BLUA, FEDERICA
BLUA, FEDERICA
SCIENZA E TECNOLOGIA DEL FARMACO
Chemical modulation of the 1-(Piperidin-4-yl)-1,3-dihydro-2h-benzo[d]imidazole-2-one scaffold as a novel NLRP3 inhibitor
2021-01-01 Gastaldi S.; Boscaro V.; Gianquinto E.; Sandall C.F.; Giorgis M.; Marini E.; Blua F.; Gallicchio M.; Spyrakis F.; Macdonald J.A.; Bertinaria M.
Comparative Study of Different H2S Donors as Vasodilators and Attenuators of Superoxide-Induced Endothelial Damage
2023-01-01 Marini E.; Rolando B.; Sodano F.; Blua F.; Concina G.; Guglielmo S.; Lazzarato L.; Chegaev K.
Design and synthesis of encorafenib-based BRAF-V600E degraders
2022-01-01 Federica Blua, Marco Marino, Simone Gastaldi, Federica Maione, Eleonora Gianquinto, Federica Di Nicolantonio, Massimo Bertinaria
Design and synthesis of SWIR emitters for optical imaging
2022-01-01 Federica Blua, Mariangela Boccalon, Barbara Rolando, Roberta Napolitano, Massimo Bertinaria
Design, synthesis and selection of INF200, a new non-sulfonylurea based NLRP3 inhibitor
2023-01-01 Federica Blua, Eleonora Gianquinto, Maria Concetta Granieri, Valentina Boscaro, Massimo Bertinaria
Development of pharmaceutical compounds intended for diagnostics applications - Exploring the SWIR region
2024-09-22
Discovery of a novel 1,3,4-oxadiazol-2-one-based NLRP3 inhibitor as a pharmacological agent to mitigate cardiac and metabolic complications in an experimental model of diet-induced metaflammation
2023-01-01 Gastaldi, Simone; Rocca, Carmine; Gianquinto, Eleonora; Granieri, Maria Concetta; Boscaro, Valentina; Blua, Federica; Rolando, Barbara; Marini, Elisabetta; Gallicchio, Margherita; De Bartolo, Anna; Romeo, Naomi; Mazza, Rosa; Fedele, Francesco; Pagliaro, Pasquale; Penna, Claudia; Spyrakis, Francesca; Bertinaria, Massimo; Angelone, Tommaso
Discovery of a septin-4 covalent binder with antimetastatic activity in a mouse model of melanoma
2024-01-01 Blua F.; Monge C.; Gastaldi S.; Clemente N.; Pizzimenti S.; Lazzarato L.; Senetta R.; Vittorio S.; Gigliotti C.L.; Boggio E.; Dianzani U.; Vistoli G.; Altomare A.A.; Aldini G.; Dianzani C.; Marini E.; Bertinaria M.
