Sfoglia per Autore
Application of an in house bioisosteric approach to the design of innovative inhibitors of aldo-keto reductase 1C3 (AKR1C3)
2019-01-01 Chiara Vigato, Agnese Chiara Pippione, Sandra Kovachka, Francesca Spyrakis, Martina Daga, Simonetta Oliaro-Bosso, Marco Lucio Lolli, Donatella Boschi
Application of an in house bioisosteric approach to the design of innovative inhibitors of aldo-keto reductase 1C3 (AKR1C3)
2019-01-01 Chiara Vigato, Agnese Chiara Pippione, Sandra Kovachka, Francesca Spyrakis, Martina Daga, Simonetta Oliaro Bosso, Marco Lucio Lolli, Donatella Boschi
Effects of new hydroxyazoles inhibitors of AKR1C3 on vitality of prostate and colorectal cancer cell lines
2019-01-01 Valentina Boscaro, Donatella Boschi, Simonetta Oliaro-Bosso, Martina Daga, Marco Lolli, Agnese Chiara Pippione, Margherita Gallicchio
Bioisosteres of Indomethacin as Inhibitors of Aldo-Keto Reductase 1C3
2019-01-01 Lolli, Marco L; Carnovale, Irene M; Pippione, Agnese C; Wahlgren, Weixiao Y; Bonanni, Davide; Marini, Elisabetta; Zonari, Daniele; Gallicchio, Margherita; Boscaro, Valentina; Goyal, Parveen; Friemann, Rosmarie; Rolando, Barbara; Bagnati, Renzo; Adinolfi, Salvatore; Oliaro-Bosso, Simonetta; Boschi, Donatella
Thermosensitive nanocomposite hydrogels for intravitreal delivery of cefuroxime
2019-01-01 Simona Sapino; Elena Peira; Daniela Chirio; Giulia Chindamo; Stefano Guglielmo; Simonetta Oliaro-Bosso; Raffaella Barbero; Cristina Vercelli; Giovanni Re; Valentina Brunella; Chiara Riedo; Antonio Maria Fea; Marina Gallarate
Sistemi nanocompositi termosensibili per la somministrazione intravitreale di cefuroxima
2018-01-01 BRUNO CAPRARELLI, SIMONA SAPINO, ELENA PEIRA, DANIELA CHIRIO, SUSHIL A JADHAV, SIMONETTA OLIARO BOSSO, STEFANO GUGLIELMO, RAFFAELLA BARBERO, ANTONIO MARIA FEA, CLAUDIA FRUTTERO, FRANCO DOSIO, MARINA GALLARATE
Indoor illumination: A possible pitfall in toxicological assessment of photo-active nanomaterials
2018-01-01 Marucco, Arianna; Pellegrino, Francesco; Oliaro-Bosso, Simonetta; Maurino, Valter; Martra, Gianmario; Fenoglio, Ivana
Cannabinoid Delivery Systems for Pain and Inflammation Treatment
2018-01-01 Bruni, Natascia; Della Pepa, Carlo; Oliaro-Bosso, Simonetta; Pessione, Enrica; Gastaldi, Daniela; Dosio, Franco
Potent and selective aldo-keto reductase 1C3 (AKR1C3) inhibitors based on the benzoisoxazole moiety: Application of a bioisosteric scaffold hopping approach to flufenamic acid
2018-01-01 Pippione, Agnese Chiara; Carnovale, Irene Maria; Bonanni, Davide; Sini, Marcella; Goyal, Parveen; Marini, Elisabetta; Pors, Klaus; Adinolfi, Salvatore; Zonari, Daniele; Festuccia, Claudio; Wahlgren, Weixiao Yuan; Friemann, Rosmarie; Bagnati, Renzo; Boschi, Donatella; Oliaro-Bosso, Simonetta; Lolli, Marco Lucio
Androgen-AR axis in primary and metastatic prostate cancer: chasing steroidogenic enzymes for therapeutic intervention
2017-01-01 Pippione, Agnese C.; Boschi, Donatella; Pors, Klaus; Oliaro-Bosso, Simonetta; Lolli, Marco L.
