ROSSI SEBASTIANO, MATTEO
ROSSI SEBASTIANO, MATTEO
BIOTECNOLOGIE MOLECOLARI E SCIENZE PER LA SALUTE
ACSL3-PAI-1 signaling axis mediates tumor-stroma cross-talk promoting pancreatic cancer progression
2020-01-01 Sebastiano M.R.; Pozzato C.; Saliakoura M.; Yang Z.; Peng R.-W.; Galie M.; Oberson K.; Simon H.-U.; Karamitopoulou E.; Konstantinidou G.
AI-based protein structure databases have the potential to accelerate rare diseases research: AlphaFoldDB and the case of IAHSP/Alsin
2022-01-01 Rossi Sebastiano M.; Ermondi G.; Hadano S.; Caron G.
Are we ready to design oral PROTACs®?
2021-01-01 Jimenez D.G.; Sebastiano M.R.; Caron G.; Ermondi G.
Author Correction: Modeling ErbB2-p130Cas interaction to design new potential anticancer agents (Scientific Reports, (2019), 9, 1, (3089), 10.1038/s41598-019-39510-w)
2019-01-01 Costamagna A.; Rossi Sebastiano M.; Natalini D.; Simoni M.; Valabrega G.; Defilippi P.; Visentin S.; Ermondi G.; Turco E.; Caron G.; Cabodi S.
BBB-Permeable PROTACs: Where Do We Stand?
2026-01-01 Francisco, Serena; Apprato, Giulia; Rossi Sebastiano, Matteo; Ermondi, Giuseppe; Caron, Giulia
Chamelogk: A Chromatographic Chameleonicity Quantifier to Design Orally Bioavailable Beyond-Rule-of-5 Drugs
2023-01-01 GARCÍA JIMÉNEZ DIEGO; Vallaro Maura; Rossi Sebastiano Matteo; Apprato Giulia; D'Agostini Giulia; Rossetti Paolo; Ermondi Giuseppe; Caron Giulia
Conformational Sampling Deciphers the Chameleonic Properties of a VHL-Based Degrader
2023-01-01 Ermondi, Giuseppe; Jimenez, Diego Garcia; Rossi Sebastiano, Matteo; Kihlberg, Jan; Caron, Giulia
Dall’intelligenza artificiale nuove prospettive per la ricerca sulle malattie rare
2022-01-01 Matteo Rossi Sebastiano; Giuseppe Ermondi; Giulia Caron; Adriana Riccomagno
DegraderTCM: A Computationally Sparing Approach for Predicting Ternary Degradation Complexes
2024-01-01 Rossetti P.; Apprato G.; Caron G.; Ermondi G.; Rossi Sebastiano M.
Deleterious, protein-altering variants in the transcriptional coregulator ZMYM3 in 27 individuals with a neurodevelopmental delay phenotype
2023-01-01 Hiatt, Susan M; Trajkova, Slavica; Sebastiano, Matteo Rossi; Partridge, E Christopher; Abidi, Fatima E; Anderson, Ashlyn; Ansar, Muhammad; Antonarakis, Stylianos E; Azadi, Azadeh; Bachmann-Gagescu, Ruxandra; Bartuli, Andrea; Benech, Caroline; Berkowitz, Jennifer L; Betti, Michael J; Brusco, Alfredo; Cannon, Ashley; Caron, Giulia; Chen, Yanmin; Cochran, Meagan E; Coleman, Tanner F; Crenshaw, Molly M; Cuisset, Laurence; Curry, Cynthia J; Darvish, Hossein; Demirdas, Serwet; Descartes, Maria; Douglas, Jessica; Dyment, David A; Elloumi, Houda Zghal; Ermondi, Giuseppe; Faoucher, Marie; Farrow, Emily G; Felker, Stephanie A; Fisher, Heather; Hurst, Anna C E; Joset, Pascal; Kelly, Melissa A; Kmoch, Stanislav; Leadem, Benjamin R; Lyons, Michael J; Macchiaiolo, Marina; Magner, Martin; Mandrile, Giorgia; Mattioli, Francesca; McEown, Megan; Meadows, Sarah K; Medne, Livija; Meeks, Naomi J L; Montgomery, Sarah; Napier, Melanie P; Natowicz, Marvin; Newberry, Kimberly M; Niceta, Marcello; Noskova, Lenka; Nowak, Catherine B; Noyes, Amanda