Sfoglia per Autore
New lipophilic organic nitrates: Candidates for chronic skin disease therapy
2023-01-01 Marini E.; Sodano F.; Rolando B.; Chegaev K.; Maresca D.C.; Ianaro A.; Ercolano G.; Lazzarato L.
Use of Enzymatically Activated Carbon Monoxide Donors for Sensitizing Drug-Resistant Tumor Cells
2023-01-01 Sodano, Federica; Rolando, Barbara; Lazzarato, Loretta; Costamagna, Costanzo; Failla, Mariacristina; Riganti, Chiara; Chegaev, Konstantin
Comparative Study of Different H2S Donors as Vasodilators and Attenuators of Superoxide-Induced Endothelial Damage
2023-01-01 Marini E.; Rolando B.; Sodano F.; Blua F.; Concina G.; Guglielmo S.; Lazzarato L.; Chegaev K.
Multitarget antioxidant NO-donor organic nitrates: a novel approach to overcome nitrates tolerance
2022-01-01 Elisabetta Marini, Marta Giorgis, Barbara Rolando, Konstantin Chegaev
A Comprehensive Evaluation of Sdox, a Promising H2S-Releasing Doxorubicin for the Treatment of Chemoresistant Tumors
2022-01-01 Alov P.; Al Sharif M.; Aluani D.; Chegaev K.; Dinic J.; Divac Rankov A.; Fernandes M.X.; Fusi F.; Garcia-Sosa A.T.; Juvonen R.; Kondeva-Burdina M.; Padron J.M.; Pajeva I.; Pencheva T.; Puerta A.; Raunio H.; Riganti C.; Tsakovska I.; Tzankova V.; Yordanov Y.; Saponara S.
N-[1,3-Dialkyl(aryl)-2-oxoimidazolidin-4-ylidene]-aryl(alkyl)sulphonamides as Novel Selective Human Cannabinoid Type 2 Receptor (hCB2R) Ligands; Insights into the Mechanism of Receptor Activation/Deactivation
2022-01-01 Gianquinto, Eleonora; Sodano, Federica; Rolando, Barbara; Kostrzewa, Magdalena; Allarà, Marco; Mahmoud, Ali Mokhtar; Kumar, Poulami; Spyrakis, Francesca; Ligresti, Alessia; Chegaev, Konstantin
Multitarget antioxidant NO-donor organic nitrates: a novel ap-proach to overcome nitrates tolerance, an ex vivo study
2022-01-01 Elisabetta Marini*, Marta Giorgis, Marta Leporati, Barbara Rolando, Konstantin Chegaev, Loretta Lazzarato, Massimo Bertinaria, Marco Vincenti, Antonella Di Stilo
Naked and Decorated Nanoparticles Containing H2S-Releasing Doxorubicin: Preparation, Characterization and Assessment of Their Antitumoral Efficiency on Various Resistant Tumor Cells
2022-01-01 Elena PEIRA; Daniela Chirio; Simona Sapino; Konstantin CHEGAEV; Giulia Chindamo; IRIS CHIARA SALAROGLIO; Chiara Riganti; Marina GALLARATE
Sdox, a H2S releasing anthracycline, with a safer profile than doxorubicin toward vasculature
2022-01-01 Durante M, Frosini M, Chiaino E, Fusi F, Gamberucci A, Gorelli B, Chegaev K, Riganti C, Saponara S
In vitro vascular toxicity assessment of NitDOX, a novel NO-releasing doxorubicin
2020-01-01 Durante M.; Frosini M.; Fusi F.; Gamberucci A.; Chegaev K.; Rolando B.; Riganti C.; Fruttero R.; Saponara S.
NO release regulated by doxorubicin as the green light-harvesting antenna
2020-01-01 Fraix A.; Parisi C.; Failla M.; Chegaev K.; Spyrakis F.; Lazzarato L.; Fruttero R.; Gasco A.; Sortino S.
