Sfoglia per Autore
NO-Donor Cyanines As Potential Anti-Alzheimer Drugs
2011-01-01 Federico A.; Chegaev K.; Lazzarato L.; Marini E.; Fruttero R.; Gasco A.
CYANINE-NO DONORS AS POTENTIAL ANTI ALZHEIMER DRUGS
2012-01-01 Federico Antonella
The Multi Target Drug Approach in Alzheimer Disease Therapy
2012-01-01 Federico Antonella
Multitarget drugs: NO-donor doxorubicins
2012-01-01 Chegaev K.; Riganti C.; Rolando B.; Federico A.; Fruttero R.; Gasco A.
Nitrooxy-doxorubicin: A New Weapon Against Multidrug Resistance.
2013-01-01 Joanna Kopecka; Chiara Riganti; Barbara Rolando; Ivana Campia; Konstantin Chegaev; Loretta Lazzarato; Antonella Federico; Roberta Fruttero; Dario Ghigo
The multi-target drug approach in Alzheimer's disease therapy
2013-01-01 Antonella Federico
Mitochondrial-targeting nitrooxy-doxorubicin: a new approach to overcome drug resistance.
2013-01-01 Chiara Riganti; Barbara Rolando; Joanna Kopecka; Ivana Campia; Konstantin Chegaev; Loretta Lazzarato; Antonella Federico; Roberta Fruttero; Dario Ghigo
Synthesis of new Plasmodium Falciparum dihydroorotate dehydrogenase inhibitors through the application of an isosteric portfolio
2013-01-01 Pippione A. C.;1 Federico A.;1 Boschi D.;S.2 Lolli M. L.1
SUBSTITUTED 4-HYDROXY-1H-1,2,3-TRIAZOLES: SYNTHESIS AND BIOISOSTERIC APPLICATIONS
2014-01-01 Agnese C. Pippione; Antonella Federico; Stefano Sainas; Alex Ducime; Marco L. Lolli; Donatella Boschi
TOWARD A BIOISOSTERIC ALKAEST – APPLICATION TO THE BIOISOSTERIC MODULATION OF IMD-0354
2014-01-01 Marco L. Lolli; Alex Ducime; Antonella Federico; Agnese Chiara Pippione; Stefano Sainas; Alessandro Barge; Katia Martina; Donatella Boschi; Elisa Lupino; Marco Piccinini; Michael Kubbutat; Christoph Schächtele; Jean Marie Contreras; Christophe Morice; Joel Sussman; Yoav Peleg; Bjorn Walse; Salam Kadaraghi
Towards a Bioisosteric Alkaest: application to the bioisosteric modulation of IMD-0354
2014-01-01 Lolli Marco L.; Federico Antonella; Ducime Alex; Pippione Agnese; Sainas Stefano; Barge Alessandro; Martina Katia; Boschi Donatella; Lupino Elisa; Piccinini Marco; Kubbutat Michael; Contreras Jean Marie; Morice Christophe; Sussman Joel; Peleg Yoav; Walse Bjorn; Al-Kadaraghi Salam
Synthesis and Structural Characterization of Regio Substituted 4-Hydroxy-1H-1,2,3-triazols as Possible Tool in Bioisosteric Applications
2014-01-01 A Federico; S.Sainas; A. Ducime;K. Martina; F. Bosca; D. Boschi; M.L. Lolli.
4-Hydroxy-1H-1,2,3-Triazol-5-yl moiety as bioisoster of carboxylic group. Synthesis and pharmacological ionotropic glutamate receptors characterization of Glu analogues
2014-01-01 S. Sainas; A. Federico;C. Bertolotti; B. Nielsen; D. Boschi; B. Frølund and M. L. Lolli
APPLICATION OF THE ARACHNO™ TECHNOLOGY FOR THE PARALLEL SYNTHESIS OF A LIBRARY OF ASPIRIN ANALOGUES
2015-01-01 Moreo, Angela; Barge, Alessandro; Boschi, Donatella; Costale, Annalisa; Dosio, Franco; Federico, Antonella; Stevanato, Livio; L. Lolli., Marco
NO-donor thiacarbocyanines as multifunctional agents for Alzheimer’s disease
2015-01-01 Chegaev, Konstantin; Federico, Antonella; Marini, Elisabetta; Rolando, Barbara; Fruttero, Roberta; Morbin, Michela; Rossi, Giacomina; Fugnanesi, Valeria; Bastone, Antonio; Salmona, Mario; Badiola, Nahuai B.; Gasparini, Laura; Cocco, Sara; Ripoli, Cristian; Grassi, Claudio; Gasco, Alberto
Substituted 4-hydroxy-1,2,3-triazoles: synthesis, characterization and first drug design applications through bioisosteric modulation and scaffold hopping approaches
2015-01-01 Pippione, Agnese C; Dosio, Franco; Ducime, Alex; Federico, Antonella; Martina, Katia; Sainas, Stefano; Frølund, Bente; Gooyit, Major; Janda, Kim D.; Boschi, Donatella; Lolli, Marco L.
