Sfoglia per Autore
Identification of novel aza-analogs of TN-16 as disrupters of microtubule dynamics through a multicomponent reaction
2023-01-01 Foroutan, Arash; Corazzari, Marco; Grolla, Ambra A; Colombo, Giorgia; Travelli, Cristina; Genazzani, Armando A; Theeramunkong, Sewan; Galli, Ubaldina; Tron, Gian Cesare
The 115 year old multicomponent Bargellini reaction: Perspectives and new applications
2021-01-01 Serafini M.; Murgia I.; Giustiniano M.; Pirali T.; Tron G.C.
Tritylamine as an ammonia surrogate in the ugi reaction provides access to unprecedented 5-sulfamido oxazoles using burgess-type reagents
2021-01-01 Bhela I.P.; Serafini M.; Del Grosso E.; Tron G.C.; Pirali T.
What's in a Name? Drug Nomenclature and Medicinal Chemistry Trends using INN Publications
2021-01-01 Serafini M.; Cargnin S.; Massarotti A.; Tron G. C.; Pirali T.; Genazzani A.
Icilio Guareschi and his amazing “1897 reaction”
2021-01-01 Tron, Gian Cesare; Minassi, Alberto; Sorba, Giovanni; Fausone, Mara; Appendino, Giovanni
Recent Advances in NAMPT Inhibitors: A Novel Immunotherapic Strategy
2020-01-01 Galli, Ubaldina; Colombo, Giorgia; Travelli, Cristina; Tron, Gian Cesare; Genazzani, Armando; Grolla, Ambra
Structure activity relationship studies on Amb639752: toward the identification of a common pharmacophoric structure for DGKα inhibitors
2020-01-01 Velnati S.; Massarotti A.; Antona A.; Talmon M.; Fresu L.G.; Galetto A.S.; Capello D.; Bertoni A.; Mercalli V.; Graziani A.; Tron G.C.; Baldanzi G.
Drug Discovery for Soft Drugs on TRPV1 and TRPM8 Channels Using the Passerini Reaction
2019-01-01 Pirali, Tracey; Galli, Ubaldina; Serafini, Marta; Griglio, Alessia; Genazzani, Armando; Tron, Gian Cesare
Identification of potent triazolylpyridine nicotinamide phosphoribosyltransferase (NAMPT) inhibitors bearing a 1,2,3-triazole tail group
2019-01-01 Travelli, Cristina; Aprile, Silvio; Mattoteia, Daiana; Colombo, Giorgia; Clemente, Nausicaa; Scanziani, Eugenio; Terrazzino, Salvatore; Alisi, Maria Alessandra; Polenzani, Lorenzo; Grosa, Giorgio; Genazzani, Armando; Tron, Gian Cesare; Galli, Ubaldina
Inhalation of the prodrug PI3K inhibitor CL27c improves lung function in asthma and fibrosis
2018-01-01 Campa, Carlo C.; Silva, Rangel L.; Margaria, Jean P.; Pirali, Tracey; Mattos, Matheus S.; Kraemer, Lucas R.; Reis, Diego C.; Grosa, Giorgio; Copperi, Francesca; Dalmarco, Eduardo M.; Lima-Júnior, Roberto C. P.; Aprile, Silvio; Sala, Valentina; Dal Bello, Federica; Prado, Douglas Silva; Alves-Filho, Jose Carlos; Medana, Claudio; Cassali, Geovanni D.; Tron, Gian Cesare; Teixeira, Mauro M.; Ciraolo, Elisa; Russo, Remo C.; Hirsch, Emilio
Identification of a Potent Phosphoinositide 3-Kinase Pan Inhibitor Displaying a Strategic Carboxylic Acid Group and Development of Its Prodrugs
2017-01-01 Pirali, Tracey; Ciraolo, Elisa; Aprile, Silvio; Massarotti, Alberto; Berndt, Alex; Griglio, Alessia; Serafini, Marta; Mercalli, Valentina; Landoni, Clarissa; Campa, Carlo Cosimo; Margaria, Jean Piero; Silva, Rangel L.; Grosa, Giorgio; Sorba, Giovanni; Williams, Roger; Hirsch, Emilio; Tron, Gian Cesare
The use of 2-hydroxymethyl benzoic acid as an effective water surrogate in the Passerini reaction: A straightforward access to α-hydroxyamides
2017-01-01 Serafini M.; Griglio A.; Oberto E.; Pirali T.; Tron G.C.