Exploiting the 2(1,3,4,9-tetrahydropyrano[3,4b]indol-1-yl)acetic Acid Scaffold to Generate COXTRANs: A New Class of Dual Cyclooxygenase Inhibitors-Thromboxane Receptor Antagonists
2025-01-01 Federica Blua; Francesca Boccato; Carola Buccellati; Patrizia Risè; Silvia Barbieri; Laura Castiglioni; Annika Balzulat; Barbara Rolando; Elisabetta Marini; Marta Balestra; Maria Luisa Introvigne; Marta Giorgis; Luigi Sironi; Stefania Tacconelli; Kerstin Hiesinger; Paola Patrignani; Achim Schmidtko; Dieter Steinhilber; Ewgenij Proschak; Angelo Sala; G Enrico Rovati; Massimo Bertinaria
Exploring flavylium-based SWIR emitters: Design, synthesis and optical characterization of dyes derivatized with polar moieties
2024-01-01 Blua, Federica; Boccalon, Mariangela; Rolando, Barbara; Napolitano, Roberta; Arena, Francesca; Blasi, Francesco; Bertinaria, Massimo
In the search for new NLRP3 inhibitors: chemical modulation of the 1-(piperidin-4-yl)-1,3-dihydro-2 Hbenzo[d]imidazole-2-one scaffold
2021-01-01 Simone Gastaldi, Valentina Boscaro, Eleonora Gianquinto, Christina F. Sandall, Marta Giorgis, Elisabetta Marini, Federica Blua, Margherita Gallicchio, Francesca Spyrakis, Justin A. MacDonald, Massimo Bertinaria
Inhibition of NLRP3 ATPase activity: a new strategy to fight chronic inflammatory diseases
2019-01-01 Simone Gastaldi, Federica Blua, Marta Giorgis, Elisabetta Marini, Massimo Bertinaria
Investigation into the Use of Encorafenib to Develop Potential PROTACs Directed against BRAFV600E Protein
2022-01-01 Marini, Elisabetta; Marino, Marco; Gionfriddo, Giulia; Maione, Federica; Pandini, Marta; Oddo, Daniele; Giorgis, Marta; Rolando, Barbara; Blua, Federica; Gastaldi, Simone; Marchiò, Serena; Kovachka, Sandra; Spyrakis, Francesca; Gianquinto, Eleonora; Di Nicolantonio, Federica; Bertinaria, Massimo
Macrophage and cardiomyocyte roles in cardioprotection: Exploiting the NLRP3 Inflammasome inhibitor INF150
2025-01-01 Giordano, Magalì; Femminò, Saveria; Blua, Federica; Boccato, Francesca; Rubeo, Chiara; Mantuano, Beatrice; Cioffi, Francesca; Comità, Stefano; Brovero, Arianna; Ciullo, Rosa; Bertinaria, Massimo; Penna, Claudia; Pagliaro, Pasquale
Modulation of the 2-(1,3,4,9-tetrahydropyrano[3,4-b]indol-1-yl)acetic acid scaffold to generate COXTRANs: a new class of dual cyclooxygenase inhibitors/thromboxane receptor antagonists
2025-01-01 F. Boccato, F. Blua, P. Patrignani, A. Sala, D. Steinhilber, A. Balzulat, A. Schimdtko, E. Marini, M. Bertinaria
Modulation of the aspartic acid scaffold to identify a new septin-4 covalent binder with anti-metastatic activity in a mouse model of melanoma
2024-01-01 F. Boccato, F. Blua, A. A. Altomare, S. Vittoriob, N. Clemente, C. Monge, E. Marini, M. Bertinaria
New inhibitors of NLRP3 inflammasome activation: pharmacological characterization in differentiated THP-1.
2022-01-01 Valentina Boscaro, Simone Gastaldi, Federica Blua, Massimo Bertinaria, Margherita Gallicchio
New non-sulfonylurea NLRP3 inhibitors: discovery and selection of INF200, a 1,3,4-oxadiazol-2-one-based NLRP3 inhibitor
2024-01-01 Alberto Gasparotto, Federica Blua, Maria Concetta Granieri, Eleonora Gianquinto, Valentina Boscaro, Massimo Bertinaria
NLRP3 inhibition protects human coronary endothelial cells from oxidative and lipotoxic stress