Antileishmanial activity of some 4-phenyl-3-amino-1H-pyrazols designed as CRK3 kinase inhibitors
2016-01-01 Agnese Chiara Pippione, Piermichele Kobauri, Stefano Sainas, Alberto Gimenez, Antonella Federico, Rodolpho Campos Braga, Carolina Horta Andrade, Donatella Boschi, Efrain Salamanca, Juan Carlos Ticona, Marco Lucio Lolli
4-Hydroxy-N-[3,5-bis(trifluoromethyl)phenyl]-1,2,5-thiadiazole-3-carboxamide: a novel inhibitor of the canonical NF-κB cascade
2017-01-01 Pippione, Agnese C.; Federico, Antonella; Ducime, Alex; Sainas, Stefano; Boschi, Donatella; Barge, Alessandro; Lupino, Elisa; Piccinini, Marco; Kubbutat, Michael; Contreras, Jean-Marie; Morice, Christophe; Al-Karadaghi, Salam; Lolli, Marco L.
N-Acetyl-3-aminopyrazoles block the non canonical NF-kB cascade by selectively inhibiting NIK
2018-01-01 Agnese C. Pippione, Stefano Sainas, Antonella Federico, Elisa Lupino, Marco Piccinini, Michael Kubbutat, Jean-Marie Contreras, Christophe Morice, Alessandro Barge, Alex Ducime, Donatella Boschi, Salam Al-Karadaghi, Marco L. Lolli
Regioselective N‐Alkylation of Ethyl 4‐Benzyloxy‐1,2,3‐triazolecarboxylate: A Useful Tool for the Synthesis of Carboxylic Acid Bioisosteres
2019-01-01 Sainas, Stefano; Pippione, Agnese C.; Giraudo, Alessandro; Martina, Katia; Bosca, Federica; Rolando, Barbara; Barge, Alessandro; Ducime, Alex; Federico, Antonella; Grossert, Stuart J.; White, Robert L.; Boschi, Donatella; Lolli, Marco L.
| Titolo | Data di pubblicazione | Autore(i) | File |
|---|---|---|---|
| NO-Donor Cyanines As Potential Anti-Alzheimer Drugs | 2011 | Federico A.; Chegaev K.; Lazzarato L.; Marini E.; Fruttero R.; Gasco A. | |
| CYANINE-NO DONORS AS POTENTIAL ANTI ALZHEIMER DRUGS | 2012 | Federico Antonella | |
| The Multi Target Drug Approach in Alzheimer Disease Therapy | 2012 | Federico Antonella | |
| Multitarget drugs: NO-donor doxorubicins | 2012 | Chegaev K.; Riganti C.; Rolando B.; Federico A.; Fruttero R.; Gasco A. | |
| Nitrooxy-doxorubicin: A New Weapon Against Multidrug Resistance. | 2013 | Joanna Kopecka; Chiara Riganti; Barbara Rolando; Ivana Campia; Konstantin Chegaev; Loretta Lazzarato; Antonella Federico; Roberta Fruttero; Dario Ghigo | |
| The multi-target drug approach in Alzheimer's disease therapy | 2013 | Antonella Federico | |
| Mitochondrial-targeting nitrooxy-doxorubicin: a new approach to overcome drug resistance. | 2013 | Chiara Riganti; Barbara Rolando; Joanna Kopecka; Ivana Campia; Konstantin Chegaev; Loretta Lazzarato; Antonella Federico; Roberta Fruttero; Dario Ghigo | |
| Synthesis of new Plasmodium Falciparum dihydroorotate dehydrogenase inhibitors through the application of an isosteric portfolio | 2013 | Pippione A. C.;1 Federico A.;1 Boschi D.;S.2 Lolli M. L.1 | |
| SUBSTITUTED 4-HYDROXY-1H-1,2,3-TRIAZOLES: SYNTHESIS AND BIOISOSTERIC APPLICATIONS | 2014 | Agnese C. Pippione; Antonella Federico; Stefano Sainas; Alex Ducime; Marco L. Lolli; Donatella Boschi | |
| TOWARD A BIOISOSTERIC ALKAEST – APPLICATION TO THE BIOISOSTERIC MODULATION OF IMD-0354 | 2014 | Marco L. Lolli; Alex Ducime; Antonella Federico; Agnese Chiara Pippione; Stefano Sainas; Alessandro Barge; Katia Martina; Donatella Boschi; Elisa Lupino; Marco Piccinini; Michael Kubbutat; Christoph Schächtele; Jean Marie Contreras; Christophe Morice; Joel Sussman; Yoav Peleg; Bjorn Walse; Salam Kadaraghi | |