Identification of Novel Triazole-Based Nicotinamide Phosphoribosyltransferase (NAMPT) Inhibitors Endowed with Antiproliferative and Antiinflammatory Activity
2017-01-01 TRAVELLI, Cristina; APRILE, SILVIO; Rahimian, Reza; Grolla, Ambra A.; ROGATI, FEDERICA; Bertolotti, Mattia; Malagnino, Floriana; Di Paola, Rosanna; Impellizzeri, Daniela; FUSCO, Roberta; MERCALLI, VALENTINA; MASSAROTTI, Alberto; Stortini, Giorgio; TERRAZZINO, SALVATORE; DEL GROSSO, Erika; Fakhfouri, Gohar; Troiani, Maria Pia; Alisi, Maria Alessandra; GROSA, Giorgio; SORBA, Giovanni; CANONICO, Pier Luigi; Orsomando, Giuseppe; Cuzzocrea, Salvatore; GENAZZANI, Armando; GALLI, Ubaldina; TRON, Gian Cesare
Design, synthesis, and biological evaluation of combretabenzodiazepines: a novel class of anti-tubulin agents
2015-01-01 GALLI, Ubaldina; TRAVELLI, Cristina; APRILE, SILVIO; Arrigoni, Elena; TORRETTA, SIMONE; GROSA, Giorgio; MASSAROTTI, Alberto; SORBA, Giovanni; CANONICO, Pier Luigi; GENAZZANI, Armando; TRON, Gian Cesare
Identification of a novel NAMPT inhibitor by combinatorial click chemistry and chemical refinement
2015-01-01 Theeramunkong, S.; GALLI, Ubaldina; GROLLA, AMBRA; CALDARELLI, ANTONIO; TRAVELLI, Cristina; MASSAROTTI, Alberto; Troiani, M. P.; Alisi, M. A.; Orsomando, G.; GENAZZANI, Armando; TRON, Gian Cesare
Medicinal chemistry of nicotinamide phosphoribosyltransferase (NAMPT) inhibitors
2013-01-01 GALLI, Ubaldina; TRAVELLI, Cristina; MASSAROTTI, Alberto; Fakhfouri, G; Rahimian, R; TRON, Gian Cesare; GENAZZANI, Armando
The NAMPT inhibitor FK866 reverts the damage in spinal cord injury
2012-01-01 Esposito E; Impellizzeri D; Mazzon E; Fakhfouri G; Rahimian R; Travelli C; TRON, Gian Cesare; GENAZZANI, Armando; Cuzzocrea S.
Identification of a sirtuin 3 inhibitor that displays selectivity over sirtuin 1 and 2
2012-01-01 GALLI, Ubaldina; MESENZANI, Ornella; Coppo C; SORBA, Giovanni; CANONICO, Pier Luigi; TRON, Gian Cesare; GENAZZANI, Armando
Reciprocal potentiation of the antitumoral activities of FK866, an inhibitor of nicotinamide phosphoribosyltransferase, and etoposide or cisplatin in neuroblastoma cells
2011-01-01 TRAVELLI, Cristina; DRAGO, VALENTINA; Maldi E; Kaludercic N; GALLI, Ubaldina; BOLDORINI, Renzo Luciano; Di Lisa F; TRON, Gian Cesare; CANONICO, Pier Luigi; GENAZZANI, Armando
Regioselective Suzuki coupling of dihaloheteroaromatic compounds as a rapid strategy to synthesize potent rigid combretastatin analogues
2011-01-01 Theeramunkong S; CALDARELLI, ANTONIO; MASSAROTTI, Alberto; APRILE, SILVIO; CAPRIOGLIO, DIEGO; ZANINETTI, ROBERTA; Teruggi A; PIRALI, Tracey; GROSA, Giorgio; TRON, Gian Cesare; GENAZZANI, Armando
| Titolo | Data di pubblicazione | Autore(i) | File |
|---|---|---|---|
| Identification of novel aza-analogs of TN-16 as disrupters of microtubule dynamics through a multicomponent reaction | 2023 | Foroutan, Arash; Corazzari, Marco; Grolla, Ambra A; Colombo, Giorgia; Travelli, Cristina; Genazzani, Armando A; Theeramunkong, Sewan; Galli, Ubaldina; Tron, Gian Cesare | |
