Sfoglia per Autore
SangsterLogP - the largest publicly available dataset of logP values
2026-01-01 Cirino, Thalita; Caron, Giulia; Ermondi, Giuseppe; Charochkina, Larysa; Tetko, Igor V.
BBB-Permeable PROTACs: Where Do We Stand?
2026-01-01 Francisco, Serena; Apprato, Giulia; Rossi Sebastiano, Matteo; Ermondi, Giuseppe; Caron, Giulia
Smart Integration of Structural Biology and Medicinal Chemistry to Unlock Target‐Driven Drug Discovery
2026-01-01 Rossi Sebastiano, Matteo; Apprato, Giulia; Francisco, Serena; Ermondi, Giuseppe; Caron, Giulia
MK4 Repositioning for IAHSP: Overcoming In Vivo Data Gaps through In Silico Refinement and In Vitro Validation
2026-01-01 Rossi Sebastiano, Matteo; Vicidomini, Antonio; Francisco, Serena; Pullano, Verdiana; Defilippi, Paola; Baj, Gabriele; Cesca, Fabrizia; Caron, Giulia; Ermondi, Giuseppe
Restoring adapter protein complex 4 function with small molecules: an in silico approach to spastic paraplegia 50
2025-01-01 Francisco, Serena; Lamacchia, Lorenzo; Turco, Attilio; Ermondi, Giuseppe; Caron, Giulia; Rossi Sebastiano, Matteo
Linker Methylation as a Strategy to Enhance PROTAC Oral Bioavailability: Insights from Molecular Properties and Conformational Analysis
2025-01-01 Garcia Jimenez, Diego; Ermondi, Giuseppe; Jandova, Zuzana; Vallaro, Maura; Caron, Giulia; Arnhof, Heribert
Macrocyclization: Enhancing Drug-like Properties of Discoidin Domain Receptor Kinase Inhibitors
2025-01-01 Carzaniga, Laura; Mazzucato, Roberta; Mileo, Valentina; Rizzi, Andrea; Vallaro, Maura; Ermondi, Giuseppe; Cattani, Silvia; Secchi, Andrea; Caron, Giulia
Exploring the chemical space of orally bioavailable PROTACs
2024-01-01 Apprato G.; Poongavanam V.; Garcia Jimenez D.; Atilaw Y.; Erdelyi M.; Ermondi G.; Caron G.; Kihlberg J.
Molecular properties, including chameleonicity, as essential tools for designing the next generation of oral beyond rule of five drugs
2024-01-01 GARCÍA JIMÉNEZ D.; Vallaro M.; Vitagliano L.; Lopez L.L.; Apprato G.; Ermondi G.; Caron G.
IMHB-Mediated Chameleonicity in Drug Design: A Focus on Structurally Related PROTACs
2024-01-01 Diego Garcia Jimenez; Matteo Rossi Sebastiano; Maura Vallaro; Giuseppe Ermondi; Giulia Caron
DegraderTCM: A Computationally Sparing Approach for Predicting Ternary Degradation Complexes
2024-01-01 Rossetti P.; Apprato G.; Caron G.; Ermondi G.; Rossi Sebastiano M.
Preclinical alternative drug discovery programs for monogenic rare diseases. Should small molecules or gene therapy be used? The case of hereditary spastic paraplegias
2024-01-01 Rossi Sebastiano, Matteo; Hadano, Shinji; Cesca, Fabrizia; Ermondi, Giuseppe; Caron, Giulia; Francisco, Serena; Brusco, Alfredo; Pullano, Verdiana; Chiantia, Giuseppe; Giustetto, Maurizio ; Baj, Gabriele; Della Vecchia, Stefania; Lamacchia, Lorenzo; Russo, Silvia; Higgins, Anna J.; van Putte, Wouter; Gurgone, Antonia
High-throughput and reliable assessments of the ionization constant of monoprotic organic acids through an arginine based mixed mode HPLC
2023-01-01 Russo G.; Kajtazi A.; Vallaro M.; Surmont P.; Ermondi G.; Anderson S.; Grumetto L.; Caron G.; Lynen F.
