Sfoglia per Autore
Icilio Guareschi and his amazing “1897 reaction”
2021-01-01 Tron, Gian Cesare; Minassi, Alberto; Sorba, Giovanni; Fausone, Mara; Appendino, Giovanni
Targeting Transient Receptor Potential Vanilloid 1 (TRPV1) Channel Softly: The Discovery of Passerini Adducts as a Topical Treatment for Inflammatory Skin Disorders
2018-01-01 Serafini, Marta; Griglio, Alessia; Aprile, Silvio; Seiti, Fabio; Travelli, Cristina; Pattarino, Franco; Grosa, Giorgio; Sorba, Giovanni; Genazzani, Armando; Gonzalez-Rodriguez, Sara; Butron, Laura; Devesa, Isabel; Fernandez-Carvajal, Asia; Pirali, Tracey; Ferrer-Montiel, Antonio
Pyrtriazoles, a Novel Class of Store-Operated Calcium Entry Modulators: Discovery, Biological Profiling, and in Vivo Proof-of-Concept Efficacy in Acute Pancreatitis
2018-01-01 Riva, Beatrice; Griglio, Alessia; Serafini, Marta; CORDERO SANCHEZ, CELIA; Aprile, Silvio; Di Paola, Rosanna; Gugliandolo, Enrico; Alansary, Dalia; BIOCOTINO, Isabella; Lim, Dmitry; Grosa, Giorgio; Galli, Ubaldina; Niemeyer, Barbara; Sorba, Giovanni; Canonico, Pier Luigi; Cuzzocrea, Salvatore; Genazzani, Armando; Pirali, Tracey
Identification of Novel Triazole-Based Nicotinamide Phosphoribosyltransferase (NAMPT) Inhibitors Endowed with Antiproliferative and Antiinflammatory Activity
2017-01-01 TRAVELLI, Cristina; APRILE, SILVIO; Rahimian, Reza; Grolla, Ambra A.; ROGATI, FEDERICA; Bertolotti, Mattia; Malagnino, Floriana; Di Paola, Rosanna; Impellizzeri, Daniela; FUSCO, Roberta; MERCALLI, VALENTINA; MASSAROTTI, Alberto; Stortini, Giorgio; TERRAZZINO, SALVATORE; DEL GROSSO, Erika; Fakhfouri, Gohar; Troiani, Maria Pia; Alisi, Maria Alessandra; GROSA, Giorgio; SORBA, Giovanni; CANONICO, Pier Luigi; Orsomando, Giuseppe; Cuzzocrea, Salvatore; GENAZZANI, Armando; GALLI, Ubaldina; TRON, Gian Cesare
Design, synthesis, and biological evaluation of combretabenzodiazepines: a novel class of anti-tubulin agents
2015-01-01 GALLI, Ubaldina; TRAVELLI, Cristina; APRILE, SILVIO; Arrigoni, Elena; TORRETTA, SIMONE; GROSA, Giorgio; MASSAROTTI, Alberto; SORBA, Giovanni; CANONICO, Pier Luigi; GENAZZANI, Armando; TRON, Gian Cesare
A Concise Synthesis of Pyrazole Analogues of Combretastatin A1 as Potent Antitubulin Agents
2013-01-01 ZANINETTI, ROBERTA; Cortese SV; APRILE, SILVIO; MASSAROTTI, Alberto; CANONICO, Pier Luigi; SORBA, Giovanni; GROSA, Giorgio; GENAZZANI, Armando; PIRALI, Tracey
QUINOLIN-4 (1H) -ONE DERIVATIVES AS INHIBITORS OF PHOSPHATIDYLINOSITOL 3-KINASES
2012-01-01 Giovanni Sorba; Gian Cesare Tron; Tracey Pirali; Ubaldina Galli; Alberto Massarotti; Emilio Hirsch; Elisa Ciraolo
Identification of a sirtuin 3 inhibitor that displays selectivity over sirtuin 1 and 2
2012-01-01 GALLI, Ubaldina; MESENZANI, Ornella; Coppo C; SORBA, Giovanni; CANONICO, Pier Luigi; TRON, Gian Cesare; GENAZZANI, Armando
Replacement of the double bond of antitubulin chalcones with triazoles and tetrazoles: synthesis and biological evaluation
2011-01-01 MESENZANI, Ornella; MASSAROTTI, Alberto; Giustiniano, M; PIRALI, Tracey; Bevilacqua, V; CALDARELLI, ANTONIO; CANONICO, Pier Luigi; SORBA, Giovanni; Novellino, E; GENAZZANI, Armando; TRON, Gian Cesare