| The 115 year old multicomponent Bargellini reaction: Perspectives and new applications | 2021 | Serafini M.; Murgia I.; Giustiniano M.; Pirali T.; Tron G.C. | |
| Tritylamine as an ammonia surrogate in the ugi reaction provides access to unprecedented 5-sulfamido oxazoles using burgess-type reagents | 2021 | Bhela I.P.; Serafini M.; Del Grosso E.; Tron G.C.; Pirali T. | |
| What's in a Name? Drug Nomenclature and Medicinal Chemistry Trends using INN Publications | 2021 | Serafini M.; Cargnin S.; Massarotti A.; Tron G. C.; Pirali T.; Genazzani A. | |
| Icilio Guareschi and his amazing “1897 reaction” | 2021 | Tron, Gian Cesare; Minassi, Alberto; Sorba, Giovanni; Fausone, Mara; Appendino, Giovanni | |
| Recent Advances in NAMPT Inhibitors: A Novel Immunotherapic Strategy | 2020 | Galli, Ubaldina; Colombo, Giorgia; Travelli, Cristina; Tron, Gian Cesare; Genazzani, Armando; Grolla, Ambra | |
| Structure activity relationship studies on Amb639752: toward the identification of a common pharmacophoric structure for DGKα inhibitors | 2020 | Velnati S.; Massarotti A.; Antona A.; Talmon M.; Fresu L.G.; Galetto A.S.; Capello D.; Bertoni A.; Mercalli V.; Graziani A.; Tron G.C.; Baldanzi G. | |
| Drug Discovery for Soft Drugs on TRPV1 and TRPM8 Channels Using the Passerini Reaction | 2019 | Pirali, Tracey; Galli, Ubaldina; Serafini, Marta; Griglio, Alessia; Genazzani, Armando; Tron, Gian Cesare | |
| Identification of potent triazolylpyridine nicotinamide phosphoribosyltransferase (NAMPT) inhibitors bearing a 1,2,3-triazole tail group | 2019 | Travelli, Cristina; Aprile, Silvio; Mattoteia, Daiana; Colombo, Giorgia; Clemente, Nausicaa; Scanziani, Eugenio; Terrazzino, Salvatore; Alisi, Maria Alessandra; Polenzani, Lorenzo; Grosa, Giorgio; Genazzani, Armando; Tron, Gian Cesare; Galli, Ubaldina | |
| Inhalation of the prodrug PI3K inhibitor CL27c improves lung function in asthma and fibrosis | 2018 | Campa, Carlo C.; Silva, Rangel L.; Margaria, Jean P.; Pirali, Tracey; Mattos, Matheus S.; Kraemer, Lucas R.; Reis, Diego C.; Grosa, Giorgio; Copperi, Francesca; Dalmarco, Eduardo M.; Lima-Júnior, Roberto C. P.; Aprile, Silvio; Sala, Valentina; Dal Bello, Federica; Prado, Douglas Silva; Alves-Filho, Jose Carlos; Medana, Claudio; Cassali, Geovanni D.; Tron, Gian Cesare; Teixeira, Mauro M.; Ciraolo, Elisa; Russo, Remo C.; Hirsch, Emilio | |
| Identification of a Potent Phosphoinositide 3-Kinase Pan Inhibitor Displaying a Strategic Carboxylic Acid Group and Development of Its Prodrugs | 2017 | Pirali, Tracey; Ciraolo, Elisa; Aprile, Silvio; Massarotti, Alberto; Berndt, Alex; Griglio, Alessia; Serafini, Marta; Mercalli, Valentina; Landoni, Clarissa; Campa, Carlo Cosimo; Margaria, Jean Piero; Silva, Rangel L.; Grosa, Giorgio; Sorba, Giovanni; Williams, Roger; Hirsch, Emilio; Tron, Gian Cesare | |