G; Osmond, Matthew; Prijoles, Eloise J; Pugh, Jada; Pullano, Verdiana; Quélin, Chloé; Rahimi-Aliabadi, Simin; Rauch, Anita; Redon, Sylvia; Reymond, Alexandre; Schwager, Caitlin R; Sellars, Elizabeth A; Scheuerle, Angela E; Shukarova-Angelovska, Elena; Skraban, Cara; Stolerman, Elliot; Sullivan, Bonnie R; Tartaglia, Marco; Thiffault, Isabelle; Uguen, Kevin; Umaña, Luis A; van Bever, Yolande; van der Crabben, Saskia N; van Slegtenhorst, Marjon A; Waisfisz, Quinten; Washington, Camerun; Rodan, Lance H; Myers, Richard M; Cooper, Gregory M
Designing Soluble PROTACs: Strategies and Preliminary Guidelines
2022-01-01 Diego García Jiménez; Matteo Rossi Sebastiano; Maura Vallaro; Valentina Mileo; Daniela Pizzirani; Elisa Moretti; Giuseppe Ermondi; Giulia Caron
DNA methylation analysis in patients with neurodevelopmental disorders improves variant interpretation and reveals complexity
2024-01-01 Trajkova, Slavica; Kerkhof, Jennifer; Rossi Sebastiano, Matteo; Pavinato, Lisa; Ferrero, Enza; Giovenino, Chiara; Carli, Diana; Di Gregorio, Eleonora; Marinoni, Roberta; Mandrile, Giorgia; Palermo, Flavia; Carestiato, Silvia; Cardaropoli, Simona; Pullano, Verdiana; Rinninella, Antonina; Giorgio, Elisa; Pippucci, Tommaso; Dimartino, Paola; Rzasa, Jessica; Rooney, Kathleen; McConkey, Haley; Petlichkovski, Aleksandar; Pasini, Barbara; Sukarova-Angelovska, Elena; Campbell, Christopher M; Metcalfe, Kay; Jenkinson, Sarah; Banka, Siddharth; Mussa, Alessandro; Ferrero, Giovanni Battista; Sadikovic, Bekim; Brusco, Alfredo
IMHB-Mediated Chameleonicity in Drug Design: A Focus on Structurally Related PROTACs
2024-01-01 Diego Garcia Jimenez; Matteo Rossi Sebastiano; Maura Vallaro; Giuseppe Ermondi; Giulia Caron
Impact of Dynamically Exposed Polarity on Permeability and Solubility of Chameleonic Drugs beyond the Rule of 5
2018-01-01 Rossi Sebastiano, Matteo; Doak, Bradley C.; Backlund, Maria; Poongavanam, Vasanthanathan; Over, Björn; Ermondi, Giuseppe; Caron, Giulia; Matsson, Pär*; Kihlberg, Jan
MK4 Repositioning for IAHSP: Overcoming In Vivo Data Gaps through In Silico Refinement and In Vitro Validation
2026-01-01 Rossi Sebastiano, Matteo; Vicidomini, Antonio; Francisco, Serena; Pullano, Verdiana; Defilippi, Paola; Baj, Gabriele; Cesca, Fabrizia; Caron, Giulia; Ermondi, Giuseppe
Modeling ErbB2-p130Cas interaction to design new potential anticancer agents.
2019-01-01 Andrea Costamagna, Matteo Rossi Sebastiano, Dora Natalini, Matilde Simoni, Giorgio Valabrega, Paola Defilippi, Sonja Visentin, Giuseppe Ermondi, Emilia Turco, Giulia Caron, Sara Cabodi
Personalized Treatment for Infantile Ascending Hereditary Spastic Paralysis Based on In Silico Strategies
2022-01-01 Rossi Sebastiano, Matteo; Ermondi, Giuseppe; Sato, Kai; Otomo, Asako; Hadano, Shinji; Caron, Giulia
PLCγ1 suppression promotes the adaptation of KRAS-mutant lung adenocarcinomas to hypoxia
2020-01-01 Saliakoura M.; Rossi Sebastiano M.; Pozzato C.; Heidel F.H.; Schnoder T.M.; Savic Prince S.; Bubendorf L.; Pinton P.; A. Schmid R.; Baumgartner J.; Freigang S.; Berezowska S.A.; Rimessi A.; Konstantinidou G.
