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Prodotti della tipologia (ordinati per Data di deposito in Decrescente ordine): 1 a 20 di 1.691
Titolo | Data di deposito | Autore(i) |
---|---|---|
Targeting PAD-mediated citrullination to treat human papillomavirus infections | 20-apr-2022 | CAMILLA ALBANO, MATTEO BIOLATTI, SELINA PASQUERO, FRANCESCA GUGLIESI, SERGIO F. CASTILLO PACHECO, GLORIA GRIFFANTE, ELENA CAT GENOVA, IRENE LO CIGNO, MARISA GARIGLIO, MARCO DE ANDREA, SANTO LANDOLFO, JASENKA MAZIBRADA, VALENTINA DELL’OSTE |
Targeting myeloid leukemias using human Dihydroorotate Dehydrogenase inhibitors based on 2-hydroxypyrazolo[1,5-a]pyridine scaffold: overcoming of metabolic issues | 9-apr-2022 | Chiara Vigato, Stefano Sainas, Marta Giorgis, Paola Circosta, Alice Passoni, Agnese Chiara Pippione, Renzo Bagnati, Giuseppe Saglio, Donatella Boschi, Marco Lucio Lolli. |
A new pro-apoptotic therapy for Acute Myeloid Leukaemia using MEDS433, a potent human Dihydroorotate Dehydrogenase inhibitor | 9-apr-2022 | Sainas Sainas, Paola Circosta, Noemi Villella, Elena Martino, Agnese Chiara Pippione, Mohammad Houshmand, Marta Giorgis, Valentina Gaidano, Alessandro Cignetti, Caterina Peraldo Neia, Giovanna Chiorino, Salam Al-Karadaghi, Donatella Boschi, Giuseppe Saglio, Marco Lucio Lolli. |
A differentiating and apoptotic therapy for Acute Myeloid Leukaemia using MEDS433, a potent human Dihydroorotate Dehydrogenase inhibitor | 9-apr-2022 | Stefano Sainas, Paola Circosta, Marta Giorgis, Agnese Chiara Pippione, Marilena Marraudino, Mohammad Houshmand, Brigitta Bonaldo, Valentina Gaidano, Alessandro Cignetti, Stefano Gotti, Giuseppe Saglio, Salam Al-Karadaghi, Donatella Boschi, Marco Lucio Lolli |
Design and synthesis of a library of pyrazolo[1,5-a]pyridine fluorophores for developing new fluorescent probes | 9-apr-2022 | Elena Martino, Stefano Sainas, Francesco Bavo, Claudio Garino, Donatella Boschi, Bente Frølund, Marco Lucio Lolli |
Multiple-targeting ligands for AKR1C3 enzyme and androgen receptor to target prostate cancer | 4-apr-2022 | Agnese Chiara Pippione, Zuhal Kilic-Kurt, Stefano Sainas, Iole Mannella, Barbara Rolando, Sandra Kovachka, Francesca Spyrakis, Annamaria Buschini, Serena Montalbano, Simonetta Oliaro Bosso, Marco Lolli, Donatella Boschi |
Improvement of metabolic weakness of new human Dihydroorotate Dehydrogenase inhibitors based on 2-hydroxypyrazolo[1,5-a]pyridine scaffold | 4-apr-2022 | Chiara Vigato, Stefano Sainas, Marta Giorgis, Paola Circosta, Alice Passoni, Agnese Chiara Pippione, Renzo Bagnati, Giuseppe Saglio, Donatella Boschi, Marco Lucio Lolli |
Design of new human Dihydroorotate Dehydrogenase inhibitors: amide bioisosterism in MEDS433 optimization | 4-apr-2022 | Martino, Elena; Villella, Noemi;Vigato, Chiara; Cerrina, Matteo; Bersani, Matteo; Giorgis Marta, Sainas, Stefano.; Boschi, Donatella; Lolli, Marco Lucio |
New inhibitors of Aldo-Keto Reductase 1C3 (AKR1C3) based on benzoisoxazole scaffold and their potential application in cancer | 4-apr-2022 | Mannella, Iole, Vigato, Chiara, Pasha, Rabia; Pippione Agnese Chiara, Sainas, Stefano, Oliaro Bosso Simonetta; Rolando, Barbara; Kovachka, Sandra, Spyrakis, Francesca; Boschi, Donatella, Lolli. Marco Lucio |
