Valorisation of waste by-products from olive pomace industry by using black soldier fly larvae as bioconverter
2022-01-01 G.I. Ascrizzi, F. Grosso, R. Fortina, M. Meneguz
Confronto tra epidurale toracica vs morfina spinale in cani sottoposti a chirurgia toracica e dell'addome craniale
2022-01-01 Lardone E, Sarotti D, Franci P
HSC transplant: role of amino acid substitutions in antigen binding sites
2022-01-01 D. Bongioanni, F.E. Bertinetto, N.M. Ferrero, E. Garino, A. Giordano, P. Magistroni, G.A. Mazzola, T. Melchiorre, A. De Masi, L. Rocchi, C.M. Dellacasa, L. Giaccone, I. Dogliotti, S. Deaglio, A. Busca, A. Amoroso
Targeting PAD-mediated citrullination to treat human papillomavirus infections
2021-01-01 CAMILLA ALBANO, MATTEO BIOLATTI, SELINA PASQUERO, FRANCESCA GUGLIESI, SERGIO F. CASTILLO PACHECO, GLORIA GRIFFANTE, ELENA CAT GENOVA, IRENE LO CIGNO, MARISA GARIGLIO, MARCO DE ANDREA, SANTO LANDOLFO, JASENKA MAZIBRADA, VALENTINA DELL’OSTE
Targeting myeloid leukemias using human Dihydroorotate Dehydrogenase inhibitors based on 2-hydroxypyrazolo[1,5-a]pyridine scaffold: overcoming of metabolic issues
2021-01-01 Chiara Vigato, Stefano Sainas, Marta Giorgis, Paola Circosta, Alice Passoni, Agnese Chiara Pippione, Renzo Bagnati, Giuseppe Saglio, Donatella Boschi, Marco Lucio Lolli.
A new pro-apoptotic therapy for Acute Myeloid Leukaemia using MEDS433, a potent human Dihydroorotate Dehydrogenase inhibitor
2021-01-01 Sainas Sainas, Paola Circosta, Noemi Villella, Elena Martino, Agnese Chiara Pippione, Mohammad Houshmand, Marta Giorgis, Valentina Gaidano, Alessandro Cignetti, Caterina Peraldo Neia, Giovanna Chiorino, Salam Al-Karadaghi, Donatella Boschi, Giuseppe Saglio, Marco Lucio Lolli.
A differentiating and apoptotic therapy for Acute Myeloid Leukaemia using MEDS433, a potent human Dihydroorotate Dehydrogenase inhibitor
2021-01-01 Stefano Sainas, Paola Circosta, Marta Giorgis, Agnese Chiara Pippione, Marilena Marraudino, Mohammad Houshmand, Brigitta Bonaldo, Valentina Gaidano, Alessandro Cignetti, Stefano Gotti, Giuseppe Saglio, Salam Al-Karadaghi, Donatella Boschi, Marco Lucio Lolli
Design and synthesis of a library of pyrazolo[1,5-a]pyridine fluorophores for developing new fluorescent probes
2021-01-01 Elena Martino, Stefano Sainas, Francesco Bavo, Claudio Garino, Donatella Boschi, Bente Frølund, Marco Lucio Lolli
Multiple-targeting ligands for AKR1C3 enzyme and androgen receptor to target prostate cancer
2021-01-01 Agnese Chiara Pippione, Zuhal Kilic-Kurt, Stefano Sainas, Iole Mannella, Barbara Rolando, Sandra Kovachka, Francesca Spyrakis, Annamaria Buschini, Serena Montalbano, Simonetta Oliaro Bosso, Marco Lolli, Donatella Boschi
Improvement of metabolic weakness of new human Dihydroorotate Dehydrogenase inhibitors based on 2-hydroxypyrazolo[1,5-a]pyridine scaffold
2021-01-01 Chiara Vigato, Stefano Sainas, Marta Giorgis, Paola Circosta, Alice Passoni, Agnese Chiara Pippione, Renzo Bagnati, Giuseppe Saglio, Donatella Boschi, Marco Lucio Lolli
Design of new human Dihydroorotate Dehydrogenase inhibitors: amide bioisosterism in MEDS433 optimization