Ionization and lipophilicity in nonpolar media mimicking the cell membrane interior
2023-01-01 Vallaro, Maura; Ermondi, Giuseppe; Saame, Jaan; Leito, Ivo; Caron, Giulia
In Silico Tools to Extract the Drug Design Information Content of Degradation Data: The Case of PROTACs Targeting the Androgen Receptor
2023-01-01 Apprato Giulia; D’Agostini Giulia; Rossetti Paolo; Ermondi Giuseppe; Caron Giulia
Chamelogk: A Chromatographic Chameleonicity Quantifier to Design Orally Bioavailable Beyond-Rule-of-5 Drugs
2023-01-01 GARCÍA JIMÉNEZ DIEGO; Vallaro Maura; Rossi Sebastiano Matteo; Apprato Giulia; D'Agostini Giulia; Rossetti Paolo; Ermondi Giuseppe; Caron Giulia
Deleterious, protein-altering variants in the transcriptional coregulator ZMYM3 in 27 individuals with a neurodevelopmental delay phenotype
2023-01-01 Hiatt, Susan M; Trajkova, Slavica; Sebastiano, Matteo Rossi; Partridge, E Christopher; Abidi, Fatima E; Anderson, Ashlyn; Ansar, Muhammad; Antonarakis, Stylianos E; Azadi, Azadeh; Bachmann-Gagescu, Ruxandra; Bartuli, Andrea; Benech, Caroline; Berkowitz, Jennifer L; Betti, Michael J; Brusco, Alfredo; Cannon, Ashley; Caron, Giulia; Chen, Yanmin; Cochran, Meagan E; Coleman, Tanner F; Crenshaw, Molly M; Cuisset, Laurence; Curry, Cynthia J; Darvish, Hossein; Demirdas, Serwet; Descartes, Maria; Douglas, Jessica; Dyment, David A; Elloumi, Houda Zghal; Ermondi, Giuseppe; Faoucher, Marie; Farrow, Emily G; Felker, Stephanie A; Fisher, Heather; Hurst, Anna C E; Joset, Pascal; Kelly, Melissa A; Kmoch, Stanislav; Leadem, Benjamin R; Lyons, Michael J; Macchiaiolo, Marina; Magner, Martin; Mandrile, Giorgia; Mattioli, Francesca; McEown, Megan; Meadows, Sarah K; Medne, Livija; Meeks, Naomi J L; Montgomery, Sarah; Napier, Melanie P; Natowicz, Marvin; Newberry, Kimberly M; Niceta, Marcello; Noskova, Lenka; Nowak, Catherine B; Noyes, Amanda G; Osmond, Matthew; Prijoles, Eloise J; Pugh, Jada; Pullano, Verdiana; Quélin, Chloé; Rahimi-Aliabadi, Simin; Rauch, Anita; Redon, Sylvia; Reymond, Alexandre; Schwager, Caitlin R; Sellars, Elizabeth A; Scheuerle, Angela E; Shukarova-Angelovska, Elena; Skraban, Cara; Stolerman, Elliot; Sullivan, Bonnie R; Tartaglia, Marco; Thiffault, Isabelle; Uguen, Kevin; Umaña, Luis A; van Bever, Yolande; van der Crabben, Saskia N; van Slegtenhorst, Marjon A; Waisfisz, Quinten; Washington, Camerun; Rodan, Lance H; Myers, Richard M; Cooper, Gregory M
Conformational Sampling Deciphers the Chameleonic Properties of a VHL-Based Degrader
2023-01-01 Ermondi, Giuseppe; Jimenez, Diego Garcia; Rossi Sebastiano, Matteo; Kihlberg, Jan; Caron, Giulia
The Quest for Oral PROTAC drugs: Evaluating the Weaknesses of the Screening Pipeline
2023-01-01 Apprato, Giulia; Ermondi, Giuseppe; Caron, Giulia
Personalized Treatment for Infantile Ascending Hereditary Spastic Paralysis Based on In Silico Strategies
2022-01-01 Rossi Sebastiano, Matteo; Ermondi, Giuseppe; Sato, Kai; Otomo, Asako; Hadano, Shinji; Caron, Giulia
| Titolo | Data di pubblicazione | Autore(i) | File |
|---|---|---|---|