Preclinical alternative drug discovery programs for monogenic rare diseases. Should small molecules or gene therapy be used? The case of hereditary spastic paraplegias
2024-01-01 Rossi Sebastiano, Matteo; Hadano, Shinji; Cesca, Fabrizia; Ermondi, Giuseppe; Caron, Giulia; Francisco, Serena; Brusco, Alfredo; Pullano, Verdiana; Chiantia, Giuseppe; Giustetto, Maurizio ; Baj, Gabriele; Della Vecchia, Stefania; Lamacchia, Lorenzo; Russo, Silvia; Higgins, Anna J.; van Putte, Wouter; Gurgone, Antonia
Rational Control of Molecular Properties Is Mandatory to Exploit the Potential of PROTACs as Oral Drugs
2021-01-01 Ermondi, Giuseppe; Garcia Jimenez, Diego; Rossi Sebastiano, Matteo; Caron, Giulia
| Titolo | Data di pubblicazione | Autore(i) | File |
|---|---|---|---|
| ACSL3-PAI-1 signaling axis mediates tumor-stroma cross-talk promoting pancreatic cancer progression | 2020 | Sebastiano M.R.; Pozzato C.; Saliakoura M.; Yang Z.; Peng R.-W.; Galie M.; Oberson K.; Simon H.-U.; Karamitopoulou E.; Konstantinidou G. | |
| AI-based protein structure databases have the potential to accelerate rare diseases research: AlphaFoldDB and the case of IAHSP/Alsin | 2022 | Rossi Sebastiano M.; Ermondi G.; Hadano S.; Caron G. | |
| Are we ready to design oral PROTACs®? | 2021 | Jimenez D.G.; Sebastiano M.R.; Caron G.; Ermondi G. | |
| Author Correction: Modeling ErbB2-p130Cas interaction to design new potential anticancer agents (Scientific Reports, (2019), 9, 1, (3089), 10.1038/s41598-019-39510-w) | 2019 | Costamagna A.; Rossi Sebastiano M.; Natalini D.; Simoni M.; Valabrega G.; Defilippi P.; Visentin S.; Ermondi G.; Turco E.; Caron G.; Cabodi S. | |
| BBB-Permeable PROTACs: Where Do We Stand? | 2026 | Francisco, Serena; Apprato, Giulia; Rossi Sebastiano, Matteo; Ermondi, Giuseppe; Caron, Giulia | |
| Chamelogk: A Chromatographic Chameleonicity Quantifier to Design Orally Bioavailable Beyond-Rule-of-5 Drugs | 2023 | GARCÍA JIMÉNEZ DIEGO; Vallaro Maura; Rossi Sebastiano Matteo; Apprato Giulia; D'Agostini Giulia; Rossetti Paolo; Ermondi Giuseppe; Caron Giulia | |
| Conformational Sampling Deciphers the Chameleonic Properties of a VHL-Based Degrader | 2023 | Ermondi, Giuseppe; Jimenez, Diego Garcia; Rossi Sebastiano, Matteo; Kihlberg, Jan; Caron, Giulia | |
| Dall’intelligenza artificiale nuove prospettive per la ricerca sulle malattie rare | 2022 | Matteo Rossi Sebastiano; Giuseppe Ermondi; Giulia Caron; Adriana Riccomagno | |
| DegraderTCM: A Computationally Sparing Approach for Predicting Ternary Degradation Complexes | 2024 | Rossetti P.; Apprato G.; Caron G.; Ermondi G.; Rossi Sebastiano M. | |
| Deleterious, protein-altering variants in the transcriptional coregulator ZMYM3 in 27 individuals with a neurodevelopmental delay phenotype | 2023 | Hiatt, Susan M; Trajkova, Slavica; Sebastiano, Matteo Rossi; Partridge, E Christopher; Abidi, Fatima E; Anderson, Ashlyn; Ansar, Muhammad; Antonarakis, Stylianos E; Azadi, Azadeh; Bachmann-Gagescu, Ruxandra; Bartuli, Andrea; Benech, Caroline; Berkowitz, Jennifer L; Betti, Michael J; Brusco, Alfredo; Cannon, Ashley; Caron, Giulia; Chen, Yanmin; Cochran, Meagan E; Coleman, Tanner F; Crenshaw, Molly M; Cuisset, Laurence; Curry, Cynthia J; Darvish, Hossein; Demirdas, Serwet; Descartes, Maria; Douglas, Jessica; Dyment, David A; Elloumi, Houda Zghal; Ermondi, Giuseppe; Faoucher, Marie; Farrow, Emily G; Felker, Stephanie A; Fisher, Heather; Hurst, Anna C E; Joset, Pascal; Kelly, Melissa A; Kmoch, Stanislav; Leadem, Benjamin R; Lyons, Michael J; Macchiaiolo, Marina; Magner, Martin; Mandrile, Giorgia; Mattioli, Francesca; McEown, Megan; Meadows, Sarah K; Medne, Livija; Meeks, Naomi J L; Montgomery, Sarah; Napier, Melanie P; Natowicz, Marvin; Newberry, Kimberly M; Niceta, Marcello; Noskova, Lenka; Nowak, Catherine B; Noyes, Amanda G; Osmond, Matthew; Prijoles, Eloise J; Pugh, Jada; Pullano, Verdiana; Quélin, Chloé; Rahimi-Aliabadi, Simin; Rauch, Anita; Redon, Sylvia; Reymond, Alexandre; Schwager, Caitlin R; Sellars, Elizabeth A; Scheuerle, Angela E; Shukarova-Angelovska, Elena; Skraban, Cara; Stolerman, Elliot; Sullivan, Bonnie R; Tartaglia, Marco; Thiffault, Isabelle; Uguen, Kevin; Umaña, Luis A; van Bever, Yolande; van der Crabben, Saskia N; van Slegtenhorst, Marjon A; Waisfisz, Quinten; Washington, Camerun; Rodan, Lance H; Myers, Richard M; Cooper, Gregory M | |
