CARNOVALE, IRENE MARIA
CARNOVALE, IRENE MARIA
Bioisosteres of Indomethacin as Inhibitors of Aldo-Keto Reductase 1C3
2019-01-01 Lolli, Marco L; Carnovale, Irene M; Pippione, Agnese C; Wahlgren, Weixiao Y; Bonanni, Davide; Marini, Elisabetta; Zonari, Daniele; Gallicchio, Margherita; Boscaro, Valentina; Goyal, Parveen; Friemann, Rosmarie; Rolando, Barbara; Bagnati, Renzo; Adinolfi, Salvatore; Oliaro-Bosso, Simonetta; Boschi, Donatella
Exploring the intramolecular catalysis of the proton exchange process to modulate the relaxivity of Gd(iii)-complexes of HP-DO3A-like ligands
2018-01-01 Carnovale, Irene Maria; Lolli, Marco Lucio; Serra, Sonia Colombo; Mingo, Alberto Fringuello; Napolitano, Roberta; Boi, Valeria; Guidolin, Nicol; Lattuada, Luciano; Tedoldi, Fabio; Baranyai, Zsolt; Aime, Silvio
H-Bonding and intramolecular catalysis of proton exchange affect the CEST properties of EuIIIcomplexes with HP-DO3A-like ligands
2021-01-01 Baroni S.; Carnovale I.M.; Carrera C.; Boccalon M.; Guidolin N.; Demitri N.; Lattuada L.; Tedoldi F.; Baranyai Z.; Aime S.
Hydroxytriazole derivatives as potent and selective aldo-keto reductase 1C3 (AKR1C3) inhibitors discovered by bioisosteric scaffold hopping approach
2017-01-01 Pippione, Agnese C.; Giraudo, Alessandro; Bonanni, Davide; Carnovale, Irene M.; Marini, Elisabetta; Cena, Clara; Costale, Annalisa; Zonari, Daniele; Pors, Klaus; Sadiq, Maria; Boschi, Donatella; Oliaro-Bosso, Simonetta; Lolli, Marco L
Macrocyclic paramagnetic agents for MRI: Determinants of relaxivity and strategies for their improvement
2017-01-01 Fringuello Mingo, Alberto; Colombo Serra, Sonia; Baroni, Simona; Cabella, Claudia; Napolitano, Roberta; Hawala, Ivan; Carnovale, Irene Maria; Lattuada, Luciano; Tedoldi, Fabio; Aime, Silvio
NEW HYDROXYAZOLES INHIBITORS OF AKR1C3 OBTAINED FROM NSAIDS BY SCAFFOLD HOPPING APPROACH AGAINST CASTRATE RESISTANT PROSTATE CANCER
2016-01-01 Boschi, Donatella; Pippione, Agnese Chiara; Giraudo, Alessandro; Carnovale, Irene Maria; Zorniotti, Sonia; Oliaro-Bosso, Simonetta; Ferrante, Terenzio; Marini, Elisabetta; Pors, Klaus; Festuccia, Claudio; Monache, Simona Delle; Zaffaroni, Nadia; Braga, Rodolpho Campos; Lucio Lolli, Marco
NEW HYDROXYAZOLES INHIBITORS OF ALDO-KETO REDUCTASE 1C3 (AKR1C3) OBTAINED BY SCAFFOLD HOPPING FROM FLUFENAMIC ACID AND INDOMETHACIN FOR CASTRATE RESISTANT PROSTATE CANCER
2016-01-01 Boschi, Donatella; Pippione, Agnese Chiara; Giraudo, Alessandro; Carnovale, Irene Maria; Zorniotti, Sonia; Oliaro-Bosso, Simonetta; Ferrante, Terenzio; Marini, Elisabetta; Pors, Klaus; Festuccia, Claudio; Monache, Simona Delle; Zaffaroni, Nadia; Braga, Rodolpho Campos; Lucio, Marco; Lolli,
Potent and selective aldo-keto reductase 1C3 (AKR1C3) inhibitors based on the benzoisoxazole moiety: Application of a bioisosteric scaffold hopping approach to flufenamic acid
2018-01-01 Pippione, Agnese Chiara; Carnovale, Irene Maria; Bonanni, Davide; Sini, Marcella; Goyal, Parveen; Marini, Elisabetta; Pors, Klaus; Adinolfi, Salvatore; Zonari, Daniele; Festuccia, Claudio; Wahlgren, Weixiao Yuan; Friemann, Rosmarie; Bagnati, Renzo; Boschi, Donatella; Oliaro-Bosso, Simonetta; Lolli, Marco Lucio
Synthesis of new gadolinium complexes for magnetic resonance imaging with improved relaxivity
2017-01-01 Irene Maria Carnovale, ; Sonia Colombo Serra, ; Alberto Fringuello Mingo, ; Luciano, Lattuada; Marco Lucio Lolli,
Synthesis of new gadolinium complexes for magnetic resonance imaging with improved relaxivity
2017-01-01 Carnovale, I. M.; Colombo Serra, S.; Fringuello Mingo, A.; Lattuada, L.; Lolli, M. L.
