Sfoglia per Autore
Principi di Chimica Farmaceutica
2014-01-01 Fruttero R.; Guglielmo S.
A multi-photoresponsive molecular-hybrid for dual-modal photoinactivation of cancer cells
2014-01-01 Aurore Fraix;Stefano Guglielmo;Venera Cardile;Adriana C. E. Graziano;Ruxandra Gref;Barbara Rolando;Roberta Fruttero;Alberto Gasco;Salvatore Sortino
New praziquantel derivatives containing NO-donor furoxans and related furazans as active agents against Schistosoma mansoni
2014-01-01 Stefano Guglielmo;Daniela Cortese;Francesca Vottero;Barbara Rolando;Valerie P. Kommer;David L. Williams;Roberta Fruttero;Alberto Gasco
New furoxan derivatives with Schistosomicidal activity.
2014-01-01 Daniela Cortese; David L. Williams; Peter D. Ziniel; Latasha Day; Stefano Guglielmo; Roberta Fruttero; Alberto Gasco.
Leishmanicidal Activity of Novel Synthetic Furoxan and Benzofuroxan Derivatives
2014-01-01 L. A. Dutra;L. De Almeida;T. G. Passalacqua;J. S. Reis;F. A. E. Torres;I. Martinez;R. G. Peccinini;C. Man Chin;K. Chegaev;S. Guglielmo;R. Fruttero;M. A. S. Graminha;J. L. Dos Santos
NO-Donor Dihydroartemisinin Derivatives as Multitarget Agents for the Treatment of Cerebral Malaria
2015-01-01 Bertinaria, Massimo; Orjuela-Sanchez, Pamela; Marini, Elisabetta; Guglielmo, Stefano; Hofer, Anthony; Martins, Yuri C.; Zanini, Graziela M.; Frangos, John A.; Gasco, Alberto; Fruttero, Roberta; Carvalho, Leonardo J. M.
Synthesis and biological activity of furoxan derivatives against Mycobacterium tuberculosis
2016-01-01 Fernandes, Guilherme Felipe dos Santos; de Souza, Paula Carolina; Marino, Leonardo Biancolino; Chegaev, Konstantin; Guglielmo, Stefano; Lazzarato, Loretta; Fruttero, Roberta; Chung, Man Chin; Pavan, Fernando Rogério; dos Santos, Jean Leandro
Light-Tunable Generation of Singlet Oxygen and Nitric Oxide with a Bichromophoric Molecular Hybrid: a Bimodal Approach to Killing Cancer Cells
2016-01-01 Fraix, Aurore; Blangetti, Marco; Guglielmo, Stefano; Lazzarato, Loretta; Marino, Nino; Cardile, Venera; Graziano, Adriana C.E.; Manet, Ilse; Fruttero, Roberta; Gasco, Alberto; Sortino, Salvatore
Synthesis and Biological Evaluation of N2-Substituted 2,4-Diamino-6-cyclohexylmethoxy-5-nitrosopyrimidines and Related 5-Cyano-NNO-azoxy Derivatives as Cyclin-Dependent Kinase 2 (CDK2) Inhibitors
2016-01-01 Cortese, Daniela; Chegaev, Konstantin; Guglielmo, Stefano; Wang, Lan Z.; Golding, Bernard T.; Cano, Céline; Fruttero, Roberta
A Potent and Selective P-gp Modulator for Altering Multidrug Resistance Due to Pump Overexpression
2016-01-01 Guglielmo, Stefano; Contino, Marialessandra; Lazzarato, Loretta; Perrone, Maria Grazia; Blangetti, Marco; Fruttero, Roberta; Colabufo, Nicola Antonio
Structure-Activity Relationship Studies on Tetrahydroisoquinoline Derivatives: [4′-(6,7-Dimethoxy-3,4-dihydro-1H-isoquinolin-2-ylmethyl)biphenyl-4-ol] (MC70) Conjugated through Flexible Alkyl Chains with Furazan Moieties Gives Rise to Potent and Selective Ligands of P-glycoprotein
2016-01-01 Guglielmo, Stefano; Lazzarato, Loretta; Contino, Marialessandra; Perrone, Maria G.; Chegaev, Konstantin; Carrieri, Antonio; Fruttero, Roberta; Colabufo, Nicola A.; Gasco, Alberto