A novel potent nicotinamide phosphoribosyltransferase inhibitor synthesized via click chemistry
2010-01-01 COLOMBANO, GIAMPIERO; TRAVELLI, Cristina; GALLI, Ubaldina; CALDARELLI, ANTONIO; Chini MG; CANONICO, Pier Luigi; SORBA, Giovanni; Bifulco G; TRON, Gian Cesare; GENAZZANI, Armando
Essential Role of the p110β Subunit of Phosphoinositide 3-OH Kinase in Male Fertility
2010-01-01 Elisa Ciraolo; Fulvio Morello; Robin M. Hobbs; Frieder Wolf; Romina Marone; Manuela Iezzi; Xiaoyun Lu; Giulio Mengozzi; Fiorella Altruda; Giovanni Sorba; Kaomei Guan; Pier Paolo Pandolfi; Matthias P. Wymann; Emilio Hirsch
Synthesis, biological evaluation, and molecular docking of Ugi products containing a zinc-chelating moiety as novel inhibitors of histone deacetylase
2009-01-01 GROLLA, AMBRA; Podesta V; Chini MG; Di Micco S; Vallario A; GENAZZANI, Armando; CANONICO, Pier Luigi; Bifulco G; TRON, Gian Cesare; SORBA, Giovanni; PIRALI, Tracey
Synthesis and biological evaluation of isosteric analogues of FK866, an inhibitor of NAD salvage
2008-01-01 GALLI, Ubaldina; ERCOLANO, EMANUELA; CARRARO, Lorenzo Roberto; Blasi Roman CR; SORBA, Giovanni; CANONICO, Pier Luigi; GENAZZANI, Armando; TRON, Gian Cesare; BILLINGTON, Richard Andrew
Click chemistry reactions in medicinal chemistry: applications of the 1,3-dipolar cycloaddition between azides and alkynes
2008-01-01 TRON, Gian Cesare; PIRALI, Tracey; BILLINGTON, Richard Andrew; CANONICO, Pier Luigi; SORBA, Giovanni; GENAZZANI, Armando
Solution-phase parallel synthesis and biological evaluation of combretatriazoles
2008-01-01 CAFICI L; PIRALI, Tracey; CONDORELLI, Fabrizio; DEL GROSSO, Erika; MASSAROTTI, Alberto; SORBA, Giovanni; CANONICO, Pier Luigi; TRON, Gian Cesare; GENAZZANI, Armando
Triazole-modified histone deacetylase inhibitors as a rapid route to drug discovery
2008-01-01 PIRALI, Tracey; PAGLIAI, Francesca; Mercurio C; Boggio R; CANONICO, Pier Luigi; SORBA, Giovanni; TRON, Gian Cesare; GENAZZANI, Armando
Design, Synthesis, and Biological Evaluation of New (2E,6E)-10-(Dimethylamino)-3,7-dimethyl-2,6-decadien-1-ol Ethers as Inhibitors of Human and Trypanosoma cruzi Oxidosqualene Cyclase.
2007-01-01 U. GALLI; S. OLIARO-BOSSO; S. TARAMINO; S. VENEGONI; E. PASTORE; GC. TRON; G. BALLIANO; F. VIOLA; G. SORBA
Estrogenic analogues synthesized by click chemistry
2007-01-01 PIRALI, Tracey; GATTI S; DI BRISCO R; TACCHI, Sara; ZANINETTI, ROBERTA; BRUNELLI, Elisa; MASSAROTTI, Alberto; SORBA, Giovanni; CANONICO, Pier Luigi; MORO, Laura; GENAZZANI, Armando; TRON, Gian Cesare; BILLINGTON, Richard Andrew
Replacement of the lactone moiety on podophyllotoxin and steganacin analogues with a 1,5-disubstituted 1,2,3-triazole via ruthenium-catalyzed click chemistry
2007-01-01 IMPERIO, DANIELA; PIRALI, Tracey; GALLI, Ubaldina; PAGLIAI, Francesca; Cafici L; CANONICO, Pier Luigi; SORBA, Giovanni; GENAZZANI, Armando; TRON, Gian Cesare
Medicinal chemistry of combretastatin A4: present and future directions
2006-01-01 TRON, Gian Cesare; PIRALI, Tracey; SORBA, Giovanni; PAGLIAI F; BUSACCA S; GENAZZANI, Armando
| Titolo | Data di pubblicazione | Autore(i) | File |
|---|---|---|---|