2021-01-01 Martino, Elena; Villella, Noemi;Vigato, Chiara; Cerrina, Matteo; Bersani, Matteo; Giorgis Marta, Sainas, Stefano.; Boschi, Donatella; Lolli, Marco Lucio
New inhibitors of Aldo-Keto Reductase 1C3 (AKR1C3) based on benzoisoxazole scaffold and their potential application in cancer
2021-01-01 Mannella, Iole, Vigato, Chiara, Pasha, Rabia; Pippione Agnese Chiara, Sainas, Stefano, Oliaro Bosso Simonetta; Rolando, Barbara; Kovachka, Sandra, Spyrakis, Francesca; Boschi, Donatella, Lolli. Marco Lucio
Synthesis of [18F]Brequinar as PET Imaging probes for human dihydroorotate dehydrogenase
2019-01-01 Elena Martino, Stefano Sainas, Agnese C. Pippione, Donatella Boschi, Yu- Shin Ding, Marco L. Lolli
Preliminary ADME/PK studies of new hDHODH inhibitors effective for treatment of acute myeloid leukaemia (AML)
2019-01-01 Giulia De Simone, Stefano Sainas, Marilena Marraudino, Agnese Chiara Pippione, Brigitta Bonaldo, Alice Passoni, Marta Giorgis, Barbara Rolando, Donatella Boschi, Marco Lucio Lolli
Design, synthesis and co-crystallization of new Plasmodium falciparum dihydroorotate dehydrogenase inhibitors based on hydroxypyrazole scaffold
2019-01-01 Noemi Villella, Agnese Chiara Pippione, Stefano Sainas, Donatella Boschi, Rosmarie Friemann, Alberto Gimenéz, Efrain Salamanca, Marco Lucio Lolli
Targeting the human Dihydroorotate Dehydrogenase (hDHODH) by a Scaffold Hopping Bioisosteric approach using Hydroxylated Pentatomic Heterocycles
2016-01-01 Stefano Sainas, Agnese Chiara Pippione, Irene Maria Carnovale, Alessandro Giraudo, Marta Giorgis, Rodolpho B. Braga, Carolina H. Andrade, Noemi Villella, Marco Piccinini, Elisa Lupino, Rosmarie Friemann, Salam Al-Kadaraghi, Donatella Boschi, Marco L. Lolli
Antileishmanial activity of some 4-phenyl-3-amino-1H-pyrazols designed as CRK3 kinase inhibitors
2016-01-01 Agnese Chiara Pippione, Piermichele Kobauri, Stefano Sainas, Alberto Gimenez, Antonella Federico, Rodolpho Campos Braga, Carolina Horta Andrade, Donatella Boschi, Efrain Salamanca, Juan Carlos Ticona, Marco Lucio Lolli
Toward a Bioisosteric Alkahest: Targeting the human Dihydroorotate Dehydrogenase (hDHODH) by a Scaffold Hopping Bioisosteric approach using Hydroxylated Pentatomic Heterocycles
2015-01-01 Marco L. Lolli, Agnese Chiara Pippione, Stefano Sainas, Stefano Mensa, Marta Giorgis, Marco Piccinini, Elisa Lupino, Salam Al-Kadaraghi, Donatella Boschi
Fatal Asphyxia by Bolus in Elders With Mental Illness: The Role of Oral Health and Antimuscarinic Action of Drug Treatment
2017-01-01 Aquila I; Di Nunzio C; Nuzzolese E; Ricci P
The impact of Workshop in Forensic Odontology in Human Rights Workshop in the United Arab Emirates
2019-01-01 Salem Altalie, Emilio Nuzzolese, Joe Adserias-Garriga, Alexander S. Forrest,
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
Valorisation of waste by-products from olive pomace industry by using black soldier fly larvae as bioconverter | 2022 | G.I. Ascrizzi, F. Grosso, R. Fortina, M. Meneguz | |
Confronto tra epidurale toracica vs morfina spinale in cani sottoposti a chirurgia toracica e dell'addome craniale | 2022 | Lardone E, Sarotti D, Franci P | |