MRP5 nitration by NO-releasing gemcitabine encapsulated in liposomes confers sensitivity in chemoresistant pancreatic adenocarcinoma cells
2020-01-01 Masetto F.; Chegaev K.; Gazzano E.; Mullappilly N.; Rolando B.; Arpicco S.; Fruttero R.; Riganti C.; Donadelli M.
Endoplasmic reticulum-targeting doxorubicin: a new tool effective against doxorubicin-resistant osteosarcoma
2019-01-01 Buondonno, Ilaria; Gazzano, Elena; Tavanti, Elisa; Chegaev, Konstantin; Kopecka, Joanna; Fanelli, Marilù; Rolando, Barbara; Fruttero, Roberta; Gasco, Alberto; Hattinger, Claudia; Serra, Massimo; Riganti, Chiara*
INCAPSULATED NO-GEMCITABINE: GASEOUS SOLUTION FOR MDR PANCREATIC CANCER
2019-01-01 Chegaev, K.; Masetto, F.; Gazzano, E.; Mullappily, N.; Rolando, B.; Donadelli, M.; Arpicco, S.; Riganti, C.; Fruttero, R.
Paracetamol-Galactose Conjugate: A Novel Prodrug for an Old Analgesic Drug
2019-01-01 Sodano F.; Lazzarato L.; Rolando B.; Spyrakis F.; De Caro C.; Magliocca S.; Marabello D.; Chegaev K.; Gazzano E.; Riganti C.; Calignano A.; Russo R.; Rimoli M.G.
Hyaluronated liposomes containing H2S-releasing doxorubicin are effective against P-glycoprotein-positive/doxorubicin-resistant osteosarcoma cells and xenografts
2019-01-01 Gazzano E.; Buondonno I.; Marengo A.; Rolando B.; Chegaev K.; Kopecka J.; Saponara S.; Sorge M.; Hattinger C.M.; Gasco A.; Fruttero R.; Brancaccio M.; Serra M.; Stella B.; Fattal E.; Arpicco S.; Riganti C.
New tetrahydroisoquinoline-based P-glycoprotein modulators: Decoration of the biphenyl core gives selective ligands
2018-01-01 Contino, Marialessandra; Guglielmo, Stefano*; Perrone, Maria Grazia; Giampietro, Roberta; Rolando, Barbara; Carrieri, Antonio; Zaccaria, Daniele; Chegaev, Konstantin; Borio, Vanessa; Riganti, Chiara; Zabielska-Koczywas, Katarzyna; Colabufo, Nicola A.; Fruttero, Roberta
New tetrahydroisoquinoline derivatives overcome pgp activity in brain-blood barrier and glioblastoma multiforme in vitro
2018-01-01 Salaroglio, Iris Chiara; Gazzano, Elena; Kopecka, Joanna; Chegaev, Konstantin; Costamagna, Costanzo; Fruttero, Roberta; Guglielmo, Stefano*; Riganti, Chiara
New NO- and H2S-releasing doxorubicins as targeted therapy against chemoresistance in castration-resistant prostate cancer: in vitro and in vivo evaluations
2018-01-01 Bigagli, Elisabetta; Luceri, Cristina; de Angioletti, Maria; Chegaev, Konstantin; D’Ambrosio, Mario; Riganti, Chiara; Gazzano, Elena; Saponara, Simona; Longini, Mariangela; Luceri, Francesca; Cinci, Lorenzo*
Discovery of phenylsulfonylfuroxan derivatives as gamma globin inducers by histone acetylation
2018-01-01 Melo, Thais Regina Ferreira de; Kumkhaek, Chutima; Fernandes, Guilherme Felipe dos Santos; Lopes Pires, Maria Elisa; Chelucci, Rafael Consolin; Barbieri, Karina Pereira; Coelho, Fernanda; Capote, Ticiana Sidorenko de Oliveira; Lanaro, Carolina; Carlos, Iracilda Zeppone; Marcondes, Sisi; Chegaev, Konstantin; Guglielmo, Stefano; Fruttero, Roberta; Chung, Man Chin; Costa, Fernando Ferreira; Rodgers, Griffin P.; dos Santos, Jean Leandro*