Hydroxytriazole derivatives as potent and selective aldo-keto reductase 1C3 (AKR1C3) inhibitors discovered by bioisosteric scaffold hopping approach
2017-01-01 Pippione, Agnese C.; Giraudo, Alessandro; Bonanni, Davide; Carnovale, Irene M.; Marini, Elisabetta; Cena, Clara; Costale, Annalisa; Zonari, Daniele; Pors, Klaus; Sadiq, Maria; Boschi, Donatella; Oliaro-Bosso, Simonetta; Lolli, Marco L
Mesoporous silica nanoparticles as a promising skin delivery system for methotrexate
2017-01-01 Sapino, Simona; Oliaro-Bosso, Simonetta; Zonari, Daniele; Zattoni, Andrea; Ugazio, Elena
Design, synthesis, and biological evaluation of flufenamic acid derived bioisosteres as inhibitors of aldo-keto reductase 1C3 (AKR1C3) expressed in prostate cancer
2016-01-01 Lolli, Marco; Cena, Clara; Giraudo, Alessandro; Marini, Elisabetta; Pippione, Agnese; Oliaro-Bosso, Simonetta; Ferrante, Terenzio; Sadiq, Maria; Pors, Klaus; Boschi, Donatella; Braga, Rudolpho; Andrade, Carolina.
NEW HYDROXYAZOLES INHIBITORS OF AKR1C3 OBTAINED FROM NSAIDS BY SCAFFOLD HOPPING APPROACH AGAINST CASTRATE RESISTANT PROSTATE CANCER
2016-01-01 Boschi, Donatella; Pippione, Agnese Chiara; Giraudo, Alessandro; Carnovale, Irene Maria; Zorniotti, Sonia; Oliaro-Bosso, Simonetta; Ferrante, Terenzio; Marini, Elisabetta; Pors, Klaus; Festuccia, Claudio; Monache, Simona Delle; Zaffaroni, Nadia; Braga, Rodolpho Campos; Lucio Lolli, Marco
NEW HYDROXYAZOLES INHIBITORS OF ALDO-KETO REDUCTASE 1C3 (AKR1C3) OBTAINED BY SCAFFOLD HOPPING FROM FLUFENAMIC ACID AND INDOMETHACIN FOR CASTRATE RESISTANT PROSTATE CANCER
2016-01-01 Boschi, Donatella; Pippione, Agnese Chiara; Giraudo, Alessandro; Carnovale, Irene Maria; Zorniotti, Sonia; Oliaro-Bosso, Simonetta; Ferrante, Terenzio; Marini, Elisabetta; Pors, Klaus; Festuccia, Claudio; Monache, Simona Delle; Zaffaroni, Nadia; Braga, Rodolpho Campos; Lucio, Marco; Lolli,
Targeting Castration Resistant Prostate Cancer (CRPC) by innovative AKR1C3 inhibitors based on the 3-hydroxybenzoisoxazole structure
2016-01-01 Carnovale, Irene Maria; Pippione, Agnese Chiara; Giraudo, Alessandro; Federico, Antonella; Zorniotti, Sonia; Simonetta Oliaro Bosso, ; Ferrante, Terenzio; Marini, Elisabetta; Pors, Klaus; Braga, Rodolpho Campos; Boschi, Donatella; Lucio Lolli, Marco
4-Methylzymosterone and Other Intermediates of Sterol Biosynthesis from Yeast Mutants Engineered in the ERG27 Gene Encoding 3-Ketosteroid Reductase
2016-01-01 Ferrante, T; Barge, A; Taramino, S; Oliaro-Bosso, S; Balliano, G
Difference in the late ergosterol biosynthesis between yeast spheroplasts and intact cells
2016-01-01 Ferrante, T; Viola, F; Balliano, G; Oliaro-Bosso, S
Thermoresponsive mesoporous silica nanoparticles as a carrier for skin delivery of quercetin
2016-01-01 Ugazio, Elena; Gastaldi, Lucia; Brunella, Valentina; Scalarone, Dominique; Jadhav, Sushilkumar A.; Oliaro-Bosso, Simonetta; Zonari, Daniele; Berlier, Gloria; Miletto, Ivana; Sapino, Simona
Arylpiperidines as a new class of oxidosqualene cyclase inhibitors
2016-01-01 Keller, M.; Wolfgardt, A.; Müller, C.; Wilcken, R.; Böckler, F.M.; Oliaro-Bosso, S.; Ferrante, T.; Balliano, G.; Bracher, F.