| Towards a Bioisosteric Alkaest: application to the bioisosteric modulation of IMD-0354 | 2014 | Lolli Marco L.; Federico Antonella; Ducime Alex; Pippione Agnese; Sainas Stefano; Barge Alessandro; Martina Katia; Boschi Donatella; Lupino Elisa; Piccinini Marco; Kubbutat Michael; Contreras Jean Marie; Morice Christophe; Sussman Joel; Peleg Yoav; Walse Bjorn; Al-Kadaraghi Salam | |
| Synthesis and Structural Characterization of Regio Substituted 4-Hydroxy-1H-1,2,3-triazols as Possible Tool in Bioisosteric Applications | 2014 | A Federico; S.Sainas; A. Ducime;K. Martina; F. Bosca; D. Boschi; M.L. Lolli. | |
| 4-Hydroxy-1H-1,2,3-Triazol-5-yl moiety as bioisoster of carboxylic group. Synthesis and pharmacological ionotropic glutamate receptors characterization of Glu analogues | 2014 | S. Sainas; A. Federico;C. Bertolotti; B. Nielsen; D. Boschi; B. Frølund and M. L. Lolli | |
| APPLICATION OF THE ARACHNO™ TECHNOLOGY FOR THE PARALLEL SYNTHESIS OF A LIBRARY OF ASPIRIN ANALOGUES | 2015 | Moreo, Angela; Barge, Alessandro; Boschi, Donatella; Costale, Annalisa; Dosio, Franco; Federico, Antonella; Stevanato, Livio; L. Lolli., Marco | |
| NO-donor thiacarbocyanines as multifunctional agents for Alzheimer’s disease | 2015 | Chegaev, Konstantin; Federico, Antonella; Marini, Elisabetta; Rolando, Barbara; Fruttero, Roberta; Morbin, Michela; Rossi, Giacomina; Fugnanesi, Valeria; Bastone, Antonio; Salmona, Mario; Badiola, Nahuai B.; Gasparini, Laura; Cocco, Sara; Ripoli, Cristian; Grassi, Claudio; Gasco, Alberto | |
| Substituted 4-hydroxy-1,2,3-triazoles: synthesis, characterization and first drug design applications through bioisosteric modulation and scaffold hopping approaches | 2015 | Pippione, Agnese C; Dosio, Franco; Ducime, Alex; Federico, Antonella; Martina, Katia; Sainas, Stefano; Frølund, Bente; Gooyit, Major; Janda, Kim D.; Boschi, Donatella; Lolli, Marco L. | |
| Antileishmanial activity of some 4-phenyl-3-amino-1H-pyrazols designed as CRK3 kinase inhibitors | 2016 | Agnese Chiara Pippione, Piermichele Kobauri, Stefano Sainas, Alberto Gimenez, Antonella Federico, Rodolpho Campos Braga, Carolina Horta Andrade, Donatella Boschi, Efrain Salamanca, Juan Carlos Ticona, Marco Lucio Lolli | |
| 4-Hydroxy-N-[3,5-bis(trifluoromethyl)phenyl]-1,2,5-thiadiazole-3-carboxamide: a novel inhibitor of the canonical NF-κB cascade | 2017 | Pippione, Agnese C.; Federico, Antonella; Ducime, Alex; Sainas, Stefano; Boschi, Donatella; Barge, Alessandro; Lupino, Elisa; Piccinini, Marco; Kubbutat, Michael; Contreras, Jean-Marie; Morice, Christophe; Al-Karadaghi, Salam; Lolli, Marco L. | |
| N-Acetyl-3-aminopyrazoles block the non canonical NF-kB cascade by selectively inhibiting NIK | 2018 | Agnese C. Pippione, Stefano Sainas, Antonella Federico, Elisa Lupino, Marco Piccinini, Michael Kubbutat, Jean-Marie Contreras, Christophe Morice, Alessandro Barge, Alex Ducime, Donatella Boschi, Salam Al-Karadaghi, Marco L. Lolli | |
| Regioselective N‐Alkylation of Ethyl 4‐Benzyloxy‐1,2,3‐triazolecarboxylate: A Useful Tool for the Synthesis of Carboxylic Acid Bioisosteres | 2019 | Sainas, Stefano; Pippione, Agnese C.; Giraudo, Alessandro; Martina, Katia; Bosca, Federica; Rolando, Barbara; Barge, Alessandro; Ducime, Alex; Federico, Antonella; Grossert, Stuart J.; White, Robert L.; Boschi, Donatella; Lolli, Marco L. |
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