Synthesis of new Gadolinium complexes for magnetic resonance imaging with improved relaxivity
2017-01-01 Carnovale, Irene Maria; Serra, Sonia Colombo; Fringuello Mingo, Alberto; Lattuada, Luciano; Lolli, Marco Lucio
Targeting Castration Resistant Prostate Cancer (CRPC) by innovative AKR1C3 inhibitors based on the 3-hydroxybenzoisoxazole structure
2016-01-01 Carnovale, Irene Maria; Pippione, Agnese Chiara; Giraudo, Alessandro; Federico, Antonella; Zorniotti, Sonia; Simonetta Oliaro Bosso, ; Ferrante, Terenzio; Marini, Elisabetta; Pors, Klaus; Braga, Rodolpho Campos; Boschi, Donatella; Lucio Lolli, Marco
Targeting the human Dihydroorotate Dehydrogenase (hDHODH) by a Scaffold Hopping Bioisosteric approach using Hydroxylated Pentaatomic Heterocycles
2016-01-01 Sainas, Stefano; Pippione, Agnese Chiara; Carnovale, IRENE MARIA; Giraudo, Alessandro; Giorgis, Marta; Braga Rodolpho Campos, ; Andrade Carolina Horta, ; Piccinini, Marco; Lupino, Elisa; Guedes, Rita; AL KARADAGHI, Salam; Boschi, Donatella; Lolli, Marco Lucio
Targeting the human Dihydroorotate Dehydrogenase (hDHODH) by a Scaffold Hopping Bioisosteric approach using Hydroxylated Pentatomic Heterocycles
2016-01-01 Sainas Stefano; Pippione Agnese Chiara; Carnovale Irene Maria; Giraudo Alessandro; Giorgis Marta; de Campos Braga Rodolpho; Andrade Carolina H; Villella Noemi; Friemann Rosmarie; Piccinini Marco; Lupino Elisa; Al-karadaghi Salam; Boschi Donatella;Lolli Marco Lucio
Targeting the human Dihydroorotate Dehydrogenase (hDHODH) by a Scaffold Hopping Bioisosteric approach using Hydroxylated Pentatomic Heterocycles
2016-01-01 Stefano Sainas, Agnese Chiara Pippione, Irene Maria Carnovale, Alessandro Giraudo, Marta Giorgis, Rodolpho B. Braga, Carolina H. Andrade, Noemi Villella, Marco Piccinini, Elisa Lupino, Rosmarie Friemann, Salam Al-Kadaraghi, Donatella Boschi, Marco L. Lolli
Targeting the human Dihydroorotate Dehydrogenase (hDHODH) by combination of in-silico ligand/structural pharmacophore models and scaffold hopping bioisosteric approaches
2015-01-01 Mensa, Stefano; Carnovale, Irene M.; Pippione, Agnese Chiara; Sainas, Stefano; Giorgis, Marta; Piccinini, Marco; Lupino, Elisa; Al-Karadaghi, Salam; Boschi, Donatella; L. Lolli., Marco
| Titolo | Data di pubblicazione | Autore(i) | File |
|---|---|---|---|
| Bioisosteres of Indomethacin as Inhibitors of Aldo-Keto Reductase 1C3 | 2019 | Lolli, Marco L; Carnovale, Irene M; Pippione, Agnese C; Wahlgren, Weixiao Y; Bonanni, Davide; Marini, Elisabetta; Zonari, Daniele; Gallicchio, Margherita; Boscaro, Valentina; Goyal, Parveen; Friemann, Rosmarie; Rolando, Barbara; Bagnati, Renzo; Adinolfi, Salvatore; Oliaro-Bosso, Simonetta; Boschi, Donatella | |
