GUGLIELMO, Stefano

GUGLIELMO, Stefano  

SCIENZA E TECNOLOGIA DEL FARMACO  

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A multi-photoresponsive molecular-hybrid for dual-modal photoinactivation of cancer cells 2014 Aurore Fraix;Stefano Guglielmo;Venera Cardile;Adriana C. E. Graziano;Ruxandra Gref;Barbara Rolando;Roberta Fruttero;Alberto Gasco;Salvatore Sortino
A new series of amodiaquine analogues modified in the basic side chain with in vitro antileishmanial and antiplasmodial activity 2009 Stefano Guglielmo; Massimo Bertinaria; Barbara Rolando; Marco Crosetti; Roberta Fruttero; Vanessa Yardley; Simon L. Croft; Alberto Gasco
A Potent and Selective P-gp Modulator for Altering Multidrug Resistance Due to Pump Overexpression 2016 Guglielmo, Stefano; Contino, Marialessandra; Lazzarato, Loretta; Perrone, Maria Grazia; Blangetti, Marco; Fruttero, Roberta; Colabufo, Nicola Antonio
Amodiaquine analogues containing NO-donor substructures: Synthesis and their preliminary evaluation as potential tools in the treatment of cerebral malaria 2011 Massimo Bertinaria; Stefano Guglielmo; Barbara Rolando; Marta Giorgis; Cristina Aragno; Roberta Fruttero; Alberto Gasco; Silvia Parapini; Donatella Taramelli; Yuri C. Martins; Leonardo J.M. Carvalho
Anti-pseudomonas activity of 3-nitro-4-phenylfuroxan 2018 Orlandi, Viviana Teresa*; Bolognese, Fabrizio; Rolando, Barbara; Guglielmo, Stefano; Lazzarato, Loretta; Fruttero, Roberta
Comparative Study of Different H2S Donors as Vasodilators and Attenuators of Superoxide-Induced Endothelial Damage 2023 Marini E.; Rolando B.; Sodano F.; Blua F.; Concina G.; Guglielmo S.; Lazzarato L.; Chegaev K.
Design, Biological Evaluation, and Molecular Modeling of Tetrahydroisoquinoline Derivatives: Discovery of A Potent P-Glycoprotein Ligand Overcoming Multidrug Resistance in Cancer Stem Cells 2019 Riganti, Chiara; Contino, Marialessandra*; Guglielmo, Stefano; Perrone, Maria G.; Salaroglio, Iris C.; Milosevic, Vladan; Giampietro, Roberta; Leonetti, Francesco; Rolando, Barbara; Lazzarato, Loretta; Colabufo, Nicola A.; Fruttero, Roberta
Design, Synthesis, and Characterization of N-Oxide-Containing Heterocycles with in Vivo Sterilizing Antitubercular Activity 2017 Dos Santos Fernandes, Guilherme Felipe; De Souza, Paula Carolina; Moreno-viguri, Elsa; Santivaã±ez-veliz, Mery; Paucar, Rocio; Pã©rez-silanes, Silvia; Chegaev, Konstantin; Guglielmo, Stefano; Lazzarato, Loretta; Fruttero, Roberta; Man Chin, Chung; Da Silva, Patricia Bento; Chorilli, Marlus; Solcia, Mariana Cristina; Ribeiro, Camila Marã­ngolo; Silva, Caio Sander Paiva; Marino, Leonardo Biancolino; Bosquesi, Priscila Longhin; Hunt, Debbie M.; De Carvalho, Luiz Pedro S.; De Souza Costa, Carlos Alberto; Cho, Sang Hyun; Wang, Yuehong; Franzblau, Scott Gary; Pavan, Fernando Rogã©rio; Dos Santos, Jean Leandro
Direct introduction of cyano group on furoxan ring 2017 Annaratone, Lorenzo; Guglielmo, Stefano; Chegaev, Konstantin
