SERAFINI, MARTA

SERAFINI, MARTA  

SCIENZA E TECNOLOGIA DEL FARMACO  

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Risultati 1 - 20 di 27 (tempo di esecuzione: 0.024 secondi).
Titolo Data di pubblicazione Autore(i) File
1,2,4-Oxadiazole-Bearing Pyrazoles as Metabolically Stable Modulators of Store-Operated Calcium Entry 2021 Aprile, Silvio; Riva, Beatrice; Bhela, Irene Preet; Cordero-Sanchez, Celia; Avino, Giulia; Genazzani, Armando; Serafini, Marta; Pirali, Tracey
A capsaicinoid-based soft drug, AG1529, for attenuating TRPV1-mediated histaminergic and inflammatory sensory neuron excitability 2021 Nikolaeva-Koleva M.; Butron L.; Gonzalez-Rodriguez S.; Devesa I.; Valente P.; Serafini M.; Genazzani A.; Pirali T.; Ballester G. F.; Fernandez-Carvajal A.; Ferrer-Montiel A.
A multicomponent approach in the discovery of indoleamine 2,3-dioxygenase 1 inhibitors: Synthesis, biological investigation and docking studies 2018 Griglio A.; Torre E.; Serafini M.; Bianchi A.; Schmid R.; Coda Zabetta G.; Massarotti A.; Sorba G.; Pirali T.; Fallarini S.
A primer of deuterium in drug design 2019 Cargnin S.; Serafini M.; Pirali T.
A Versatile and Sustainable Multicomponent Platform for the Synthesis of Protein Degraders: Proof-of-Concept Application to BRD4-Degrading PROTACs 2022 Bhela I.P.; Ranza A.; Balestrero F.C.; Serafini M.; Aprile S.; Di Martino R.M.C.; Condorelli F.; Pirali T.
An aryne-based three-component access to α-aroylamino amides 2017 Serafini M.; Griglio A.; Viarengo S.; Aprile S.; Pirali T.
An Unexpected Deuterium-Induced Metabolic Switch in Doxophylline 2022 Aprile S.; Colombo G.; Serafini M.; Di Paola R.; Pisati F.; Bhela I.P.; Cuzzocrea S.; Grosa G.; Pirali T.
Applications of deuterium in medicinal chemistry 2019 Pirali, Tracey; Serafini, Marta; Cargnin, Sarah; Genazzani, Armando
Arynes and isocyanides: Two close-knit partners in multicomponent reactions 2018 Serafini M.; Pirali T.
CIC-39Na reverses the thrombocytopenia that characterizes tubular aggregate myopathy 2022 Cordero-Sanchez, Celia; Pessolano, Emanuela; Riva, Beatrice; Vismara, Mauro; Trivigno, Silvia Maria Grazia; Clemente, Nausicaa; Aprile, Silvio; Ruffinatti, Federico Alessandro; Portararo, Paola; Filigheddu, Nicoletta; Zaggia, Ivan; Bhela, Irene P; Serafini, Marta; Pirali, Tracey; Colombo, Mario P; Torti, Mauro; Sangaletti, Sabina; Bertoni, Alessandra; Genazzani, Armando A
Click 1,2,3-triazoles in drug discovery and development: From the flask to the clinic? 2021 Serafini M.; Pirali T.; Tron G.C.
Discovery of Highly Potent Benzimidazole Derivatives as Indoleamine 2,3-Dioxygenase-1 (IDO1) Inhibitors: From Structure-Based Virtual Screening to in Vivo Pharmacodynamic Activity 2020 Serafini, M.; Torre, E.; Aprile, S.; Grosso, E.D.; Ges{\`u}, A.; Griglio, A.; Colombo, G.; Travelli, C.; Paiella, S.; Adamo, A.; Orecchini, E.; Coletti, A.; Pallotta, M.T.; Ugel, S.; Massarotti, A.; Pirali, T.; Fallarini, S.
Drug Discovery for Soft Drugs on TRPV1 and TRPM8 Channels Using the Passerini Reaction 2019 Pirali, Tracey; Galli, Ubaldina; Serafini, Marta; Griglio, Alessia; Genazzani, Armando; Tron, Gian Cesare
Erratum: An Unexpected Deuterium-Induced Metabolic Switch in Doxophylline (ACS Medicinal Chemistry Letters (2022) 13: 8 (1278−1285) DOI: 10.1021/acsmedchemlett.2c00166) 2023 Silvio Aprile; Giorgia Colombo; Marta Serafini; Rosanna Di Paola; Federica Pisati; Irene Preet Bhela; Salvatore Cuzzocrea; Giorgio Grosa; Tracey Pirali
Mutate and Conjugate: A Method to Enable Rapid In-Cell Target Validation 2023 Thomas A.M.; Serafini M.; Grant E.K.; Coombs E.A.J.; Bluck J.P.; Schiedel M.; McDonough M.A.; Reynolds J.K.; Lee B.; Platt M.; Sharlandjieva V.; Biggin P.C.; Duarte F.; Milne T.A.; Bush J.T.; Conway S.J.
Pyrtriazoles, a Novel Class of Store-Operated Calcium Entry Modulators: Discovery, Biological Profiling, and in Vivo Proof-of-Concept Efficacy in Acute Pancreatitis 2018 Riva, Beatrice; Griglio, Alessia; Serafini, Marta; CORDERO SANCHEZ, CELIA; Aprile, Silvio; Di Paola, Rosanna; Gugliandolo, Enrico; Alansary, Dalia; BIOCOTINO, Isabella; Lim, Dmitry; Grosa, Giorgio; Galli, Ubaldina; Niemeyer, Barbara; Sorba, Giovanni; Canonico, Pier Luigi; Cuzzocrea, Salvatore; Genazzani, Armando; Pirali, Tracey
Soft drugs for dermatological applications: recent trends 2019 Aprile S.; Serafini M.; Pirali T.
STIM1 and ORAI1 mutations leading to tubular aggregate myopathies are sensitive to the Store-operated Ca2+-entry modulators CIC-37 and CIC-39 2022 Riva, Beatrice; Pessolano, Emanuela; Quaglia, Edoardo; Cordero-Sanchez, Celia; Bhela, Irene P; Topf, Ana; Serafini, Marta; Cox, Daniel; Harris, Elizabeth; Garibaldi, Matteo; Barresi, Rita; Pirali, Tracey; Genazzani, Armando
Store-Operated Calcium Entry as a Therapeutic Target in Acute Pancreatitis: Discovery and Development of Drug-Like SOCE Inhibitors 2020 Serafini M.; Cordero Sanchez C.; Di Paola R.; Bhela I. P.; Aprile S.; Purghe B.; Fusco R.; Cuzzocrea S.; Genazzani A.; Riva B.; Pirali T.
Synthesis, docking and biological evaluation of a novel class of imidazothiazoles as IDO1 inhibitors 2019 Serafini M.; Torre E.; Aprile S.; Massarotti A.; Fallarini S.; Pirali T.