| Exploring the intramolecular catalysis of the proton exchange process to modulate the relaxivity of Gd(iii)-complexes of HP-DO3A-like ligands | 2018 | Carnovale, Irene Maria; Lolli, Marco Lucio; Serra, Sonia Colombo; Mingo, Alberto Fringuello; Napolitano, Roberta; Boi, Valeria; Guidolin, Nicol; Lattuada, Luciano; Tedoldi, Fabio; Baranyai, Zsolt; Aime, Silvio | |
| H-Bonding and intramolecular catalysis of proton exchange affect the CEST properties of EuIIIcomplexes with HP-DO3A-like ligands | 2021 | Baroni S.; Carnovale I.M.; Carrera C.; Boccalon M.; Guidolin N.; Demitri N.; Lattuada L.; Tedoldi F.; Baranyai Z.; Aime S. | |
| Hydroxytriazole derivatives as potent and selective aldo-keto reductase 1C3 (AKR1C3) inhibitors discovered by bioisosteric scaffold hopping approach | 2017 | Pippione, Agnese C.; Giraudo, Alessandro; Bonanni, Davide; Carnovale, Irene M.; Marini, Elisabetta; Cena, Clara; Costale, Annalisa; Zonari, Daniele; Pors, Klaus; Sadiq, Maria; Boschi, Donatella; Oliaro-Bosso, Simonetta; Lolli, Marco L | |
| Macrocyclic paramagnetic agents for MRI: Determinants of relaxivity and strategies for their improvement | 2017 | Fringuello Mingo, Alberto; Colombo Serra, Sonia; Baroni, Simona; Cabella, Claudia; Napolitano, Roberta; Hawala, Ivan; Carnovale, Irene Maria; Lattuada, Luciano; Tedoldi, Fabio; Aime, Silvio | |
| NEW HYDROXYAZOLES INHIBITORS OF AKR1C3 OBTAINED FROM NSAIDS BY SCAFFOLD HOPPING APPROACH AGAINST CASTRATE RESISTANT PROSTATE CANCER | 2016 | Boschi, Donatella; Pippione, Agnese Chiara; Giraudo, Alessandro; Carnovale, Irene Maria; Zorniotti, Sonia; Oliaro-Bosso, Simonetta; Ferrante, Terenzio; Marini, Elisabetta; Pors, Klaus; Festuccia, Claudio; Monache, Simona Delle; Zaffaroni, Nadia; Braga, Rodolpho Campos; Lucio Lolli, Marco | |
| NEW HYDROXYAZOLES INHIBITORS OF ALDO-KETO REDUCTASE 1C3 (AKR1C3) OBTAINED BY SCAFFOLD HOPPING FROM FLUFENAMIC ACID AND INDOMETHACIN FOR CASTRATE RESISTANT PROSTATE CANCER | 2016 | Boschi, Donatella; Pippione, Agnese Chiara; Giraudo, Alessandro; Carnovale, Irene Maria; Zorniotti, Sonia; Oliaro-Bosso, Simonetta; Ferrante, Terenzio; Marini, Elisabetta; Pors, Klaus; Festuccia, Claudio; Monache, Simona Delle; Zaffaroni, Nadia; Braga, Rodolpho Campos; Lucio, Marco; Lolli, | |
| Potent and selective aldo-keto reductase 1C3 (AKR1C3) inhibitors based on the benzoisoxazole moiety: Application of a bioisosteric scaffold hopping approach to flufenamic acid | 2018 | Pippione, Agnese Chiara; Carnovale, Irene Maria; Bonanni, Davide; Sini, Marcella; Goyal, Parveen; Marini, Elisabetta; Pors, Klaus; Adinolfi, Salvatore; Zonari, Daniele; Festuccia, Claudio; Wahlgren, Weixiao Yuan; Friemann, Rosmarie; Bagnati, Renzo; Boschi, Donatella; Oliaro-Bosso, Simonetta; Lolli, Marco Lucio | |
