoribosyltransferase (NAMPT) is over-expressed in melanoma lesions | 2013 | Maldi E; TRAVELLI, Cristina; CALDARELLI, ANTONIO; Agazzone N; Cintura S; GALLI, Ubaldina; Scatolini M; Ostano P; Miglino B; Chiorino G; BOLDORINI, Renzo Luciano; GENAZZANI, Armando | |
Medicinal chemistry of nicotinamide phosphoribosyltransferase (NAMPT) inhibitors | 2013 | GALLI, Ubaldina; TRAVELLI, Cristina; MASSAROTTI, Alberto; Fakhfouri, G; Rahimian, R; TRON, Gian Cesare; GENAZZANI, Armando | |
Design, synthesis, and biological evaluation of combretabenzodiazepines: a novel class of anti-tubulin agents | 2015 | GALLI, Ubaldina; TRAVELLI, Cristina; APRILE, SILVIO; Arrigoni, Elena; TORRETTA, SIMONE; GROSA, Giorgio; MASSAROTTI, Alberto; SORBA, Giovanni; CANONICO, Pier Luigi; GENAZZANI, Armando; TRON, Gian Cesare | |
Identification of a novel NAMPT inhibitor by combinatorial click chemistry and chemical refinement | 2015 | Theeramunkong, S.; GALLI, Ubaldina; GROLLA, AMBRA; CALDARELLI, ANTONIO; TRAVELLI, Cristina; MASSAROTTI, Alberto; Troiani, M. P.; Alisi, M. A.; Orsomando, G.; GENAZZANI, Armando; TRON, Gian Cesare | |
Identification of Novel Triazole-Based Nicotinamide Phosphoribosyltransferase (NAMPT) Inhibitors Endowed with Antiproliferative and Antiinflammatory Activity | 2017 | TRAVELLI, Cristina; APRILE, SILVIO; Rahimian, Reza; Grolla, Ambra A.; ROGATI, FEDERICA; Bertolotti, Mattia; Malagnino, Floriana; Di Paola, Rosanna; Impellizzeri, Daniela; FUSCO, Roberta; MERCALLI, VALENTINA; MASSAROTTI, Alberto; Stortini, Giorgio; TERRAZZINO, SALVATORE; DEL GROSSO, Erika; Fakhfouri, Gohar; Troiani, Maria Pia; Alisi, Maria Alessandra; GROSA, Giorgio; SORBA, Giovanni; CANONICO, Pier Luigi; Orsomando, Giuseppe; Cuzzocrea, Salvatore; GENAZZANI, Armando; GALLI, Ubaldina; TRON, Gian Cesare | |
Pyrtriazoles, a Novel Class of Store-Operated Calcium Entry Modulators: Discovery, Biological Profiling, and in Vivo Proof-of-Concept Efficacy in Acute Pancreatitis | 2018 | Riva, Beatrice; Griglio, Alessia; Serafini, Marta; CORDERO SANCHEZ, CELIA; Aprile, Silvio; Di Paola, Rosanna; Gugliandolo, Enrico; Alansary, Dalia; BIOCOTINO, Isabella; Lim, Dmitry; Grosa, Giorgio; Galli, Ubaldina; Niemeyer, Barbara; Sorba, Giovanni; Canonico, Pier Luigi; Cuzzocrea, Salvatore; Genazzani, Armando; Pirali, Tracey | |
Drug Discovery for Soft Drugs on TRPV1 and TRPM8 Channels Using the Passerini Reaction | 2019 | Pirali, Tracey; Galli, Ubaldina; Serafini, Marta; Griglio, Alessia; Genazzani, Armando; Tron, Gian Cesare | |
Identification of potent triazolylpyridine nicotinamide phosphoribosyltransferase (NAMPT) inhibitors bearing a 1,2,3-triazole tail group | 2019 | Travelli, Cristina; Aprile, Silvio; Mattoteia, Daiana; Colombo, Giorgia; Clemente, Nausicaa; Scanziani, Eugenio; Terrazzino, Salvatore; Alisi, Maria Alessandra; Polenzani, Lorenzo; Grosa, Giorgio; Genazzani, Armando; Tron, Gian Cesare; Galli, Ubaldina |
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