In corso di stampa Parenti, Astrid; Titi, Costanza; Brovero, Arianna; Blua, Federica; Boccato, Francesca; Silvano, Angela; Fedele, Francesco; Mattioli, Anna Vittoria; Bertinaria, Massimo; Pagliaro, Pasquale; Penna, Claudia
Novel NLRP3 inhibitor INF195: Low doses provide effective protection against myocardial ischemia/reperfusion injury
2024-01-01 Gastaldi, Simone; Giordano, Magalì; Blua, Federica; Rubeo, Chiara; Boscaro, Valentina; Femminò, Saveria; Comità, Stefano; Gianquinto, Eleonora; Landolfi, Vanessa; Marini, Elisabetta; Gallicchio, Margherita; Spyrakis, Francesca; Pagliaro, Pasquale; Bertinaria, Massimo; Penna, Claudia
| Titolo | Data di pubblicazione | Autore(i) | File |
|---|---|---|---|
| Chemical modulation of the 1-(Piperidin-4-yl)-1,3-dihydro-2h-benzo[d]imidazole-2-one scaffold as a novel NLRP3 inhibitor | 2021 | Gastaldi S.; Boscaro V.; Gianquinto E.; Sandall C.F.; Giorgis M.; Marini E.; Blua F.; Gallicchio M.; Spyrakis F.; Macdonald J.A.; Bertinaria M. | |
| Comparative Study of Different H2S Donors as Vasodilators and Attenuators of Superoxide-Induced Endothelial Damage | 2023 | Marini E.; Rolando B.; Sodano F.; Blua F.; Concina G.; Guglielmo S.; Lazzarato L.; Chegaev K. | |
| Design and synthesis of encorafenib-based BRAF-V600E degraders | 2022 | Federica Blua, Marco Marino, Simone Gastaldi, Federica Maione, Eleonora Gianquinto, Federica Di Nicolantonio, Massimo Bertinaria | |
| Design and synthesis of SWIR emitters for optical imaging | 2022 | Federica Blua, Mariangela Boccalon, Barbara Rolando, Roberta Napolitano, Massimo Bertinaria | |
| Design, synthesis and selection of INF200, a new non-sulfonylurea based NLRP3 inhibitor | 2023 | Federica Blua, Eleonora Gianquinto, Maria Concetta Granieri, Valentina Boscaro, Massimo Bertinaria | |
| Development of pharmaceutical compounds intended for diagnostics applications - Exploring the SWIR region | 2024 | - | |
| Discovery of a novel 1,3,4-oxadiazol-2-one-based NLRP3 inhibitor as a pharmacological agent to mitigate cardiac and metabolic complications in an experimental model of diet-induced metaflammation | 2023 | Gastaldi, Simone; Rocca, Carmine; Gianquinto, Eleonora; Granieri, Maria Concetta; Boscaro, Valentina; Blua, Federica; Rolando, Barbara; Marini, Elisabetta; Gallicchio, Margherita; De Bartolo, Anna; Romeo, Naomi; Mazza, Rosa; Fedele, Francesco; Pagliaro, Pasquale; Penna, Claudia; Spyrakis, Francesca; Bertinaria, Massimo; Angelone, Tommaso | |
| Discovery of a septin-4 covalent binder with antimetastatic activity in a mouse model of melanoma | 2024 | Blua F.; Monge C.; Gastaldi S.; Clemente N.; Pizzimenti S.; Lazzarato L.; Senetta R.; Vittorio S.; Gigliotti C.L.; Boggio E.; Dianzani U.; Vistoli G.; Altomare A.A.; Aldini G.; Dianzani C.; Marini E.; Bertinaria M. | |
| Exploiting the 2(1,3,4,9-tetrahydropyrano[3,4b]indol-1-yl)acetic Acid Scaffold to Generate COXTRANs: A New Class of Dual Cyclooxygenase Inhibitors-Thromboxane Receptor Antagonists | 2025 | Federica Blua; Francesca Boccato; Carola Buccellati; Patrizia Risè; Silvia Barbieri; Laura Castiglioni; Annika Balzulat; Barbara Rolando; Elisabetta Marini; Marta Balestra; Maria Luisa Introvigne; Marta Giorgis; Luigi Sironi; Stefania Tacconelli; Kerstin Hiesinger; Paola Patrignani; Achim Schmidtko; Dieter Steinhilber; Ewgenij Proschak; Angelo Sala; G Enrico Rovati; Massimo Bertinaria | |
