Sfoglia per Autore
Author Correction: Modeling ErbB2-p130Cas interaction to design new potential anticancer agents (Scientific Reports, (2019), 9, 1, (3089), 10.1038/s41598-019-39510-w)
2019-01-01 Costamagna A.; Rossi Sebastiano M.; Natalini D.; Simoni M.; Valabrega G.; Defilippi P.; Visentin S.; Ermondi G.; Turco E.; Caron G.; Cabodi S.
Modeling ErbB2-p130Cas interaction to design new potential anticancer agents.
2019-01-01 Andrea Costamagna, Matteo Rossi Sebastiano, Dora Natalini, Matilde Simoni, Giorgio Valabrega, Paola Defilippi, Sonja Visentin, Giuseppe Ermondi, Emilia Turco, Giulia Caron, Sara Cabodi
Intramolecular hydrogen bonding: An opportunity for improved design in medicinal chemistry
2019-01-01 Caron G.; Kihlberg J.; Ermondi G.
Learning how to use IAM chromatography for predicting permeability
2018-01-01 Ermondi, Giuseppe; Vallaro, Maura; Caron, Giulia
Block relevance (BR) analysis and polarity descriptors in property-based drug design
2018-01-01 Ermondi, Giuseppe; Caron, Giulia*
Charged cyclic hexapeptides: Updating molecular descriptors for permeability purposes
2018-01-01 Ermondi, G.; Vallaro, M.; Camacho-Leal, M.P.; Potter, T.; Visentin, S.; Caron, G.*
Conformational Sampling of Macrocyclic Drugs in Different Environments: Can We Find the Relevant Conformations?
2018-01-01 Poongavanam, Vasanthanathan; Danelius, Emma; Peintner, Stefan; Alcaraz, Lilian; Caron, Giulia; Cummings, Maxwell D.; Wlodek, Stanislaw; Erdelyi, Mate; Hawkins, Paul C. D.; Ermondi, Giuseppe*; Kihlberg, Jan
Log P as a tool in intramolecular hydrogen bond considerations
2018-01-01 Caron, Giulia*; Vallaro, Maura; Ermondi, Giuseppe
Impact of Dynamically Exposed Polarity on Permeability and Solubility of Chameleonic Drugs beyond the Rule of 5
2018-01-01 Rossi Sebastiano, Matteo; Doak, Bradley C.; Backlund, Maria; Poongavanam, Vasanthanathan; Over, Björn; Ermondi, Giuseppe; Caron, Giulia; Matsson, Pär*; Kihlberg, Jan
Why we need to implement intramolecular hydrogen-bonding considerations in drug discovery
2017-01-01 Caron, Giulia; Ermondi, Giuseppe
Relationship between passive permeability and molecular polarity using block relevance analysis
2017-01-01 Goetz, Gilles H; Shalaeva, Marina; Caron, Giulia; Ermondi, Giuseppe; Philippe, Laurence
Updating molecular properties during early drug discovery
2017-01-01 Caron, Giulia; Ermondi, Giuseppe
High throughput methods to measure the propensity of compounds to form intramolecular hydrogen bonding
2017-01-01 Caron, Giulia; Vallaro, Maura; Ermondi, Giuseppe
IAM chromatography: information provided and relevance in the prediction of permeability
2017-01-01 Maura Vallaro, Giuseppe Ermondi, Sonja Visentin, Giulia Caron
Do surface-based match solution-based techniques? the case of drug-liposome interaction
2016-01-01 Ermondi, Giuseppe; Caron, Giulia
Molecular descriptors for polarity: The need for going beyond polar surface area
2016-01-01 Caron, Giulia; Ermondi, Giuseppe
BR ANALYSIS: A TOOL TO UNRAVEL MOLECULAR INTERACTIONS BALANCE
2016-01-01 Ermondi, Giuseppe; Vallaro, Maura; Caron, Giulia
ZWITTERIONS IN DRUG DISCOVERY: STUDIES OF THE TAUTOMERIC EQUILIBRIUM WITH IN-SILICO AND EXPERIMENTAL TOOLS
2016-01-01 Caron, Giulia; Vallaro, Maura; Ermondi, Giuseppe
A Fast Chromatographic Method for Estimating Lipophilicity and Ionization in Nonpolar Membrane-Like Environment
2016-01-01 Caron, Giulia; Vallaro, Maura; Ermondi, Giuseppe; Goetz, Gilles H.; Abramov, Yuriy A.; Philippe, Laurence; Shalaeva, Marina
Multivariate analysis applied to Raman mapping of dye-functionalized carbon nanotubes: A novel approach to support the rational design of functional nanostructures
2015-01-01 Visentin, Sonja; Barbero, Nadia; Bertani, Francesca Romana; Guidi, Mariangela Cestelli; Ermondi, Giuseppe; Viscardi, Guido; Mussi, Valentina
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