| The use of 2-hydroxymethyl benzoic acid as an effective water surrogate in the Passerini reaction: A straightforward access to α-hydroxyamides | 2017 | Serafini M.; Griglio A.; Oberto E.; Pirali T.; Tron G.C. | |
| Identification of Novel Triazole-Based Nicotinamide Phosphoribosyltransferase (NAMPT) Inhibitors Endowed with Antiproliferative and Antiinflammatory Activity | 2017 | TRAVELLI, Cristina; APRILE, SILVIO; Rahimian, Reza; Grolla, Ambra A.; ROGATI, FEDERICA; Bertolotti, Mattia; Malagnino, Floriana; Di Paola, Rosanna; Impellizzeri, Daniela; FUSCO, Roberta; MERCALLI, VALENTINA; MASSAROTTI, Alberto; Stortini, Giorgio; TERRAZZINO, SALVATORE; DEL GROSSO, Erika; Fakhfouri, Gohar; Troiani, Maria Pia; Alisi, Maria Alessandra; GROSA, Giorgio; SORBA, Giovanni; CANONICO, Pier Luigi; Orsomando, Giuseppe; Cuzzocrea, Salvatore; GENAZZANI, Armando; GALLI, Ubaldina; TRON, Gian Cesare | |
| Design, synthesis, and biological evaluation of combretabenzodiazepines: a novel class of anti-tubulin agents | 2015 | GALLI, Ubaldina; TRAVELLI, Cristina; APRILE, SILVIO; Arrigoni, Elena; TORRETTA, SIMONE; GROSA, Giorgio; MASSAROTTI, Alberto; SORBA, Giovanni; CANONICO, Pier Luigi; GENAZZANI, Armando; TRON, Gian Cesare | |
| Identification of a novel NAMPT inhibitor by combinatorial click chemistry and chemical refinement | 2015 | Theeramunkong, S.; GALLI, Ubaldina; GROLLA, AMBRA; CALDARELLI, ANTONIO; TRAVELLI, Cristina; MASSAROTTI, Alberto; Troiani, M. P.; Alisi, M. A.; Orsomando, G.; GENAZZANI, Armando; TRON, Gian Cesare | |
| Medicinal chemistry of nicotinamide phosphoribosyltransferase (NAMPT) inhibitors | 2013 | GALLI, Ubaldina; TRAVELLI, Cristina; MASSAROTTI, Alberto; Fakhfouri, G; Rahimian, R; TRON, Gian Cesare; GENAZZANI, Armando | |
| The NAMPT inhibitor FK866 reverts the damage in spinal cord injury | 2012 | Esposito E; Impellizzeri D; Mazzon E; Fakhfouri G; Rahimian R; Travelli C; TRON, Gian Cesare; GENAZZANI, Armando; Cuzzocrea S. | |
| Identification of a sirtuin 3 inhibitor that displays selectivity over sirtuin 1 and 2 | 2012 | GALLI, Ubaldina; MESENZANI, Ornella; Coppo C; SORBA, Giovanni; CANONICO, Pier Luigi; TRON, Gian Cesare; GENAZZANI, Armando | |
| Reciprocal potentiation of the antitumoral activities of FK866, an inhibitor of nicotinamide phosphoribosyltransferase, and etoposide or cisplatin in neuroblastoma cells | 2011 | TRAVELLI, Cristina; DRAGO, VALENTINA; Maldi E; Kaludercic N; GALLI, Ubaldina; BOLDORINI, Renzo Luciano; Di Lisa F; TRON, Gian Cesare; CANONICO, Pier Luigi; GENAZZANI, Armando | |
| Regioselective Suzuki coupling of dihaloheteroaromatic compounds as a rapid strategy to synthesize potent rigid combretastatin analogues | 2011 | Theeramunkong S; CALDARELLI, ANTONIO; MASSAROTTI, Alberto; APRILE, SILVIO; CAPRIOGLIO, DIEGO; ZANINETTI, ROBERTA; Teruggi A; PIRALI, Tracey; GROSA, Giorgio; TRON, Gian Cesare; GENAZZANI, Armando |
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