| Icilio Guareschi and his amazing “1897 reaction” | 2021 | Tron, Gian Cesare; Minassi, Alberto; Sorba, Giovanni; Fausone, Mara; Appendino, Giovanni | |
| Targeting Transient Receptor Potential Vanilloid 1 (TRPV1) Channel Softly: The Discovery of Passerini Adducts as a Topical Treatment for Inflammatory Skin Disorders | 2018 | Serafini, Marta; Griglio, Alessia; Aprile, Silvio; Seiti, Fabio; Travelli, Cristina; Pattarino, Franco; Grosa, Giorgio; Sorba, Giovanni; Genazzani, Armando; Gonzalez-Rodriguez, Sara; Butron, Laura; Devesa, Isabel; Fernandez-Carvajal, Asia; Pirali, Tracey; Ferrer-Montiel, Antonio | |
| Pyrtriazoles, a Novel Class of Store-Operated Calcium Entry Modulators: Discovery, Biological Profiling, and in Vivo Proof-of-Concept Efficacy in Acute Pancreatitis | 2018 | Riva, Beatrice; Griglio, Alessia; Serafini, Marta; CORDERO SANCHEZ, CELIA; Aprile, Silvio; Di Paola, Rosanna; Gugliandolo, Enrico; Alansary, Dalia; BIOCOTINO, Isabella; Lim, Dmitry; Grosa, Giorgio; Galli, Ubaldina; Niemeyer, Barbara; Sorba, Giovanni; Canonico, Pier Luigi; Cuzzocrea, Salvatore; Genazzani, Armando; Pirali, Tracey | |
| Identification of Novel Triazole-Based Nicotinamide Phosphoribosyltransferase (NAMPT) Inhibitors Endowed with Antiproliferative and Antiinflammatory Activity | 2017 | TRAVELLI, Cristina; APRILE, SILVIO; Rahimian, Reza; Grolla, Ambra A.; ROGATI, FEDERICA; Bertolotti, Mattia; Malagnino, Floriana; Di Paola, Rosanna; Impellizzeri, Daniela; FUSCO, Roberta; MERCALLI, VALENTINA; MASSAROTTI, Alberto; Stortini, Giorgio; TERRAZZINO, SALVATORE; DEL GROSSO, Erika; Fakhfouri, Gohar; Troiani, Maria Pia; Alisi, Maria Alessandra; GROSA, Giorgio; SORBA, Giovanni; CANONICO, Pier Luigi; Orsomando, Giuseppe; Cuzzocrea, Salvatore; GENAZZANI, Armando; GALLI, Ubaldina; TRON, Gian Cesare | |
| Design, synthesis, and biological evaluation of combretabenzodiazepines: a novel class of anti-tubulin agents | 2015 | GALLI, Ubaldina; TRAVELLI, Cristina; APRILE, SILVIO; Arrigoni, Elena; TORRETTA, SIMONE; GROSA, Giorgio; MASSAROTTI, Alberto; SORBA, Giovanni; CANONICO, Pier Luigi; GENAZZANI, Armando; TRON, Gian Cesare | |
| A Concise Synthesis of Pyrazole Analogues of Combretastatin A1 as Potent Antitubulin Agents | 2013 | ZANINETTI, ROBERTA; Cortese SV; APRILE, SILVIO; MASSAROTTI, Alberto; CANONICO, Pier Luigi; SORBA, Giovanni; GROSA, Giorgio; GENAZZANI, Armando; PIRALI, Tracey | |
| QUINOLIN-4 (1H) -ONE DERIVATIVES AS INHIBITORS OF PHOSPHATIDYLINOSITOL 3-KINASES | 2012 | Giovanni Sorba; Gian Cesare Tron; Tracey Pirali; Ubaldina Galli; Alberto Massarotti; Emilio Hirsch; Elisa Ciraolo | |
| Identification of a sirtuin 3 inhibitor that displays selectivity over sirtuin 1 and 2 | 2012 | GALLI, Ubaldina; MESENZANI, Ornella; Coppo C; SORBA, Giovanni; CANONICO, Pier Luigi; TRON, Gian Cesare; GENAZZANI, Armando | |
| Replacement of the double bond of antitubulin chalcones with triazoles and tetrazoles: synthesis and biological evaluation | 2011 | MESENZANI, Ornella; MASSAROTTI, Alberto; Giustiniano, M; PIRALI, Tracey; Bevilacqua, V; CALDARELLI, ANTONIO; CANONICO, Pier Luigi; SORBA, Giovanni; Novellino, E; GENAZZANI, Armando; TRON, Gian Cesare | |
