DUCIME, ALEX
DUCIME, ALEX
Discovery and optimization of new OvCHT1 inhibitors based on the 4-hydroxy-1H-1,2,3-triazole ring
2014-01-01 A. Ducime; A. C. Pippione; A. Moreo; A. Piccinelli; M. Gooyit; K. D. Janda; D. Boschi; M. L. Lolli
Hydroxypyrazolo[1,5-a]pyridine as a fluorescent carboxylic acid isostere: introducing GABAA receptor system affinities in the scaffold
2013-01-01 A. Ducime; B. Nielsen; D. Boschi; B. Frølund; M. L. Lolli
Hydroxypyrazolo[1,5-a]pyridine as a fluorescent carboxylic acid isostere: probing first MedChem bioisosteric applications
2013-01-01 A. Ducime
PROBING THE BICYCLIC HYDROXYPYRAZOLO[1,5-a]PYRIDINE SCAFFOLD AS A CARBOXYLIC ACID BIOISOSTERE IN THE GABAa RECEPTOR SYSTEM
2012-01-01 Ducime Alex; Nielsen Birgitte; Lolli Marco L. ;Frølund Bente
Probing the bicyclic hydroxypyrazolo[1,5-a]pyridine scaffold as a carboxylic acid bioisostere in theGABAA receptor system
2012-01-01 A. Ducime; B. Nielsen; B. Frølund; M. L. Lolli
SUBSTITUTED 4-HYDROXY-1H-1,2,3-TRIAZOLES: SYNTHESIS AND BIOISOSTERIC APPLICATIONS
2014-01-01 Agnese C. Pippione; Antonella Federico; Stefano Sainas; Alex Ducime; Marco L. Lolli; Donatella Boschi
Synthesis and Structural Characterization of Regio Substituted 4-Hydroxy-1H-1,2,3-triazols as Possible Tool in Bioisosteric Applications
2014-01-01 A Federico; S.Sainas; A. Ducime;K. Martina; F. Bosca; D. Boschi; M.L. Lolli.
TOWARD A BIOISOSTERIC ALKAEST – APPLICATION TO THE BIOISOSTERIC MODULATION OF IMD-0354
2014-01-01 Marco L. Lolli; Alex Ducime; Antonella Federico; Agnese Chiara Pippione; Stefano Sainas; Alessandro Barge; Katia Martina; Donatella Boschi; Elisa Lupino; Marco Piccinini; Michael Kubbutat; Christoph Schächtele; Jean Marie Contreras; Christophe Morice; Joel Sussman; Yoav Peleg; Bjorn Walse; Salam Kadaraghi
Towards a Bioisosteric Alkaest: application to the bioisosteric modulation of IMD-0354
2014-01-01 Lolli Marco L.; Federico Antonella; Ducime Alex; Pippione Agnese; Sainas Stefano; Barge Alessandro; Martina Katia; Boschi Donatella; Lupino Elisa; Piccinini Marco; Kubbutat Michael; Contreras Jean Marie; Morice Christophe; Sussman Joel; Peleg Yoav; Walse Bjorn; Al-Kadaraghi Salam
| Titolo | Data di pubblicazione | Autore(i) | File |
|---|---|---|---|
| Discovery and optimization of new OvCHT1 inhibitors based on the 4-hydroxy-1H-1,2,3-triazole ring | 2014 | A. Ducime; A. C. Pippione; A. Moreo; A. Piccinelli; M. Gooyit; K. D. Janda; D. Boschi; M. L. Lolli | |
| Hydroxypyrazolo[1,5-a]pyridine as a fluorescent carboxylic acid isostere: introducing GABAA receptor system affinities in the scaffold | 2013 | A. Ducime; B. Nielsen; D. Boschi; B. Frølund; M. L. Lolli | |
| Hydroxypyrazolo[1,5-a]pyridine as a fluorescent carboxylic acid isostere: probing first MedChem bioisosteric applications | 2013 | A. Ducime | |
| PROBING THE BICYCLIC HYDROXYPYRAZOLO[1,5-a]PYRIDINE SCAFFOLD AS A CARBOXYLIC ACID BIOISOSTERE IN THE GABAa RECEPTOR SYSTEM | 2012 | Ducime Alex; Nielsen Birgitte; Lolli Marco L. ;Frølund Bente | |
| Probing the bicyclic hydroxypyrazolo[1,5-a]pyridine scaffold as a carboxylic acid bioisostere in theGABAA receptor system | 2012 | A. Ducime; B. Nielsen; B. Frølund; M. L. Lolli | |
| SUBSTITUTED 4-HYDROXY-1H-1,2,3-TRIAZOLES: SYNTHESIS AND BIOISOSTERIC APPLICATIONS | 2014 | Agnese C. Pippione; Antonella Federico; Stefano Sainas; Alex Ducime; Marco L. Lolli; Donatella Boschi | |
| Synthesis and Structural Characterization of Regio Substituted 4-Hydroxy-1H-1,2,3-triazols as Possible Tool in Bioisosteric Applications | 2014 | A Federico; S.Sainas; A. Ducime;K. Martina; F. Bosca; D. Boschi; M.L. Lolli. | |
| TOWARD A BIOISOSTERIC ALKAEST – APPLICATION TO THE BIOISOSTERIC MODULATION OF IMD-0354 | 2014 | Marco L. Lolli; Alex Ducime; Antonella Federico; Agnese Chiara Pippione; Stefano Sainas; Alessandro Barge; Katia Martina; Donatella Boschi; Elisa Lupino; Marco Piccinini; Michael Kubbutat; Christoph Schächtele; Jean Marie Contreras; Christophe Morice; Joel Sussman; Yoav Peleg; Bjorn Walse; Salam Kadaraghi | |
| Towards a Bioisosteric Alkaest: application to the bioisosteric modulation of IMD-0354 | 2014 | Lolli Marco L.; Federico Antonella; Ducime Alex; Pippione Agnese; Sainas Stefano; Barge Alessandro; Martina Katia; Boschi Donatella; Lupino Elisa; Piccinini Marco; Kubbutat Michael; Contreras Jean Marie; Morice Christophe; Sussman Joel; Peleg Yoav; Walse Bjorn; Al-Kadaraghi Salam |