Discovery of phenylsulfonylfuroxan derivatives as gamma globin inducers by histone acetylation 2018 Melo, Thais Regina Ferreira de; Kumkhaek, Chutima; Fernandes, Guilherme Felipe dos Santos; Lopes Pires, Maria Elisa; Chelucci, Rafael Consolin; Barbieri, Karina Pereira; Coelho, Fernanda; Capote, Ticiana Sidorenko de Oliveira; Lanaro, Carolina; Carlos, Iracilda Zeppone; Marcondes, Sisi; Chegaev, Konstantin; Guglielmo, Stefano; Fruttero, Roberta; Chung, Man Chin; Costa, Fernando Ferreira; Rodgers, Griffin P.; dos Santos, Jean Leandro*
DNA-targeted NO release photoregulated by green light 2020 Cristina Parisi, Aurore Fraix, Stefano Guglielmo, Francesca Spyrakis, Barbara Rolando, Loretta Lazzarato, Roberta Fruttero, Alberto Gasco, Salvatore Sortino
Doxorubicin-antioxidant multitarget drugs 2013 K Chegaev; C Riganti; B Rolando; L Lazzarato; E Gazzano; S Guglielmo; D Ghigo; R Fruttero; A Gasco
EFFICIENTLY TARGETING DRUG EFFLUX THROUGH MODULATION OF P-GLYCOPROTEIN ACTIVITY BY SMALL MOLECULES: DESIGN, BIOLOGICAL AND COMPUTATIONAL STUDY. 2019 Stefano Guglielmo, Marialessandra Contino, Chiara Riganti, Barbara Rolando, Loretta Lazzarato
Furoxan nitric oxide donors disperse Pseudomonas aeruginosa biofilms, accelerate growth, and repress pyoverdine production 2017 Poh, Wee Han; Barraud, Nicolas; Guglielmo, Stefano; Lazzarato, Loretta; Fruttero, Roberta; Rolando, Barbara; Rice, Scott A.
Furoxan-, alkylnitrate-derivatives and related compoundsas anti-trypanosomatid agents: Mechanism of action studies 2008 Lucia Boiani; Gabriela Aguirre; Mercedes González; Hugo Cerecetto; Agustina Chidichimo; Juan J. Cazzulo; Massimo Bertinaria; Stefano Guglielmo
gem-Dinitroalkyl Benzenes: A Novel Class of IOP-Lowering Agents for the Treatment of Ocular Hypertension 2017 Blangetti, Marco; Rolando, Barbara; Marini, Elisabetta; Chegaev, Konstantin; Guglielmo, Stefano; Lazzarato, Loretta; Laura, Lucarini; Emanuela, Masini; Fruttero, Roberta
Hybrid praziquantel-oxadiazole oxides with activity against Schistosoma mansoni. 2011 Daniela Cortese; Francesca Vottero; Stefano Guglielmo; Roberta Fruttero; Alberto Gasco; Latasha Day and David L. Williams.
Leishmanicidal Activity of Novel Synthetic Furoxan and Benzofuroxan Derivatives 2014 L. A. Dutra;L. De Almeida;T. G. Passalacqua;J. S. Reis;F. A. E. Torres;I. Martinez;R. G. Peccinini;C. Man Chin;K. Chegaev;S. Guglielmo;R. Fruttero;M. A. S. Graminha;J. L. Dos Santos
Light-Tunable Generation of Singlet Oxygen and Nitric Oxide with a Bichromophoric Molecular Hybrid: a Bimodal Approach to Killing Cancer Cells 2016 Fraix, Aurore; Blangetti, Marco; Guglielmo, Stefano; Lazzarato, Loretta; Marino, Nino; Cardile, Venera; Graziano, Adriana C.E.; Manet, Ilse; Fruttero, Roberta; Gasco, Alberto; Sortino, Salvatore
Mitochondrial delivery of phenol substructure triggers mitochondrial depolarization and apoptosis of cancer cells 2018 Gazzano, Elena; Lazzarato, Loretta; Rolando, Barbara; Kopecka, Joanna; Guglielmo, Stefano; Costamagna, Costanzo; Chegaev, Konstantin*; Riganti, Chiara