| Synthesis of new gadolinium complexes for magnetic resonance imaging with improved relaxivity | 2017 | Irene Maria Carnovale, ; Sonia Colombo Serra, ; Alberto Fringuello Mingo, ; Luciano, Lattuada; Marco Lucio Lolli, | |
| Synthesis of new gadolinium complexes for magnetic resonance imaging with improved relaxivity | 2017 | Carnovale, I. M.; Colombo Serra, S.; Fringuello Mingo, A.; Lattuada, L.; Lolli, M. L. | |
| Synthesis of new Gadolinium complexes for magnetic resonance imaging with improved relaxivity | 2017 | Carnovale, Irene Maria; Serra, Sonia Colombo; Fringuello Mingo, Alberto; Lattuada, Luciano; Lolli, Marco Lucio | |
| Targeting Castration Resistant Prostate Cancer (CRPC) by innovative AKR1C3 inhibitors based on the 3-hydroxybenzoisoxazole structure | 2016 | Carnovale, Irene Maria; Pippione, Agnese Chiara; Giraudo, Alessandro; Federico, Antonella; Zorniotti, Sonia; Simonetta Oliaro Bosso, ; Ferrante, Terenzio; Marini, Elisabetta; Pors, Klaus; Braga, Rodolpho Campos; Boschi, Donatella; Lucio Lolli, Marco | |
| Targeting the human Dihydroorotate Dehydrogenase (hDHODH) by a Scaffold Hopping Bioisosteric approach using Hydroxylated Pentaatomic Heterocycles | 2016 | Sainas, Stefano; Pippione, Agnese Chiara; Carnovale, IRENE MARIA; Giraudo, Alessandro; Giorgis, Marta; Braga Rodolpho Campos, ; Andrade Carolina Horta, ; Piccinini, Marco; Lupino, Elisa; Guedes, Rita; AL KARADAGHI, Salam; Boschi, Donatella; Lolli, Marco Lucio | |
| Targeting the human Dihydroorotate Dehydrogenase (hDHODH) by a Scaffold Hopping Bioisosteric approach using Hydroxylated Pentatomic Heterocycles | 2016 | Sainas Stefano; Pippione Agnese Chiara; Carnovale Irene Maria; Giraudo Alessandro; Giorgis Marta; de Campos Braga Rodolpho; Andrade Carolina H; Villella Noemi; Friemann Rosmarie; Piccinini Marco; Lupino Elisa; Al-karadaghi Salam; Boschi Donatella;Lolli Marco Lucio | |
| Targeting the human Dihydroorotate Dehydrogenase (hDHODH) by a Scaffold Hopping Bioisosteric approach using Hydroxylated Pentatomic Heterocycles | 2016 | Stefano Sainas, Agnese Chiara Pippione, Irene Maria Carnovale, Alessandro Giraudo, Marta Giorgis, Rodolpho B. Braga, Carolina H. Andrade, Noemi Villella, Marco Piccinini, Elisa Lupino, Rosmarie Friemann, Salam Al-Kadaraghi, Donatella Boschi, Marco L. Lolli | |
| Targeting the human Dihydroorotate Dehydrogenase (hDHODH) by combination of in-silico ligand/structural pharmacophore models and scaffold hopping bioisosteric approaches | 2015 | Mensa, Stefano; Carnovale, Irene M.; Pippione, Agnese Chiara; Sainas, Stefano; Giorgis, Marta; Piccinini, Marco; Lupino, Elisa; Al-Karadaghi, Salam; Boschi, Donatella; L. Lolli., Marco |