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
New lipophilic organic nitrates: Candidates for chronic skin disease therapy | 2023 | Marini E.; Sodano F.; Rolando B.; Chegaev K.; Maresca D.C.; Ianaro A.; Ercolano G.; Lazzarato L. | |
Use of Enzymatically Activated Carbon Monoxide Donors for Sensitizing Drug-Resistant Tumor Cells | 2023 | Sodano, Federica; Rolando, Barbara; Lazzarato, Loretta; Costamagna, Costanzo; Failla, Mariacristina; Riganti, Chiara; Chegaev, Konstantin | |
Comparative Study of Different H2S Donors as Vasodilators and Attenuators of Superoxide-Induced Endothelial Damage | 2023 | Marini E.; Rolando B.; Sodano F.; Blua F.; Concina G.; Guglielmo S.; Lazzarato L.; Chegaev K. | |
Multitarget antioxidant NO-donor organic nitrates: a novel approach to overcome nitrates tolerance | 2022 | Elisabetta Marini, Marta Giorgis, Barbara Rolando, Konstantin Chegaev | |
A Comprehensive Evaluation of Sdox, a Promising H2S-Releasing Doxorubicin for the Treatment of Chemoresistant Tumors | 2022 | Alov P.; Al Sharif M.; Aluani D.; Chegaev K.; Dinic J.; Divac Rankov A.; Fernandes M.X.; Fusi F.; Garcia-Sosa A.T.; Juvonen R.; Kondeva-Burdina M.; Padron J.M.; Pajeva I.; Pencheva T.; Puerta A.; Raunio H.; Riganti C.; Tsakovska I.; Tzankova V.; Yordanov Y.; Saponara S. | |
N-[1,3-Dialkyl(aryl)-2-oxoimidazolidin-4-ylidene]-aryl(alkyl)sulphonamides as Novel Selective Human Cannabinoid Type 2 Receptor (hCB2R) Ligands; Insights into the Mechanism of Receptor Activation/Deactivation | 2022 | Gianquinto, Eleonora; Sodano, Federica; Rolando, Barbara; Kostrzewa, Magdalena; Allarà, Marco; Mahmoud, Ali Mokhtar; Kumar, Poulami; Spyrakis, Francesca; Ligresti, Alessia; Chegaev, Konstantin | |
Multitarget antioxidant NO-donor organic nitrates: a novel ap-proach to overcome nitrates tolerance, an ex vivo study | 2022 | Elisabetta Marini*, Marta Giorgis, Marta Leporati, Barbara Rolando, Konstantin Chegaev, Loretta Lazzarato, Massimo Bertinaria, Marco Vincenti, Antonella Di Stilo | |
Naked and Decorated Nanoparticles Containing H2S-Releasing Doxorubicin: Preparation, Characterization and Assessment of Their Antitumoral Efficiency on Various Resistant Tumor Cells | 2022 | Elena PEIRA; Daniela Chirio; Simona Sapino; Konstantin CHEGAEV; Giulia Chindamo; IRIS CHIARA SALAROGLIO; Chiara Riganti; Marina GALLARATE | |
Sdox, a H2S releasing anthracycline, with a safer profile than doxorubicin toward vasculature | 2022 | Durante M, Frosini M, Chiaino E, Fusi F, Gamberucci A, Gorelli B, Chegaev K, Riganti C, Saponara S | |
In vitro vascular toxicity assessment of NitDOX, a novel NO-releasing doxorubicin | 2020 | Durante M.; Frosini M.; Fusi F.; Gamberucci A.; Chegaev K.; Rolando B.; Riganti C.; Fruttero R.; Saponara S. | |
NO release regulated by doxorubicin as the green light-harvesting antenna | 2020 | Fraix A.; Parisi C.; Failla M.; Chegaev K.; Spyrakis F.; Lazzarato L.; Fruttero R.; Gasco A.; Sortino S. | |
