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Mostrati risultati da 41 a 60 di 168
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Log P in the bRo5 chemical space 2019 Maura Vallaro, Giuseppe Ermondi, Gilles Goetz, Marina Shalaeva, Sonja Visentin, Giulia Caron
Experimental lipophilicity for beyond Rule of 5 compounds 2019 Ermondi, Giuseppe; Vallaro, Maura; Goetz, Gilles; Shalaeva, Marina; Caron, Giulia
A mucus model to evaluate the diffusion of drugs for more efficient cystic fibrosis therapies 2019 Pacheco DP, Butnarasu C, Bertoglio F, Suarez Vargas N, Briatico-Vangosa F, van Uden S, Visai L, Petrini P, Vallaro M, Caron G, Visentin S
The NFKBIA’s amplification in cancer, emerging molecular targets for lung cancer therapy 2019 Giovanna Carrà, Rocco Piazza, Giuseppe Ermondi, Giulia Caron, Chiara Riganti, Beatrice Maffeo, Antonio Cartellà, Marcello Francesco Lingua, Mara Brancaccio, Riccardo Taulli, Silvia Novello; Alessandro Morotti
Translating unusual computational methods to drug discovery: Taking advantage of work in other fields 2019 Caron G.; Ermondi G.
MLR, PLSR-BR Analysis and MBPLSR to Interpret Multivariate QSPR Models. The Case of a Micellar Liquid Chromatography Descriptor (log K WSDS ) 2019 Ermondi G.; Caron G.
Author Correction: Modeling ErbB2-p130Cas interaction to design new potential anticancer agents (Scientific Reports, (2019), 9, 1, (3089), 10.1038/s41598-019-39510-w) 2019 Costamagna A.; Rossi Sebastiano M.; Natalini D.; Simoni M.; Valabrega G.; Defilippi P.; Visentin S.; Ermondi G.; Turco E.; Caron G.; Cabodi S.
Modeling ErbB2-p130Cas interaction to design new potential anticancer agents. 2019 Andrea Costamagna, Matteo Rossi Sebastiano, Dora Natalini, Matilde Simoni, Giorgio Valabrega, Paola Defilippi, Sonja Visentin, Giuseppe Ermondi, Emilia Turco, Giulia Caron, Sara Cabodi
Intramolecular hydrogen bonding: An opportunity for improved design in medicinal chemistry 2019 Caron G.; Kihlberg J.; Ermondi G.
Learning how to use IAM chromatography for predicting permeability 2018 Ermondi, Giuseppe; Vallaro, Maura; Caron, Giulia
Block relevance (BR) analysis and polarity descriptors in property-based drug design 2018 Ermondi, Giuseppe; Caron, Giulia*
Charged cyclic hexapeptides: Updating molecular descriptors for permeability purposes 2018 Ermondi, G.; Vallaro, M.; Camacho-Leal, M.P.; Potter, T.; Visentin, S.; Caron, G.*
Conformational Sampling of Macrocyclic Drugs in Different Environments: Can We Find the Relevant Conformations? 2018 Poongavanam, Vasanthanathan; Danelius, Emma; Peintner, Stefan; Alcaraz, Lilian; Caron, Giulia; Cummings, Maxwell D.; Wlodek, Stanislaw; Erdelyi, Mate; Hawkins, Paul C. D.; Ermondi, Giuseppe*; Kihlberg, Jan
Log P as a tool in intramolecular hydrogen bond considerations 2018 Caron, Giulia*; Vallaro, Maura; Ermondi, Giuseppe
Impact of Dynamically Exposed Polarity on Permeability and Solubility of Chameleonic Drugs beyond the Rule of 5 2018 Rossi Sebastiano, Matteo; Doak, Bradley C.; Backlund, Maria; Poongavanam, Vasanthanathan; Over, Björn; Ermondi, Giuseppe; Caron, Giulia; Matsson, Pär*; Kihlberg, Jan
HTS Assay Development: an airway mucus microenvironment modelling to be applied on cystic fibrosis drug discovery 2017 Petrini, P.; Pacheco, D.; Visai, L.; Coletti, M.; Bertoglio, F.; Caron, G.; Visentin, S.
Airway mucus microenvironment modelling to be applied on cystic fibrosis drug discovery 2017 Petrini, P; Pacheco, Dp; Pontremoli, C.; Caron, G.; Visentin, S
Why we need to implement intramolecular hydrogen-bonding considerations in drug discovery 2017 Caron, Giulia; Ermondi, Giuseppe
Relationship between passive permeability and molecular polarity using block relevance analysis 2017 Goetz, Gilles H; Shalaeva, Marina; Caron, Giulia; Ermondi, Giuseppe; Philippe, Laurence
Updating molecular properties during early drug discovery 2017 Caron, Giulia; Ermondi, Giuseppe
Mostrati risultati da 41 a 60 di 168
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