| Titolo | Data di pubblicazione | Autore(i) | File |
|---|---|---|---|
| Application of an in house bioisosteric approach to the design of innovative inhibitors of aldo-keto reductase 1C3 (AKR1C3) | 2019 | Chiara Vigato, Agnese Chiara Pippione, Sandra Kovachka, Francesca Spyrakis, Martina Daga, Simonetta Oliaro-Bosso, Marco Lucio Lolli, Donatella Boschi | |
| Application of an in house bioisosteric approach to the design of innovative inhibitors of aldo-keto reductase 1C3 (AKR1C3) | 2019 | Chiara Vigato, Agnese Chiara Pippione, Sandra Kovachka, Francesca Spyrakis, Martina Daga, Simonetta Oliaro Bosso, Marco Lucio Lolli, Donatella Boschi | |
| Effects of new hydroxyazoles inhibitors of AKR1C3 on vitality of prostate and colorectal cancer cell lines | 2019 | Valentina Boscaro, Donatella Boschi, Simonetta Oliaro-Bosso, Martina Daga, Marco Lolli, Agnese Chiara Pippione, Margherita Gallicchio | |
| Bioisosteres of Indomethacin as Inhibitors of Aldo-Keto Reductase 1C3 | 2019 | Lolli, Marco L; Carnovale, Irene M; Pippione, Agnese C; Wahlgren, Weixiao Y; Bonanni, Davide; Marini, Elisabetta; Zonari, Daniele; Gallicchio, Margherita; Boscaro, Valentina; Goyal, Parveen; Friemann, Rosmarie; Rolando, Barbara; Bagnati, Renzo; Adinolfi, Salvatore; Oliaro-Bosso, Simonetta; Boschi, Donatella | |
| Thermosensitive nanocomposite hydrogels for intravitreal delivery of cefuroxime | 2019 | Simona Sapino; Elena Peira; Daniela Chirio; Giulia Chindamo; Stefano Guglielmo; Simonetta Oliaro-Bosso; Raffaella Barbero; Cristina Vercelli; Giovanni Re; Valentina Brunella; Chiara Riedo; Antonio Maria Fea; Marina Gallarate | |
| Sistemi nanocompositi termosensibili per la somministrazione intravitreale di cefuroxima | 2018 | BRUNO CAPRARELLI, SIMONA SAPINO, ELENA PEIRA, DANIELA CHIRIO, SUSHIL A JADHAV, SIMONETTA OLIARO BOSSO, STEFANO GUGLIELMO, RAFFAELLA BARBERO, ANTONIO MARIA FEA, CLAUDIA FRUTTERO, FRANCO DOSIO, MARINA GALLARATE | |
| Indoor illumination: A possible pitfall in toxicological assessment of photo-active nanomaterials | 2018 | Marucco, Arianna; Pellegrino, Francesco; Oliaro-Bosso, Simonetta; Maurino, Valter; Martra, Gianmario; Fenoglio, Ivana | |
| Cannabinoid Delivery Systems for Pain and Inflammation Treatment | 2018 | Bruni, Natascia; Della Pepa, Carlo; Oliaro-Bosso, Simonetta; Pessione, Enrica; Gastaldi, Daniela; Dosio, Franco | |
| Potent and selective aldo-keto reductase 1C3 (AKR1C3) inhibitors based on the benzoisoxazole moiety: Application of a bioisosteric scaffold hopping approach to flufenamic acid | 2018 | Pippione, Agnese Chiara; Carnovale, Irene Maria; Bonanni, Davide; Sini, Marcella; Goyal, Parveen; Marini, Elisabetta; Pors, Klaus; Adinolfi, Salvatore; Zonari, Daniele; Festuccia, Claudio; Wahlgren, Weixiao Yuan; Friemann, Rosmarie; Bagnati, Renzo; Boschi, Donatella; Oliaro-Bosso, Simonetta; Lolli, Marco Lucio | |
| Androgen-AR axis in primary and metastatic prostate cancer: chasing steroidogenic enzymes for therapeutic intervention | 2017 | Pippione, Agnese C.; Boschi, Donatella; Pors, Klaus; Oliaro-Bosso, Simonetta; Lolli, Marco L. | |