| SangsterLogP - the largest publicly available dataset of logP values | 2026 | Cirino, Thalita; Caron, Giulia; Ermondi, Giuseppe; Charochkina, Larysa; Tetko, Igor V. | |
| BBB-Permeable PROTACs: Where Do We Stand? | 2026 | Francisco, Serena; Apprato, Giulia; Rossi Sebastiano, Matteo; Ermondi, Giuseppe; Caron, Giulia | |
| Smart Integration of Structural Biology and Medicinal Chemistry to Unlock Target‐Driven Drug Discovery | 2026 | Rossi Sebastiano, Matteo; Apprato, Giulia; Francisco, Serena; Ermondi, Giuseppe; Caron, Giulia | |
| MK4 Repositioning for IAHSP: Overcoming In Vivo Data Gaps through In Silico Refinement and In Vitro Validation | 2026 | Rossi Sebastiano, Matteo; Vicidomini, Antonio; Francisco, Serena; Pullano, Verdiana; Defilippi, Paola; Baj, Gabriele; Cesca, Fabrizia; Caron, Giulia; Ermondi, Giuseppe | |
| Restoring adapter protein complex 4 function with small molecules: an in silico approach to spastic paraplegia 50 | 2025 | Francisco, Serena; Lamacchia, Lorenzo; Turco, Attilio; Ermondi, Giuseppe; Caron, Giulia; Rossi Sebastiano, Matteo | |
| Linker Methylation as a Strategy to Enhance PROTAC Oral Bioavailability: Insights from Molecular Properties and Conformational Analysis | 2025 | Garcia Jimenez, Diego; Ermondi, Giuseppe; Jandova, Zuzana; Vallaro, Maura; Caron, Giulia; Arnhof, Heribert | |
| Macrocyclization: Enhancing Drug-like Properties of Discoidin Domain Receptor Kinase Inhibitors | 2025 | Carzaniga, Laura; Mazzucato, Roberta; Mileo, Valentina; Rizzi, Andrea; Vallaro, Maura; Ermondi, Giuseppe; Cattani, Silvia; Secchi, Andrea; Caron, Giulia | |
| Exploring the chemical space of orally bioavailable PROTACs | 2024 | Apprato G.; Poongavanam V.; Garcia Jimenez D.; Atilaw Y.; Erdelyi M.; Ermondi G.; Caron G.; Kihlberg J. | |
| Molecular properties, including chameleonicity, as essential tools for designing the next generation of oral beyond rule of five drugs | 2024 | GARCÍA JIMÉNEZ D.; Vallaro M.; Vitagliano L.; Lopez L.L.; Apprato G.; Ermondi G.; Caron G. | |
| IMHB-Mediated Chameleonicity in Drug Design: A Focus on Structurally Related PROTACs | 2024 | Diego Garcia Jimenez; Matteo Rossi Sebastiano; Maura Vallaro; Giuseppe Ermondi; Giulia Caron | |
| DegraderTCM: A Computationally Sparing Approach for Predicting Ternary Degradation Complexes | 2024 | Rossetti P.; Apprato G.; Caron G.; Ermondi G.; Rossi Sebastiano M. | |
| Preclinical alternative drug discovery programs for monogenic rare diseases. Should small molecules or gene therapy be used? The case of hereditary spastic paraplegias | 2024 | Rossi Sebastiano, Matteo; Hadano, Shinji; Cesca, Fabrizia; Ermondi, Giuseppe; Caron, Giulia; Francisco, Serena; Brusco, Alfredo; Pullano, Verdiana; Chiantia, Giuseppe; Giustetto, Maurizio ; Baj, Gabriele; Della Vecchia, Stefania; Lamacchia, Lorenzo; Russo, Silvia; Higgins, Anna J.; van Putte, Wouter; Gurgone, Antonia | |
| High-throughput and reliable assessments of the ionization constant of monoprotic organic acids through an arginine based mixed mode HPLC | 2023 | Russo G.; Kajtazi A.; Vallaro M.; Surmont P.; Ermondi G.; Anderson S.; Grumetto L.; Caron G.; Lynen F. | |