HSC transplant: role of amino acid substitutions in antigen binding sites | 2022 | D. Bongioanni, F.E. Bertinetto, N.M. Ferrero, E. Garino, A. Giordano, P. Magistroni, G.A. Mazzola, T. Melchiorre, A. De Masi, L. Rocchi, C.M. Dellacasa, L. Giaccone, I. Dogliotti, S. Deaglio, A. Busca, A. Amoroso | |
Targeting PAD-mediated citrullination to treat human papillomavirus infections | 2021 | CAMILLA ALBANO, MATTEO BIOLATTI, SELINA PASQUERO, FRANCESCA GUGLIESI, SERGIO F. CASTILLO PACHECO, GLORIA GRIFFANTE, ELENA CAT GENOVA, IRENE LO CIGNO, MARISA GARIGLIO, MARCO DE ANDREA, SANTO LANDOLFO, JASENKA MAZIBRADA, VALENTINA DELL’OSTE | |
Targeting myeloid leukemias using human Dihydroorotate Dehydrogenase inhibitors based on 2-hydroxypyrazolo[1,5-a]pyridine scaffold: overcoming of metabolic issues | 2021 | Chiara Vigato, Stefano Sainas, Marta Giorgis, Paola Circosta, Alice Passoni, Agnese Chiara Pippione, Renzo Bagnati, Giuseppe Saglio, Donatella Boschi, Marco Lucio Lolli. | |
A new pro-apoptotic therapy for Acute Myeloid Leukaemia using MEDS433, a potent human Dihydroorotate Dehydrogenase inhibitor | 2021 | Sainas Sainas, Paola Circosta, Noemi Villella, Elena Martino, Agnese Chiara Pippione, Mohammad Houshmand, Marta Giorgis, Valentina Gaidano, Alessandro Cignetti, Caterina Peraldo Neia, Giovanna Chiorino, Salam Al-Karadaghi, Donatella Boschi, Giuseppe Saglio, Marco Lucio Lolli. | |
A differentiating and apoptotic therapy for Acute Myeloid Leukaemia using MEDS433, a potent human Dihydroorotate Dehydrogenase inhibitor | 2021 | Stefano Sainas, Paola Circosta, Marta Giorgis, Agnese Chiara Pippione, Marilena Marraudino, Mohammad Houshmand, Brigitta Bonaldo, Valentina Gaidano, Alessandro Cignetti, Stefano Gotti, Giuseppe Saglio, Salam Al-Karadaghi, Donatella Boschi, Marco Lucio Lolli | |
Design and synthesis of a library of pyrazolo[1,5-a]pyridine fluorophores for developing new fluorescent probes | 2021 | Elena Martino, Stefano Sainas, Francesco Bavo, Claudio Garino, Donatella Boschi, Bente Frølund, Marco Lucio Lolli | |
Multiple-targeting ligands for AKR1C3 enzyme and androgen receptor to target prostate cancer | 2021 | Agnese Chiara Pippione, Zuhal Kilic-Kurt, Stefano Sainas, Iole Mannella, Barbara Rolando, Sandra Kovachka, Francesca Spyrakis, Annamaria Buschini, Serena Montalbano, Simonetta Oliaro Bosso, Marco Lolli, Donatella Boschi | |
Improvement of metabolic weakness of new human Dihydroorotate Dehydrogenase inhibitors based on 2-hydroxypyrazolo[1,5-a]pyridine scaffold | 2021 | Chiara Vigato, Stefano Sainas, Marta Giorgis, Paola Circosta, Alice Passoni, Agnese Chiara Pippione, Renzo Bagnati, Giuseppe Saglio, Donatella Boschi, Marco Lucio Lolli | |
Design of new human Dihydroorotate Dehydrogenase inhibitors: amide bioisosterism in MEDS433 optimization | 2021 | Martino, Elena; Villella, Noemi;Vigato, Chiara; Cerrina, Matteo; Bersani, Matteo; Giorgis Marta, Sainas, Stefano.; Boschi, Donatella; Lolli, Marco Lucio | |
