RicercaInizia una nuova ricerca
NOTA: è possibile cercare una corrispondenza esatta usando i doppi apici, ad es: "evoluzione della specie". Qualora si cerchi un identificativo, è consigliabile cercarlo in due modi differenti: tra apici con caratteri speciali es: "978-94-6366-274" oppure senza caratteri speciali solo come sequenza numerica: es 978946366274.
Optimization of MEDS433 synthesis: scale-up for preclinical evaluation studies
2023-01-01 Iole Mannella, Chiara Vigato, Stefano Sainas, Marco Lucio Lolli, Donatella Boschi
Preliminary ADME/PK studies of new hDHODH inhibitors effective for treatment of acute myeloid leukaemia (AML)
2019-01-01 Giulia De Simone, Stefano Sainas, Marilena Marraudino, Agnese Chiara Pippione, Brigitta Bonaldo, Alice Passoni, Marta Giorgis, Barbara Rolando, Donatella Boschi, Marco Lucio Lolli
Probing the bicyclic hydroxypyrazolo[1,5-a]pyridine scaffold as a carboxylic acid bioisostere in theGABAA receptor system
2012-01-01 A. Ducime; B. Nielsen; B. Frølund; M. L. Lolli
Synthesis and Structural Characterization of Regio Substituted 4-Hydroxy-1H-1,2,3-triazols as Possible Tool in Bioisosteric Applications
2014-01-01 A Federico; S.Sainas; A. Ducime;K. Martina; F. Bosca; D. Boschi; M.L. Lolli.
Synthesis of [18F]Brequinar as PET Imaging probes for human dihydroorotate dehydrogenase
2019-01-01 Elena Martino, Stefano Sainas, Agnese C. Pippione, Donatella Boschi, Yu- Shin Ding, Marco L. Lolli
Synthesis of new gadolinium complexes for magnetic resonance imaging with improved relaxivity
2017-01-01 Carnovale, I. M.; Colombo Serra, S.; Fringuello Mingo, A.; Lattuada, L.; Lolli, M. L.
Synthesis of new Gadolinium complexes for magnetic resonance imaging with improved relaxivity
2017-01-01 Carnovale, Irene Maria; Serra, Sonia Colombo; Fringuello Mingo, Alberto; Lattuada, Luciano; Lolli, Marco Lucio
Synthesis of new Plasmodium Falciparum dihydroorotate dehydrogenase inhibitors through the application of an isosteric portfolio
2013-01-01 Pippione A. C.;1 Federico A.;1 Boschi D.;S.2 Lolli M. L.1
Targeting Castration Resistant Prostate Cancer (CRPC) by innovative AKR1C3 inhibitors based on the 3-hydroxybenzoisoxazole structure
2016-01-01 Carnovale, Irene Maria; Pippione, Agnese Chiara; Giraudo, Alessandro; Federico, Antonella; Zorniotti, Sonia; Simonetta Oliaro Bosso, ; Ferrante, Terenzio; Marini, Elisabetta; Pors, Klaus; Braga, Rodolpho Campos; Boschi, Donatella; Lucio Lolli, Marco
Targeting myeloid differentiation using potent human dihydroorotate dehydrogenase (hDHODH) inhibitors
2018-01-01 Sainas Stefano, Pippione Agnese Chiara, Bonanni Davide, Giorgis Marta, Lupino Elisa, Giraudo Enrico, Goyal Parveen, Circosta Paola, Gaidano Valentina, Cignetti Alessandro, Piccinini Marco, Friemann Rosmarie, Saglio Giuseppe, Al-Karadaghi Salam, Boschi Donatella, Lolli Marco Lucio
| Titolo | Data di pubblicazione | Autore(i) | File |
|---|---|---|---|
| Optimization of MEDS433 synthesis: scale-up for preclinical evaluation studies | 2023 | Iole Mannella, Chiara Vigato, Stefano Sainas, Marco Lucio Lolli, Donatella Boschi | |