| A novel potent nicotinamide phosphoribosyltransferase inhibitor synthesized via click chemistry | 2010 | COLOMBANO, GIAMPIERO; TRAVELLI, Cristina; GALLI, Ubaldina; CALDARELLI, ANTONIO; Chini MG; CANONICO, Pier Luigi; SORBA, Giovanni; Bifulco G; TRON, Gian Cesare; GENAZZANI, Armando | |
| Essential Role of the p110β Subunit of Phosphoinositide 3-OH Kinase in Male Fertility | 2010 | Elisa Ciraolo; Fulvio Morello; Robin M. Hobbs; Frieder Wolf; Romina Marone; Manuela Iezzi; Xiaoyun Lu; Giulio Mengozzi; Fiorella Altruda; Giovanni Sorba; Kaomei Guan; Pier Paolo Pandolfi; Matthias P. Wymann; Emilio Hirsch | |
| Synthesis, biological evaluation, and molecular docking of Ugi products containing a zinc-chelating moiety as novel inhibitors of histone deacetylase | 2009 | GROLLA, AMBRA; Podesta V; Chini MG; Di Micco S; Vallario A; GENAZZANI, Armando; CANONICO, Pier Luigi; Bifulco G; TRON, Gian Cesare; SORBA, Giovanni; PIRALI, Tracey | |
| Synthesis and biological evaluation of isosteric analogues of FK866, an inhibitor of NAD salvage | 2008 | GALLI, Ubaldina; ERCOLANO, EMANUELA; CARRARO, Lorenzo Roberto; Blasi Roman CR; SORBA, Giovanni; CANONICO, Pier Luigi; GENAZZANI, Armando; TRON, Gian Cesare; BILLINGTON, Richard Andrew | |
| Click chemistry reactions in medicinal chemistry: applications of the 1,3-dipolar cycloaddition between azides and alkynes | 2008 | TRON, Gian Cesare; PIRALI, Tracey; BILLINGTON, Richard Andrew; CANONICO, Pier Luigi; SORBA, Giovanni; GENAZZANI, Armando | |
| Solution-phase parallel synthesis and biological evaluation of combretatriazoles | 2008 | CAFICI L; PIRALI, Tracey; CONDORELLI, Fabrizio; DEL GROSSO, Erika; MASSAROTTI, Alberto; SORBA, Giovanni; CANONICO, Pier Luigi; TRON, Gian Cesare; GENAZZANI, Armando | |
| Triazole-modified histone deacetylase inhibitors as a rapid route to drug discovery | 2008 | PIRALI, Tracey; PAGLIAI, Francesca; Mercurio C; Boggio R; CANONICO, Pier Luigi; SORBA, Giovanni; TRON, Gian Cesare; GENAZZANI, Armando | |
| Design, Synthesis, and Biological Evaluation of New (2E,6E)-10-(Dimethylamino)-3,7-dimethyl-2,6-decadien-1-ol Ethers as Inhibitors of Human and Trypanosoma cruzi Oxidosqualene Cyclase. | 2007 | U. GALLI; S. OLIARO-BOSSO; S. TARAMINO; S. VENEGONI; E. PASTORE; GC. TRON; G. BALLIANO; F. VIOLA; G. SORBA | |
| Estrogenic analogues synthesized by click chemistry | 2007 | PIRALI, Tracey; GATTI S; DI BRISCO R; TACCHI, Sara; ZANINETTI, ROBERTA; BRUNELLI, Elisa; MASSAROTTI, Alberto; SORBA, Giovanni; CANONICO, Pier Luigi; MORO, Laura; GENAZZANI, Armando; TRON, Gian Cesare; BILLINGTON, Richard Andrew | |
| Replacement of the lactone moiety on podophyllotoxin and steganacin analogues with a 1,5-disubstituted 1,2,3-triazole via ruthenium-catalyzed click chemistry | 2007 | IMPERIO, DANIELA; PIRALI, Tracey; GALLI, Ubaldina; PAGLIAI, Francesca; Cafici L; CANONICO, Pier Luigi; SORBA, Giovanni; GENAZZANI, Armando; TRON, Gian Cesare | |
| Medicinal chemistry of combretastatin A4: present and future directions | 2006 | TRON, Gian Cesare; PIRALI, Tracey; SORBA, Giovanni; PAGLIAI F; BUSACCA S; GENAZZANI, Armando |
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