| Hydroxytriazole derivatives as potent and selective aldo-keto reductase 1C3 (AKR1C3) inhibitors discovered by bioisosteric scaffold hopping approach | 2017 | Pippione, Agnese C.; Giraudo, Alessandro; Bonanni, Davide; Carnovale, Irene M.; Marini, Elisabetta; Cena, Clara; Costale, Annalisa; Zonari, Daniele; Pors, Klaus; Sadiq, Maria; Boschi, Donatella; Oliaro-Bosso, Simonetta; Lolli, Marco L | |
| Mesoporous silica nanoparticles as a promising skin delivery system for methotrexate | 2017 | Sapino, Simona; Oliaro-Bosso, Simonetta; Zonari, Daniele; Zattoni, Andrea; Ugazio, Elena | |
| Design, synthesis, and biological evaluation of flufenamic acid derived bioisosteres as inhibitors of aldo-keto reductase 1C3 (AKR1C3) expressed in prostate cancer | 2016 | Lolli, Marco; Cena, Clara; Giraudo, Alessandro; Marini, Elisabetta; Pippione, Agnese; Oliaro-Bosso, Simonetta; Ferrante, Terenzio; Sadiq, Maria; Pors, Klaus; Boschi, Donatella; Braga, Rudolpho; Andrade, Carolina. | |
| NEW HYDROXYAZOLES INHIBITORS OF AKR1C3 OBTAINED FROM NSAIDS BY SCAFFOLD HOPPING APPROACH AGAINST CASTRATE RESISTANT PROSTATE CANCER | 2016 | Boschi, Donatella; Pippione, Agnese Chiara; Giraudo, Alessandro; Carnovale, Irene Maria; Zorniotti, Sonia; Oliaro-Bosso, Simonetta; Ferrante, Terenzio; Marini, Elisabetta; Pors, Klaus; Festuccia, Claudio; Monache, Simona Delle; Zaffaroni, Nadia; Braga, Rodolpho Campos; Lucio Lolli, Marco | |
| NEW HYDROXYAZOLES INHIBITORS OF ALDO-KETO REDUCTASE 1C3 (AKR1C3) OBTAINED BY SCAFFOLD HOPPING FROM FLUFENAMIC ACID AND INDOMETHACIN FOR CASTRATE RESISTANT PROSTATE CANCER | 2016 | Boschi, Donatella; Pippione, Agnese Chiara; Giraudo, Alessandro; Carnovale, Irene Maria; Zorniotti, Sonia; Oliaro-Bosso, Simonetta; Ferrante, Terenzio; Marini, Elisabetta; Pors, Klaus; Festuccia, Claudio; Monache, Simona Delle; Zaffaroni, Nadia; Braga, Rodolpho Campos; Lucio, Marco; Lolli, | |
| Targeting Castration Resistant Prostate Cancer (CRPC) by innovative AKR1C3 inhibitors based on the 3-hydroxybenzoisoxazole structure | 2016 | Carnovale, Irene Maria; Pippione, Agnese Chiara; Giraudo, Alessandro; Federico, Antonella; Zorniotti, Sonia; Simonetta Oliaro Bosso, ; Ferrante, Terenzio; Marini, Elisabetta; Pors, Klaus; Braga, Rodolpho Campos; Boschi, Donatella; Lucio Lolli, Marco | |
| 4-Methylzymosterone and Other Intermediates of Sterol Biosynthesis from Yeast Mutants Engineered in the ERG27 Gene Encoding 3-Ketosteroid Reductase | 2016 | Ferrante, T; Barge, A; Taramino, S; Oliaro-Bosso, S; Balliano, G | |
| Difference in the late ergosterol biosynthesis between yeast spheroplasts and intact cells | 2016 | Ferrante, T; Viola, F; Balliano, G; Oliaro-Bosso, S | |
| Thermoresponsive mesoporous silica nanoparticles as a carrier for skin delivery of quercetin | 2016 | Ugazio, Elena; Gastaldi, Lucia; Brunella, Valentina; Scalarone, Dominique; Jadhav, Sushilkumar A.; Oliaro-Bosso, Simonetta; Zonari, Daniele; Berlier, Gloria; Miletto, Ivana; Sapino, Simona | |
| Arylpiperidines as a new class of oxidosqualene cyclase inhibitors | 2016 | Keller, M.; Wolfgardt, A.; Müller, C.; Wilcken, R.; Böckler, F.M.; Oliaro-Bosso, S.; Ferrante, T.; Balliano, G.; Bracher, F. |
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