Synthesis of [18F]Brequinar as PET Imaging probes for human dihydroorotate dehydrogenase | 3-apr-2022 | Elena Martino, Stefano Sainas, Agnese C. Pippione, Donatella Boschi, Yu- Shin Ding, Marco L. Lolli |
Preliminary ADME/PK studies of new hDHODH inhibitors effective for treatment of acute myeloid leukaemia (AML) | 3-apr-2022 | Giulia De Simone, Stefano Sainas, Marilena Marraudino, Agnese Chiara Pippione, Brigitta Bonaldo, Alice Passoni, Marta Giorgis, Barbara Rolando, Donatella Boschi, Marco Lucio Lolli |
Design, synthesis and co-crystallization of new Plasmodium falciparum dihydroorotate dehydrogenase inhibitors based on hydroxypyrazole scaffold | 3-apr-2022 | Noemi Villella, Agnese Chiara Pippione, Stefano Sainas, Donatella Boschi, Rosmarie Friemann, Alberto Gimenéz, Efrain Salamanca, Marco Lucio Lolli |
Targeting the human Dihydroorotate Dehydrogenase (hDHODH) by a Scaffold Hopping Bioisosteric approach using Hydroxylated Pentatomic Heterocycles | 3-apr-2022 | Stefano Sainas, Agnese Chiara Pippione, Irene Maria Carnovale, Alessandro Giraudo, Marta Giorgis, Rodolpho B. Braga, Carolina H. Andrade, Noemi Villella, Marco Piccinini, Elisa Lupino, Rosmarie Friemann, Salam Al-Kadaraghi, Donatella Boschi, Marco L. Lolli |
Antileishmanial activity of some 4-phenyl-3-amino-1H-pyrazols designed as CRK3 kinase inhibitors | 3-apr-2022 | Agnese Chiara Pippione, Piermichele Kobauri, Stefano Sainas, Alberto Gimenez, Antonella Federico, Rodolpho Campos Braga, Carolina Horta Andrade, Donatella Boschi, Efrain Salamanca, Juan Carlos Ticona, Marco Lucio Lolli |
Toward a Bioisosteric Alkahest: Targeting the human Dihydroorotate Dehydrogenase (hDHODH) by a Scaffold Hopping Bioisosteric approach using Hydroxylated Pentatomic Heterocycles | 3-apr-2022 | Marco L. Lolli, Agnese Chiara Pippione, Stefano Sainas, Stefano Mensa, Marta Giorgis, Marco Piccinini, Elisa Lupino, Salam Al-Kadaraghi, Donatella Boschi |
Fatal Asphyxia by Bolus in Elders With Mental Illness: The Role of Oral Health and Antimuscarinic Action of Drug Treatment | 13-mar-2022 | Aquila I; Di Nunzio C; Nuzzolese E; Ricci P |
The impact of Workshop in Forensic Odontology in Human Rights Workshop in the United Arab Emirates | 12-mar-2022 | Salem Altalie, Emilio Nuzzolese, Joe Adserias-Garriga, Alexander S. Forrest, |
Dental Injuries During General Anesthesia: Risk Management and Forensic Perspectives | 12-mar-2022 | Emilio Nuzzolese, Giulio Rosboch, Fabio Innocenzi, D. Santovito, F. Lupariello |
Digital-storytelling in health context: innovative approaches to improve patients and caregivers' therapeutic literacy and adherence | 28-feb-2022 | Sabrina Grigolo; Manuela Repetto; Melania Talarico; Simona Tirocchi; Sara Croce; Clara Cena; Lisa Iannacci-Manasia; Barbara Bruschi |
The end-moraine system of the Pleistocene Moletta Glacier (Susa Valley, NW Italy) | 24-feb-2022 | Cretì E., Gianotti F. |
Prodotti della tipologia (ordinati per Data di deposito in Decrescente ordine): 1 a 20 di 1.691
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