| Designing Soluble PROTACs: Strategies and Preliminary Guidelines | 2022 | Diego García Jiménez; Matteo Rossi Sebastiano; Maura Vallaro; Valentina Mileo; Daniela Pizzirani; Elisa Moretti; Giuseppe Ermondi; Giulia Caron | |
| DNA methylation analysis in patients with neurodevelopmental disorders improves variant interpretation and reveals complexity | 2024 | Trajkova, Slavica; Kerkhof, Jennifer; Rossi Sebastiano, Matteo; Pavinato, Lisa; Ferrero, Enza; Giovenino, Chiara; Carli, Diana; Di Gregorio, Eleonora; Marinoni, Roberta; Mandrile, Giorgia; Palermo, Flavia; Carestiato, Silvia; Cardaropoli, Simona; Pullano, Verdiana; Rinninella, Antonina; Giorgio, Elisa; Pippucci, Tommaso; Dimartino, Paola; Rzasa, Jessica; Rooney, Kathleen; McConkey, Haley; Petlichkovski, Aleksandar; Pasini, Barbara; Sukarova-Angelovska, Elena; Campbell, Christopher M; Metcalfe, Kay; Jenkinson, Sarah; Banka, Siddharth; Mussa, Alessandro; Ferrero, Giovanni Battista; Sadikovic, Bekim; Brusco, Alfredo | |
| IMHB-Mediated Chameleonicity in Drug Design: A Focus on Structurally Related PROTACs | 2024 | Diego Garcia Jimenez; Matteo Rossi Sebastiano; Maura Vallaro; Giuseppe Ermondi; Giulia Caron | |
| Impact of Dynamically Exposed Polarity on Permeability and Solubility of Chameleonic Drugs beyond the Rule of 5 | 2018 | Rossi Sebastiano, Matteo; Doak, Bradley C.; Backlund, Maria; Poongavanam, Vasanthanathan; Over, Björn; Ermondi, Giuseppe; Caron, Giulia; Matsson, Pär*; Kihlberg, Jan | |
| MK4 Repositioning for IAHSP: Overcoming In Vivo Data Gaps through In Silico Refinement and In Vitro Validation | 2026 | Rossi Sebastiano, Matteo; Vicidomini, Antonio; Francisco, Serena; Pullano, Verdiana; Defilippi, Paola; Baj, Gabriele; Cesca, Fabrizia; Caron, Giulia; Ermondi, Giuseppe | |
| Modeling ErbB2-p130Cas interaction to design new potential anticancer agents. | 2019 | Andrea Costamagna, Matteo Rossi Sebastiano, Dora Natalini, Matilde Simoni, Giorgio Valabrega, Paola Defilippi, Sonja Visentin, Giuseppe Ermondi, Emilia Turco, Giulia Caron, Sara Cabodi | |
| Personalized Treatment for Infantile Ascending Hereditary Spastic Paralysis Based on In Silico Strategies | 2022 | Rossi Sebastiano, Matteo; Ermondi, Giuseppe; Sato, Kai; Otomo, Asako; Hadano, Shinji; Caron, Giulia | |
| PLCγ1 suppression promotes the adaptation of KRAS-mutant lung adenocarcinomas to hypoxia | 2020 | Saliakoura M.; Rossi Sebastiano M.; Pozzato C.; Heidel F.H.; Schnoder T.M.; Savic Prince S.; Bubendorf L.; Pinton P.; A. Schmid R.; Baumgartner J.; Freigang S.; Berezowska S.A.; Rimessi A.; Konstantinidou G. | |
| Preclinical alternative drug discovery programs for monogenic rare diseases. Should small molecules or gene therapy be used? The case of hereditary spastic paraplegias | 2024 | Rossi Sebastiano, Matteo; Hadano, Shinji; Cesca, Fabrizia; Ermondi, Giuseppe; Caron, Giulia; Francisco, Serena; Brusco, Alfredo; Pullano, Verdiana; Chiantia, Giuseppe; Giustetto, Maurizio ; Baj, Gabriele; Della Vecchia, Stefania; Lamacchia, Lorenzo; Russo, Silvia; Higgins, Anna J.; van Putte, Wouter; Gurgone, Antonia | |
| Rational Control of Molecular Properties Is Mandatory to Exploit the Potential of PROTACs as Oral Drugs | 2021 | Ermondi, Giuseppe; Garcia Jimenez, Diego; Rossi Sebastiano, Matteo; Caron, Giulia |