VYAS, VIVEK KUMAR
VYAS, VIVEK KUMAR
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A comprehensive review of synthetic strategies and SAR studies for the discovery of PfDHODH inhibitors as antimalarial agents. Part 1: triazolopyrimidine, isoxazolopyrimidine and pyrrole-based (DSM) compounds
2024-01-01 Manmohan Sharma, Vinita Pandey, Giulio Poli, Tiziano Tuccinardi, Marco L. Lolli, Vivek K. Vyas
A comprehensive review of synthetic strategies and SAR studies for the discovery of PfDHODH inhibitors as antimalarial agents. Part 1: triazolopyrimidine, isoxazolopyrimidine and pyrrole-based (DSM) compounds
2024-01-01 Manmohan Sharma, Vinita Pandey, Giulio Poli, Tiziano Tuccinardi, Marco L. Lolli, Vivek K. Vyas
A comprehensive review of synthetic strategies and SAR studies for the discovery of PfDHODH inhibitors as antimalarial agents. Part 2: Non-DSM compounds
2024-01-01 Manmohan Sharma, Marco L. Lolli, Vivek K. Vyas
Novel benzophenone-, acetophenone-, and benzohydrazide-containing triazolopyrimidines as inhibitors of Plasmodium falciparum dihydroorotate dehydrogenase (PfDHODH): Design utilizing combined in silico approaches, synthesis, in vitro enzyme inhibition, and in vivo antimalarial activity
2025-01-01 Sharma, Manmohan; Pippione, Agnese Chiara; Tulsian, Kartik; Fornaseri, Federico; Giorgis, Marta; Boschi, Donatella; Buccinnà, Barbara; Ramondetti, Cristina; Lolli, Marco L.; Vyas, Vivek K.