Direct introduction of cyano group on furoxan ring
2017-01-01 Annaratone, Lorenzo; Guglielmo, Stefano; Chegaev, Konstantin
Design, Synthesis, and Characterization of N-Oxide-Containing Heterocycles with in Vivo Sterilizing Antitubercular Activity
2017-01-01 Dos Santos Fernandes, Guilherme Felipe; De Souza, Paula Carolina; Moreno-viguri, Elsa; Santivaã±ez-veliz, Mery; Paucar, Rocio; Pã©rez-silanes, Silvia; Chegaev, Konstantin; Guglielmo, Stefano; Lazzarato, Loretta; Fruttero, Roberta; Man Chin, Chung; Da Silva, Patricia Bento; Chorilli, Marlus; Solcia, Mariana Cristina; Ribeiro, Camila Marãngolo; Silva, Caio Sander Paiva; Marino, Leonardo Biancolino; Bosquesi, Priscila Longhin; Hunt, Debbie M.; De Carvalho, Luiz Pedro S.; De Souza Costa, Carlos Alberto; Cho, Sang Hyun; Wang, Yuehong; Franzblau, Scott Gary; Pavan, Fernando Rogã©rio; Dos Santos, Jean Leandro
New furoxan derivatives for the treatment of ocular hypertension
2017-01-01 Blangetti, Marco; Rolando, Barbara; Chegaev, Konstantin; Guglielmo, Stefano; Lazzarato, Loretta; Durante, Mariaconcetta; Masini, Emanuela; Almirante, Nicoletta; Bastia, Elena; Impagnatiello, Francesco; Fruttero, Roberta; Gasco, Alberto
Furoxan nitric oxide donors disperse Pseudomonas aeruginosa biofilms, accelerate growth, and repress pyoverdine production
2017-01-01 Poh, Wee Han; Barraud, Nicolas; Guglielmo, Stefano; Lazzarato, Loretta; Fruttero, Roberta; Rolando, Barbara; Rice, Scott A.
gem-Dinitroalkyl Benzenes: A Novel Class of IOP-Lowering Agents for the Treatment of Ocular Hypertension
2017-01-01 Blangetti, Marco; Rolando, Barbara; Marini, Elisabetta; Chegaev, Konstantin; Guglielmo, Stefano; Lazzarato, Loretta; Laura, Lucarini; Emanuela, Masini; Fruttero, Roberta
Sistemi nanocompositi termosensibili per la somministrazione intravitreale di cefuroxima
2018-01-01 BRUNO CAPRARELLI, SIMONA SAPINO, ELENA PEIRA, DANIELA CHIRIO, SUSHIL A JADHAV, SIMONETTA OLIARO BOSSO, STEFANO GUGLIELMO, RAFFAELLA BARBERO, ANTONIO MARIA FEA, CLAUDIA FRUTTERO, FRANCO DOSIO, MARINA GALLARATE
Anti-pseudomonas activity of 3-nitro-4-phenylfuroxan
2018-01-01 Orlandi, Viviana Teresa*; Bolognese, Fabrizio; Rolando, Barbara; Guglielmo, Stefano; Lazzarato, Loretta; Fruttero, Roberta
Discovery of phenylsulfonylfuroxan derivatives as gamma globin inducers by histone acetylation
2018-01-01 Melo, Thais Regina Ferreira de; Kumkhaek, Chutima; Fernandes, Guilherme Felipe dos Santos; Lopes Pires, Maria Elisa; Chelucci, Rafael Consolin; Barbieri, Karina Pereira; Coelho, Fernanda; Capote, Ticiana Sidorenko de Oliveira; Lanaro, Carolina; Carlos, Iracilda Zeppone; Marcondes, Sisi; Chegaev, Konstantin; Guglielmo, Stefano; Fruttero, Roberta; Chung, Man Chin; Costa, Fernando Ferreira; Rodgers, Griffin P.; dos Santos, Jean Leandro*
Mitochondrial delivery of phenol substructure triggers mitochondrial depolarization and apoptosis of cancer cells
2018-01-01 Gazzano, Elena; Lazzarato, Loretta; Rolando, Barbara; Kopecka, Joanna; Guglielmo, Stefano; Costamagna, Costanzo; Chegaev, Konstantin*; Riganti, Chiara
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
Principi di Chimica Farmaceutica | 2014 | Fruttero R.; Guglielmo S. | |