New inhibitors of Aldo-Keto Reductase 1C3 (AKR1C3) based on benzoisoxazole scaffold and their potential application in cancer | 2021 | Mannella, Iole, Vigato, Chiara, Pasha, Rabia; Pippione Agnese Chiara, Sainas, Stefano, Oliaro Bosso Simonetta; Rolando, Barbara; Kovachka, Sandra, Spyrakis, Francesca; Boschi, Donatella, Lolli. Marco Lucio | |
Synthesis of [18F]Brequinar as PET Imaging probes for human dihydroorotate dehydrogenase | 2019 | Elena Martino, Stefano Sainas, Agnese C. Pippione, Donatella Boschi, Yu- Shin Ding, Marco L. Lolli | |
Preliminary ADME/PK studies of new hDHODH inhibitors effective for treatment of acute myeloid leukaemia (AML) | 2019 | Giulia De Simone, Stefano Sainas, Marilena Marraudino, Agnese Chiara Pippione, Brigitta Bonaldo, Alice Passoni, Marta Giorgis, Barbara Rolando, Donatella Boschi, Marco Lucio Lolli | |
Design, synthesis and co-crystallization of new Plasmodium falciparum dihydroorotate dehydrogenase inhibitors based on hydroxypyrazole scaffold | 2019 | Noemi Villella, Agnese Chiara Pippione, Stefano Sainas, Donatella Boschi, Rosmarie Friemann, Alberto Gimenéz, Efrain Salamanca, Marco Lucio Lolli | |
Targeting the human Dihydroorotate Dehydrogenase (hDHODH) by a Scaffold Hopping Bioisosteric approach using Hydroxylated Pentatomic Heterocycles | 2016 | Stefano Sainas, Agnese Chiara Pippione, Irene Maria Carnovale, Alessandro Giraudo, Marta Giorgis, Rodolpho B. Braga, Carolina H. Andrade, Noemi Villella, Marco Piccinini, Elisa Lupino, Rosmarie Friemann, Salam Al-Kadaraghi, Donatella Boschi, Marco L. Lolli | |
Antileishmanial activity of some 4-phenyl-3-amino-1H-pyrazols designed as CRK3 kinase inhibitors | 2016 | Agnese Chiara Pippione, Piermichele Kobauri, Stefano Sainas, Alberto Gimenez, Antonella Federico, Rodolpho Campos Braga, Carolina Horta Andrade, Donatella Boschi, Efrain Salamanca, Juan Carlos Ticona, Marco Lucio Lolli | |
Toward a Bioisosteric Alkahest: Targeting the human Dihydroorotate Dehydrogenase (hDHODH) by a Scaffold Hopping Bioisosteric approach using Hydroxylated Pentatomic Heterocycles | 2015 | Marco L. Lolli, Agnese Chiara Pippione, Stefano Sainas, Stefano Mensa, Marta Giorgis, Marco Piccinini, Elisa Lupino, Salam Al-Kadaraghi, Donatella Boschi | |
Fatal Asphyxia by Bolus in Elders With Mental Illness: The Role of Oral Health and Antimuscarinic Action of Drug Treatment | 2017 | Aquila I; Di Nunzio C; Nuzzolese E; Ricci P | |
The impact of Workshop in Forensic Odontology in Human Rights Workshop in the United Arab Emirates | 2019 | Salem Altalie, Emilio Nuzzolese, Joe Adserias-Garriga, Alexander S. Forrest, |
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Scopri
Tipologia
- 04-CONTRIBUTO IN ATTI DI CONVEGNO1694
Data di pubblicazione
- In corso di stampa1
- 2020 - 2022107
- 2010 - 20191397
- 2000 - 2009188
- 1997 - 19991
Keyword
- KCC22
- midollo spinale2
- nocicezione2
- sinapsi GABAergiche2
- storia della cartografia2
- acute hospital psychiatric ward1
- ADAPTED TRAINING1
- african grey parrot1
- aggressivenes1
- aggressività1
Lingua
- eng1462
- ita227
- spa5
- fra4
- enm3
Accesso al fulltext
- no fulltext918
- open554
- reserved191
- restricted18
- partially open10
- mixed3