| Ionization and lipophilicity in nonpolar media mimicking the cell membrane interior | 2023 | Vallaro, Maura; Ermondi, Giuseppe; Saame, Jaan; Leito, Ivo; Caron, Giulia | |
| In Silico Tools to Extract the Drug Design Information Content of Degradation Data: The Case of PROTACs Targeting the Androgen Receptor | 2023 | Apprato Giulia; D’Agostini Giulia; Rossetti Paolo; Ermondi Giuseppe; Caron Giulia | |
| Chamelogk: A Chromatographic Chameleonicity Quantifier to Design Orally Bioavailable Beyond-Rule-of-5 Drugs | 2023 | GARCÍA JIMÉNEZ DIEGO; Vallaro Maura; Rossi Sebastiano Matteo; Apprato Giulia; D'Agostini Giulia; Rossetti Paolo; Ermondi Giuseppe; Caron Giulia | |
| Deleterious, protein-altering variants in the transcriptional coregulator ZMYM3 in 27 individuals with a neurodevelopmental delay phenotype | 2023 | Hiatt, Susan M; Trajkova, Slavica; Sebastiano, Matteo Rossi; Partridge, E Christopher; Abidi, Fatima E; Anderson, Ashlyn; Ansar, Muhammad; Antonarakis, Stylianos E; Azadi, Azadeh; Bachmann-Gagescu, Ruxandra; Bartuli, Andrea; Benech, Caroline; Berkowitz, Jennifer L; Betti, Michael J; Brusco, Alfredo; Cannon, Ashley; Caron, Giulia; Chen, Yanmin; Cochran, Meagan E; Coleman, Tanner F; Crenshaw, Molly M; Cuisset, Laurence; Curry, Cynthia J; Darvish, Hossein; Demirdas, Serwet; Descartes, Maria; Douglas, Jessica; Dyment, David A; Elloumi, Houda Zghal; Ermondi, Giuseppe; Faoucher, Marie; Farrow, Emily G; Felker, Stephanie A; Fisher, Heather; Hurst, Anna C E; Joset, Pascal; Kelly, Melissa A; Kmoch, Stanislav; Leadem, Benjamin R; Lyons, Michael J; Macchiaiolo, Marina; Magner, Martin; Mandrile, Giorgia; Mattioli, Francesca; McEown, Megan; Meadows, Sarah K; Medne, Livija; Meeks, Naomi J L; Montgomery, Sarah; Napier, Melanie P; Natowicz, Marvin; Newberry, Kimberly M; Niceta, Marcello; Noskova, Lenka; Nowak, Catherine B; Noyes, Amanda G; Osmond, Matthew; Prijoles, Eloise J; Pugh, Jada; Pullano, Verdiana; Quélin, Chloé; Rahimi-Aliabadi, Simin; Rauch, Anita; Redon, Sylvia; Reymond, Alexandre; Schwager, Caitlin R; Sellars, Elizabeth A; Scheuerle, Angela E; Shukarova-Angelovska, Elena; Skraban, Cara; Stolerman, Elliot; Sullivan, Bonnie R; Tartaglia, Marco; Thiffault, Isabelle; Uguen, Kevin; Umaña, Luis A; van Bever, Yolande; van der Crabben, Saskia N; van Slegtenhorst, Marjon A; Waisfisz, Quinten; Washington, Camerun; Rodan, Lance H; Myers, Richard M; Cooper, Gregory M | |
| Conformational Sampling Deciphers the Chameleonic Properties of a VHL-Based Degrader | 2023 | Ermondi, Giuseppe; Jimenez, Diego Garcia; Rossi Sebastiano, Matteo; Kihlberg, Jan; Caron, Giulia | |
| The Quest for Oral PROTAC drugs: Evaluating the Weaknesses of the Screening Pipeline | 2023 | Apprato, Giulia; Ermondi, Giuseppe; Caron, Giulia | |
| Personalized Treatment for Infantile Ascending Hereditary Spastic Paralysis Based on In Silico Strategies | 2022 | Rossi Sebastiano, Matteo; Ermondi, Giuseppe; Sato, Kai; Otomo, Asako; Hadano, Shinji; Caron, Giulia |
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