A multi-photoresponsive molecular-hybrid for dual-modal photoinactivation of cancer cells | 2014 | Aurore Fraix;Stefano Guglielmo;Venera Cardile;Adriana C. E. Graziano;Ruxandra Gref;Barbara Rolando;Roberta Fruttero;Alberto Gasco;Salvatore Sortino | |
New praziquantel derivatives containing NO-donor furoxans and related furazans as active agents against Schistosoma mansoni | 2014 | Stefano Guglielmo;Daniela Cortese;Francesca Vottero;Barbara Rolando;Valerie P. Kommer;David L. Williams;Roberta Fruttero;Alberto Gasco | |
New furoxan derivatives with Schistosomicidal activity. | 2014 | Daniela Cortese; David L. Williams; Peter D. Ziniel; Latasha Day; Stefano Guglielmo; Roberta Fruttero; Alberto Gasco. | |
Leishmanicidal Activity of Novel Synthetic Furoxan and Benzofuroxan Derivatives | 2014 | L. A. Dutra;L. De Almeida;T. G. Passalacqua;J. S. Reis;F. A. E. Torres;I. Martinez;R. G. Peccinini;C. Man Chin;K. Chegaev;S. Guglielmo;R. Fruttero;M. A. S. Graminha;J. L. Dos Santos | |
NO-Donor Dihydroartemisinin Derivatives as Multitarget Agents for the Treatment of Cerebral Malaria | 2015 | Bertinaria, Massimo; Orjuela-Sanchez, Pamela; Marini, Elisabetta; Guglielmo, Stefano; Hofer, Anthony; Martins, Yuri C.; Zanini, Graziela M.; Frangos, John A.; Gasco, Alberto; Fruttero, Roberta; Carvalho, Leonardo J. M. | |
Synthesis and biological activity of furoxan derivatives against Mycobacterium tuberculosis | 2016 | Fernandes, Guilherme Felipe dos Santos; de Souza, Paula Carolina; Marino, Leonardo Biancolino; Chegaev, Konstantin; Guglielmo, Stefano; Lazzarato, Loretta; Fruttero, Roberta; Chung, Man Chin; Pavan, Fernando Rogério; dos Santos, Jean Leandro | |
Light-Tunable Generation of Singlet Oxygen and Nitric Oxide with a Bichromophoric Molecular Hybrid: a Bimodal Approach to Killing Cancer Cells | 2016 | Fraix, Aurore; Blangetti, Marco; Guglielmo, Stefano; Lazzarato, Loretta; Marino, Nino; Cardile, Venera; Graziano, Adriana C.E.; Manet, Ilse; Fruttero, Roberta; Gasco, Alberto; Sortino, Salvatore | |
Synthesis and Biological Evaluation of N2-Substituted 2,4-Diamino-6-cyclohexylmethoxy-5-nitrosopyrimidines and Related 5-Cyano-NNO-azoxy Derivatives as Cyclin-Dependent Kinase 2 (CDK2) Inhibitors | 2016 | Cortese, Daniela; Chegaev, Konstantin; Guglielmo, Stefano; Wang, Lan Z.; Golding, Bernard T.; Cano, Céline; Fruttero, Roberta | |
A Potent and Selective P-gp Modulator for Altering Multidrug Resistance Due to Pump Overexpression | 2016 | Guglielmo, Stefano; Contino, Marialessandra; Lazzarato, Loretta; Perrone, Maria Grazia; Blangetti, Marco; Fruttero, Roberta; Colabufo, Nicola Antonio | |
Structure-Activity Relationship Studies on Tetrahydroisoquinoline Derivatives: [4′-(6,7-Dimethoxy-3,4-dihydro-1H-isoquinolin-2-ylmethyl)biphenyl-4-ol] (MC70) Conjugated through Flexible Alkyl Chains with Furazan Moieties Gives Rise to Potent and Selective Ligands of P-glycoprotein | 2016 | Guglielmo, Stefano; Lazzarato, Loretta; Contino, Marialessandra; Perrone, Maria G.; Chegaev, Konstantin; Carrieri, Antonio; Fruttero, Roberta; Colabufo, Nicola A.; Gasco, Alberto | |
Direct introduction of cyano group on furoxan ring | 2017 | Annaratone, Lorenzo; Guglielmo, Stefano; Chegaev, Konstantin | |