MRP5 nitration by NO-releasing gemcitabine encapsulated in liposomes confers sensitivity in chemoresistant pancreatic adenocarcinoma cells | 2020 | Masetto F.; Chegaev K.; Gazzano E.; Mullappilly N.; Rolando B.; Arpicco S.; Fruttero R.; Riganti C.; Donadelli M. | |
Endoplasmic reticulum-targeting doxorubicin: a new tool effective against doxorubicin-resistant osteosarcoma | 2019 | Buondonno, Ilaria; Gazzano, Elena; Tavanti, Elisa; Chegaev, Konstantin; Kopecka, Joanna; Fanelli, Marilù; Rolando, Barbara; Fruttero, Roberta; Gasco, Alberto; Hattinger, Claudia; Serra, Massimo; Riganti, Chiara* | |
INCAPSULATED NO-GEMCITABINE: GASEOUS SOLUTION FOR MDR PANCREATIC CANCER | 2019 | Chegaev, K.; Masetto, F.; Gazzano, E.; Mullappily, N.; Rolando, B.; Donadelli, M.; Arpicco, S.; Riganti, C.; Fruttero, R. | |
Paracetamol-Galactose Conjugate: A Novel Prodrug for an Old Analgesic Drug | 2019 | Sodano F.; Lazzarato L.; Rolando B.; Spyrakis F.; De Caro C.; Magliocca S.; Marabello D.; Chegaev K.; Gazzano E.; Riganti C.; Calignano A.; Russo R.; Rimoli M.G. | |
Hyaluronated liposomes containing H2S-releasing doxorubicin are effective against P-glycoprotein-positive/doxorubicin-resistant osteosarcoma cells and xenografts | 2019 | Gazzano E.; Buondonno I.; Marengo A.; Rolando B.; Chegaev K.; Kopecka J.; Saponara S.; Sorge M.; Hattinger C.M.; Gasco A.; Fruttero R.; Brancaccio M.; Serra M.; Stella B.; Fattal E.; Arpicco S.; Riganti C. | |
New tetrahydroisoquinoline-based P-glycoprotein modulators: Decoration of the biphenyl core gives selective ligands | 2018 | Contino, Marialessandra; Guglielmo, Stefano*; Perrone, Maria Grazia; Giampietro, Roberta; Rolando, Barbara; Carrieri, Antonio; Zaccaria, Daniele; Chegaev, Konstantin; Borio, Vanessa; Riganti, Chiara; Zabielska-Koczywas, Katarzyna; Colabufo, Nicola A.; Fruttero, Roberta | |
New tetrahydroisoquinoline derivatives overcome pgp activity in brain-blood barrier and glioblastoma multiforme in vitro | 2018 | Salaroglio, Iris Chiara; Gazzano, Elena; Kopecka, Joanna; Chegaev, Konstantin; Costamagna, Costanzo; Fruttero, Roberta; Guglielmo, Stefano*; Riganti, Chiara | |
New NO- and H2S-releasing doxorubicins as targeted therapy against chemoresistance in castration-resistant prostate cancer: in vitro and in vivo evaluations | 2018 | Bigagli, Elisabetta; Luceri, Cristina; de Angioletti, Maria; Chegaev, Konstantin; D’Ambrosio, Mario; Riganti, Chiara; Gazzano, Elena; Saponara, Simona; Longini, Mariangela; Luceri, Francesca; Cinci, Lorenzo* | |
Discovery of phenylsulfonylfuroxan derivatives as gamma globin inducers by histone acetylation | 2018 | Melo, Thais Regina Ferreira de; Kumkhaek, Chutima; Fernandes, Guilherme Felipe dos Santos; Lopes Pires, Maria Elisa; Chelucci, Rafael Consolin; Barbieri, Karina Pereira; Coelho, Fernanda; Capote, Ticiana Sidorenko de Oliveira; Lanaro, Carolina; Carlos, Iracilda Zeppone; Marcondes, Sisi; Chegaev, Konstantin; Guglielmo, Stefano; Fruttero, Roberta; Chung, Man Chin; Costa, Fernando Ferreira; Rodgers, Griffin P.; dos Santos, Jean Leandro* |
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