GARCÍA JIMÉNEZ, DIEGO

GARCÍA JIMÉNEZ, DIEGO  

BIOTECNOLOGIE MOLECOLARI E SCIENZE PER LA SALUTE  

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Titolo Data di pubblicazione Autore(i) File
Chamelogk: A Chromatographic Chameleonicity Quantifier to Design Orally Bioavailable Beyond-Rule-of-5 Drugs 2023 GARCÍA JIMÉNEZ DIEGO; Vallaro Maura; Rossi Sebastiano Matteo; Apprato Giulia; D'Agostini Giulia; Rossetti Paolo; Ermondi Giuseppe; Caron Giulia
Conformational Sampling Deciphers the Chameleonic Properties of a VHL-Based Degrader 2023 Ermondi, Giuseppe; Jimenez, Diego Garcia; Rossi Sebastiano, Matteo; Kihlberg, Jan; Caron, Giulia
Designing Soluble PROTACs: Strategies and Preliminary Guidelines 2022 Diego García Jiménez; Matteo Rossi Sebastiano; Maura Vallaro; Valentina Mileo; Daniela Pizzirani; Elisa Moretti; Giuseppe Ermondi; Giulia Caron
PROTACs and Building Blocks: The 2D Chemical Space in Very Early Drug Discovery 2021 Giuseppe Ermondi, Diego Garcia Jimenez, Giulia Caron
Rational Control of Molecular Properties Is Mandatory to Exploit the Potential of PROTACs as Oral Drugs 2021 Ermondi, Giuseppe; Garcia Jimenez, Diego; Rossi Sebastiano, Matteo; Caron, Giulia
Refinement of Computational Access to Molecular Physicochemical Properties: From Ro5 to bRo5 2022 Rossi Sebastiano, Matteo; Garcia Jimenez, Diego; Vallaro, Maura; Caron, Giulia; Ermondi, Giuseppe