| Exploring flavylium-based SWIR emitters: Design, synthesis and optical characterization of dyes derivatized with polar moieties | 2024 | Blua, Federica; Boccalon, Mariangela; Rolando, Barbara; Napolitano, Roberta; Arena, Francesca; Blasi, Francesco; Bertinaria, Massimo | |
| In the search for new NLRP3 inhibitors: chemical modulation of the 1-(piperidin-4-yl)-1,3-dihydro-2 Hbenzo[d]imidazole-2-one scaffold | 2021 | Simone Gastaldi, Valentina Boscaro, Eleonora Gianquinto, Christina F. Sandall, Marta Giorgis, Elisabetta Marini, Federica Blua, Margherita Gallicchio, Francesca Spyrakis, Justin A. MacDonald, Massimo Bertinaria | |
| Inhibition of NLRP3 ATPase activity: a new strategy to fight chronic inflammatory diseases | 2019 | Simone Gastaldi, Federica Blua, Marta Giorgis, Elisabetta Marini, Massimo Bertinaria | |
| Investigation into the Use of Encorafenib to Develop Potential PROTACs Directed against BRAFV600E Protein | 2022 | Marini, Elisabetta; Marino, Marco; Gionfriddo, Giulia; Maione, Federica; Pandini, Marta; Oddo, Daniele; Giorgis, Marta; Rolando, Barbara; Blua, Federica; Gastaldi, Simone; Marchiò, Serena; Kovachka, Sandra; Spyrakis, Francesca; Gianquinto, Eleonora; Di Nicolantonio, Federica; Bertinaria, Massimo | |
| Macrophage and cardiomyocyte roles in cardioprotection: Exploiting the NLRP3 Inflammasome inhibitor INF150 | 2025 | Giordano, Magalì; Femminò, Saveria; Blua, Federica; Boccato, Francesca; Rubeo, Chiara; Mantuano, Beatrice; Cioffi, Francesca; Comità, Stefano; Brovero, Arianna; Ciullo, Rosa; Bertinaria, Massimo; Penna, Claudia; Pagliaro, Pasquale | |
| Modulation of the 2-(1,3,4,9-tetrahydropyrano[3,4-b]indol-1-yl)acetic acid scaffold to generate COXTRANs: a new class of dual cyclooxygenase inhibitors/thromboxane receptor antagonists | 2025 | F. Boccato, F. Blua, P. Patrignani, A. Sala, D. Steinhilber, A. Balzulat, A. Schimdtko, E. Marini, M. Bertinaria | |
| Modulation of the aspartic acid scaffold to identify a new septin-4 covalent binder with anti-metastatic activity in a mouse model of melanoma | 2024 | F. Boccato, F. Blua, A. A. Altomare, S. Vittoriob, N. Clemente, C. Monge, E. Marini, M. Bertinaria | |
| New inhibitors of NLRP3 inflammasome activation: pharmacological characterization in differentiated THP-1. | 2022 | Valentina Boscaro, Simone Gastaldi, Federica Blua, Massimo Bertinaria, Margherita Gallicchio | |
| New non-sulfonylurea NLRP3 inhibitors: discovery and selection of INF200, a 1,3,4-oxadiazol-2-one-based NLRP3 inhibitor | 2024 | Alberto Gasparotto, Federica Blua, Maria Concetta Granieri, Eleonora Gianquinto, Valentina Boscaro, Massimo Bertinaria | |
| NLRP3 inhibition protects human coronary endothelial cells from oxidative and lipotoxic stress | In corso di stampa | Parenti, Astrid; Titi, Costanza; Brovero, Arianna; Blua, Federica; Boccato, Francesca; Silvano, Angela; Fedele, Francesco; Mattioli, Anna Vittoria; Bertinaria, Massimo; Pagliaro, Pasquale; Penna, Claudia | |
| Novel NLRP3 inhibitor INF195: Low doses provide effective protection against myocardial ischemia/reperfusion injury | 2024 | Gastaldi, Simone; Giordano, Magalì; Blua, Federica; Rubeo, Chiara; Boscaro, Valentina; Femminò, Saveria; Comità, Stefano; Gianquinto, Eleonora; Landolfi, Vanessa; Marini, Elisabetta; Gallicchio, Margherita; Spyrakis, Francesca; Pagliaro, Pasquale; Bertinaria, Massimo; Penna, Claudia |