OLIARO BOSSO, Simonetta

OLIARO BOSSO, Simonetta  

SCIENZA E TECNOLOGIA DEL FARMACO  

Mostra records
Risultati 1 - 20 di 43 (tempo di esecuzione: 0.024 secondi).
Titolo Data di pubblicazione Autore(i) File
4-methyl zymosterone and other 4-methyl intermediates of sterol biosynthesis from yeast mutants engineered in the ERG27 gene encoding 3-ketosteroid reductase 2015 Ferrante, Terenzio; Barge, Alessandro; Albezzano, Claudia; Ballestrazzi Clara; Balliano, Gianni; Oliaro-Bosso, Simonetta
A mutation in yeast oxidosqualene cyclase (Erg7) makes it independent of 3-ketoreductase activity (Erg27) 2012 Layer Jacob V; Barnes Brett M; Yamasaki Yuji; Barbuch Robert; Li Lingtao; Taramino Silvia; Oliaro-Bosso Simonetta; Balliano Gianni; Bard Martin
A new generation of AKR1C3 inhibitors on the horizon: the 3- hydroxybenzazole approach to target prostate cancer 2023 Chiara Vigato, Agnese Chiara Pippione, Stefano Sainas, Iole Mannella, Laura Bertarini, Sandra Kovachka, Barbara Rolando, Osman Asghar Mirza, Karla Frydenvang, Francesca Spyrakis, Simonetta Oliaro-Bosso, Marco Lucio Lolli, Donatella Boschi
Access of the substrate to the active site of yeast oxidosqualene cyclase: a modelling and site-directed mutagenesis approach 2009 S. Oliaro-Bosso; S. Taramino; Y. Ferrari; G. Ermondi; G. Caron; F. Viola; G. Balliano
Access of the substrate to the active site of yeast oxidosqualene cyclase: an inhibition and site-directed mutagenesis appoach. 2004 OLIARO-BOSSO S.; SCALDAFERRI M.; TARAMINO S.; F. VIOLA; G. BALLIANO
Access of the substrate to the active site of yeast oxidosqualene cyclase: an inhibition and site-directed mutagenesis approach. 2005 Balliano G.; Oliaro-Bosso S.; Taramino S.; Viola F
Application of an in house bioisosteric approach to the design of innovative inhibitors of aldo-keto reductase 1C3 (AKR1C3) 2019 Chiara Vigato, Agnese Chiara Pippione, Sandra Kovachka, Francesca Spyrakis, Martina Daga, Simonetta Oliaro Bosso, Marco Lucio Lolli, Donatella Boschi
Application of an in house bioisosteric approach to the design of innovative inhibitors of aldo-keto reductase 1C3 (AKR1C3) 2019 Chiara Vigato, Agnese Chiara Pippione, Sandra Kovachka, Francesca Spyrakis, Martina Daga, Simonetta Oliaro-Bosso, Marco Lucio Lolli, Donatella Boschi
Characterization of C-4 demethylation complex of cholesterol biosynthesis 2012 Brozzu Andrea; Oliaro-Bosso Simonetta; Zonari Daniele; Viola Franca; Poirier Donald; Cunningham David; Herman Gail; Jokela Heili; Poutanen Matti; Balliano Gianni
Comparative characterization of yeast and human 3-ketosteroid reductase, two moonlighting proteins that share a job 2015 Ferrante, Terenzio; Remani, Elisa; Baratta, Erica; Poirier, Donald; Balliano, Gianni; Oliaro-Bosso, Simonetta
Design, synthesis, and biological evaluation of flufenamic acid derived bioisosteres as inhibitors of aldo-keto reductase 1C3 (AKR1C3) expressed in prostate cancer 2016 Lolli, Marco; Cena, Clara; Giraudo, Alessandro; Marini, Elisabetta; Pippione, Agnese; Oliaro-Bosso, Simonetta; Ferrante, Terenzio; Sadiq, Maria; Pors, Klaus; Boschi, Donatella; Braga, Rudolpho; Andrade, Carolina.
Different interaction between oxidosqualene cyclase and steroid-3-ketoreductase from yeasts to mammals 2011 S. Taramino; B. Teske; S. Oliaro-Bosso; F. Viola; M. Bard; G. Balliano
Different Interaction between Oxidosqualene Cyclase and Steroid-3-ketoreductase in Yeast and Mammals 2010 Silvia Taramino; Brian Teske; Simonetta Oliaro-Bosso; Franca Viola; Martin Bard; Gianni Balliano
Effect of inhibiting the sterol biosynthesis pathway and the cholesterol content in the regulation of angiogenesis in vitro and in vivo 2011 Claudia Meda; Simonetta Oliaro-Bosso; Marina Visentin; Carlo Cerato; Valmira Lena; Federico Bussolino; Gianni Balliano; Franca Viola; Enrico Giraudo
Effects of new hydroxyazoles inhibitors of AKR1C3 on vitality of prostate and colorectal cancer cell lines 2019 Valentina Boscaro, Donatella Boschi, Simonetta Oliaro-Bosso, Martina Daga, Marco Lolli, Agnese Chiara Pippione, Margherita Gallicchio
Exploring the access of the substrate to the active site of yeast oxidosqualene cyclase by site-directed mutagenesis 2007 S. Oliaro-Bosso; S. Taramino; I. Ferrari; G. Ermondi; G. Caron; F. Viola; G. Balliano
Exploring the access of the substrate to the active site of yeast oxidosqualene cyclase by site-directed mutagenesis. 2007 S. Oliaro-Bosso; S. Taramino; I. Ferrari; G. Ermondi; G. Caron; F. Viola; G. Balliano
Functional characterization by site-directed mutagenesis of human oxidosqualene cyclase (OSC) expressed in Pichia pastoris 2012 Viola Franca; Balliano Gianni; Ruf Armin; Taramino Silvia; di Bartolo Giuseppe; Oliaro-Bosso Simonetta
HYDROXYLATED HETEROCYCLES AS BIOISOSTERES OF THE CARBOXYLIC FUNCTION: DESIGN OF NEW AKR1C3 INHIBITORS ACTIVE IN PROSTATE CANCER 2023 Agnese C. Pippione, Stefano Sainas, Chiara Vigato, Iole Mannella, Irene Castellino, Sandra Kovachka, Mariia Iakovleva, Barbara Rolando, Tomasz Wrobel, Osman A. Mirza, Karla Frydenvang, Francesca Spyrakis, Simonetta Oliaro-Bosso, Marco L. Lolli, Donatella Boschi
Interaction of oxidosqualene cyclase with C-4 sterol demethylation complex 2009 S. Taramino; M. Valachovic; S. Oliaro-Bosso; F. Viola; B. Teske; M. Bard; G. Balliano