Design, Synthesis, and Characterization of N-Oxide-Containing Heterocycles with in Vivo Sterilizing Antitubercular Activity | 2017 | Dos Santos Fernandes, Guilherme Felipe; De Souza, Paula Carolina; Moreno-viguri, Elsa; Santivaã±ez-veliz, Mery; Paucar, Rocio; Pã©rez-silanes, Silvia; Chegaev, Konstantin; Guglielmo, Stefano; Lazzarato, Loretta; Fruttero, Roberta; Man Chin, Chung; Da Silva, Patricia Bento; Chorilli, Marlus; Solcia, Mariana Cristina; Ribeiro, Camila Marãngolo; Silva, Caio Sander Paiva; Marino, Leonardo Biancolino; Bosquesi, Priscila Longhin; Hunt, Debbie M.; De Carvalho, Luiz Pedro S.; De Souza Costa, Carlos Alberto; Cho, Sang Hyun; Wang, Yuehong; Franzblau, Scott Gary; Pavan, Fernando Rogã©rio; Dos Santos, Jean Leandro | |
New furoxan derivatives for the treatment of ocular hypertension | 2017 | Blangetti, Marco; Rolando, Barbara; Chegaev, Konstantin; Guglielmo, Stefano; Lazzarato, Loretta; Durante, Mariaconcetta; Masini, Emanuela; Almirante, Nicoletta; Bastia, Elena; Impagnatiello, Francesco; Fruttero, Roberta; Gasco, Alberto | |
Furoxan nitric oxide donors disperse Pseudomonas aeruginosa biofilms, accelerate growth, and repress pyoverdine production | 2017 | Poh, Wee Han; Barraud, Nicolas; Guglielmo, Stefano; Lazzarato, Loretta; Fruttero, Roberta; Rolando, Barbara; Rice, Scott A. | |
gem-Dinitroalkyl Benzenes: A Novel Class of IOP-Lowering Agents for the Treatment of Ocular Hypertension | 2017 | Blangetti, Marco; Rolando, Barbara; Marini, Elisabetta; Chegaev, Konstantin; Guglielmo, Stefano; Lazzarato, Loretta; Laura, Lucarini; Emanuela, Masini; Fruttero, Roberta | |
Sistemi nanocompositi termosensibili per la somministrazione intravitreale di cefuroxima | 2018 | BRUNO CAPRARELLI, SIMONA SAPINO, ELENA PEIRA, DANIELA CHIRIO, SUSHIL A JADHAV, SIMONETTA OLIARO BOSSO, STEFANO GUGLIELMO, RAFFAELLA BARBERO, ANTONIO MARIA FEA, CLAUDIA FRUTTERO, FRANCO DOSIO, MARINA GALLARATE | |
Anti-pseudomonas activity of 3-nitro-4-phenylfuroxan | 2018 | Orlandi, Viviana Teresa*; Bolognese, Fabrizio; Rolando, Barbara; Guglielmo, Stefano; Lazzarato, Loretta; Fruttero, Roberta | |
Discovery of phenylsulfonylfuroxan derivatives as gamma globin inducers by histone acetylation | 2018 | Melo, Thais Regina Ferreira de; Kumkhaek, Chutima; Fernandes, Guilherme Felipe dos Santos; Lopes Pires, Maria Elisa; Chelucci, Rafael Consolin; Barbieri, Karina Pereira; Coelho, Fernanda; Capote, Ticiana Sidorenko de Oliveira; Lanaro, Carolina; Carlos, Iracilda Zeppone; Marcondes, Sisi; Chegaev, Konstantin; Guglielmo, Stefano; Fruttero, Roberta; Chung, Man Chin; Costa, Fernando Ferreira; Rodgers, Griffin P.; dos Santos, Jean Leandro* | |
Mitochondrial delivery of phenol substructure triggers mitochondrial depolarization and apoptosis of cancer cells | 2018 | Gazzano, Elena; Lazzarato, Loretta; Rolando, Barbara; Kopecka, Joanna; Guglielmo, Stefano; Costamagna, Costanzo; Chegaev, Konstantin*; Riganti, Chiara |
Legenda icone
- file ad accesso aperto
- file disponibili sulla rete interna
- file disponibili agli utenti autorizzati
- file disponibili solo agli amministratori
- file sotto embargo
- nessun file disponibile