| Preliminary ADME/PK studies of new hDHODH inhibitors effective for treatment of acute myeloid leukaemia (AML) | 2019 | Giulia De Simone, Stefano Sainas, Marilena Marraudino, Agnese Chiara Pippione, Brigitta Bonaldo, Alice Passoni, Marta Giorgis, Barbara Rolando, Donatella Boschi, Marco Lucio Lolli | |
| Probing the bicyclic hydroxypyrazolo[1,5-a]pyridine scaffold as a carboxylic acid bioisostere in theGABAA receptor system | 2012 | A. Ducime; B. Nielsen; B. Frølund; M. L. Lolli | |
| Synthesis and Structural Characterization of Regio Substituted 4-Hydroxy-1H-1,2,3-triazols as Possible Tool in Bioisosteric Applications | 2014 | A Federico; S.Sainas; A. Ducime;K. Martina; F. Bosca; D. Boschi; M.L. Lolli. | |
| Synthesis of [18F]Brequinar as PET Imaging probes for human dihydroorotate dehydrogenase | 2019 | Elena Martino, Stefano Sainas, Agnese C. Pippione, Donatella Boschi, Yu- Shin Ding, Marco L. Lolli | |
| Synthesis of new gadolinium complexes for magnetic resonance imaging with improved relaxivity | 2017 | Carnovale, I. M.; Colombo Serra, S.; Fringuello Mingo, A.; Lattuada, L.; Lolli, M. L. | |
| Synthesis of new Gadolinium complexes for magnetic resonance imaging with improved relaxivity | 2017 | Carnovale, Irene Maria; Serra, Sonia Colombo; Fringuello Mingo, Alberto; Lattuada, Luciano; Lolli, Marco Lucio | |
| Synthesis of new Plasmodium Falciparum dihydroorotate dehydrogenase inhibitors through the application of an isosteric portfolio | 2013 | Pippione A. C.;1 Federico A.;1 Boschi D.;S.2 Lolli M. L.1 | |
| Targeting Castration Resistant Prostate Cancer (CRPC) by innovative AKR1C3 inhibitors based on the 3-hydroxybenzoisoxazole structure | 2016 | Carnovale, Irene Maria; Pippione, Agnese Chiara; Giraudo, Alessandro; Federico, Antonella; Zorniotti, Sonia; Simonetta Oliaro Bosso, ; Ferrante, Terenzio; Marini, Elisabetta; Pors, Klaus; Braga, Rodolpho Campos; Boschi, Donatella; Lucio Lolli, Marco | |
| Targeting myeloid differentiation using potent human dihydroorotate dehydrogenase (hDHODH) inhibitors | 2018 | Sainas Stefano, Pippione Agnese Chiara, Bonanni Davide, Giorgis Marta, Lupino Elisa, Giraudo Enrico, Goyal Parveen, Circosta Paola, Gaidano Valentina, Cignetti Alessandro, Piccinini Marco, Friemann Rosmarie, Saglio Giuseppe, Al-Karadaghi Salam, Boschi Donatella, Lolli Marco Lucio |
Legenda icone
- file ad accesso aperto
- file disponibili sulla rete interna
- file disponibili agli utenti autorizzati
- file disponibili solo agli amministratori
- file sotto embargo
- nessun file disponibile
Opzioni
Scopri
Tipologia
- 04-CONTRIBUTO IN ATTI DI CONVEGNO 49
- 04-CONTRIBUTO IN ATTI DI CONVEGNO... 49
Data di pubblicazione
- 2020 - 2023 15
- 2012 - 2019 34
Keyword
- bioisosterism 2
- 17β-HSD5 1
- 1H-pyrazole-4-carboxylic acid 1
- AKR1C3 1
- Aldo-keto reductase 1C3 1
- bioisterism 1
- CRPC 1
- hydroxylated heterocyclic 1
- hydroxylated pentatomic heterocyclic 1
- IkB kinase 1
Lingua
- eng 47
- enm 2
Accesso al fulltext
- reserved 24
- no fulltext 16
- open 9